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Found 217 with Last Name = 'fukami' and Initial = 'h'
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227831(CHEMBL52242)
Affinity DataKi:  1.20nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227791(CHEMBL53815)
Affinity DataKi:  4.60nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227978(CHEMBL53316)
Affinity DataKi:  6.30nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50228190(CHEMBL54263)
Affinity DataKi:  9.80nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227787(CHEMBL1743933)
Affinity DataKi:  13nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227837(CHEMBL52131)
Affinity DataKi:  14nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50093789(CHEMBL541829 | Succinic acid mono-(2-dimethylamino...)
Affinity DataKi:  18nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227788(CHEMBL1743936)
Affinity DataKi:  23nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227974(CHEMBL298554)
Affinity DataKi:  26nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227976(CHEMBL299389)
Affinity DataKi:  38nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227653(CHEMBL299207)
Affinity DataKi:  41nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227977(CHEMBL300631)
Affinity DataKi:  68nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227790(CHEMBL53344)
Affinity DataKi:  71nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227789(CHEMBL412653)
Affinity DataKi:  75nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227832(CHEMBL54101)
Affinity DataKi:  198nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50228189(CHEMBL52710)
Affinity DataKi:  416nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50228052(CHEMBL52982)
Affinity DataKi:  517nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227831(CHEMBL52242)
Affinity DataIC50:  13nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50210107(7-chloro-3-(4-chlorophenylsulfonyl)quinazoline-2,4...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human recombinant chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50058973(3-(3,4-Dichloro-benzenesulfonyl)-1-phenyl-imidazol...)
Affinity DataIC50:  18nMAssay Description:Inhibitory activity against human heart chymase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50058984(3-(3,4-Dichloro-benzenesulfonyl)-1-(3,4-dimethyl-p...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against human heart chymase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50058990(3-(3,4-Dimethoxy-benzenesulfonyl)-1-(3,4-dimethyl-...)
Affinity DataIC50:  22nMAssay Description:Inhibitory activity against human heart chymase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50210098(6-(4,5-dichloro-2-methoxybenzyl)-4-(4-chlorophenyl...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human recombinant chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50058996(3-(4-Chloro-benzenesulfonyl)-1-(3,4-dichloro-pheny...)
Affinity DataIC50:  23nMAssay Description:Inhibitory activity against human heart chymase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50210116(6-(5-fluoro-2-methoxybenzyl)-4-(4-chlorophenylsulf...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human recombinant chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50210120((S)-6-(5-chloro-2-methoxybenzyl)-4-(4-chlorophenyl...)
Affinity DataIC50:  27nMAssay Description:Inhibition of human recombinant chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50210094(3-((1-(4-chlorophenylsulfonyl)-3,7-dioxo-1,4-diaze...)
Affinity DataIC50:  27nMAssay Description:Inhibition of human recombinant chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50059007(4-(2,5-Dioxo-3-phenyl-imidazolidine-1-sulfonyl)-be...)
Affinity DataIC50:  29nMAssay Description:Inhibitory activity against human heart chymase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50058964(3-(3,4-Dimethyl-benzenesulfonyl)-1-phenyl-imidazol...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against human heart chymase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227791(CHEMBL53815)
Affinity DataIC50:  34nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM100740(CHEMBL391608 | US8507714, 29)
Affinity DataIC50:  34nMAssay Description:Inhibition of human recombinant chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50058969(3-(4-Chloro-benzenesulfonyl)-1-(3,4-dimethyl-pheny...)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity against human heart chymase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50210099(CHEMBL246964 | rac-2q)
Affinity DataIC50:  39nMAssay Description:Inhibition of human recombinant chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50058972(4-(2,5-Dioxo-3-phenyl-imidazolidine-1-sulfonyl)-be...)
Affinity DataIC50:  40nMAssay Description:Inhibitory activity against human heart chymase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50210096(2-(4-chloro-2-((1-(4-chlorophenylsulfonyl)-3,7-dio...)
Affinity DataIC50:  42nMAssay Description:Inhibition of human recombinant chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM87059(CHEMBL247767 | Chymostatin)
Affinity DataIC50:  43nMAssay Description:Inhibition of human recombinant chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Suntory

Curated by ChEMBL
LigandPNGBDBM50058977(3-Benzoyl-1-phenyl-imidazolidine-2,4-dione | CHEMB...)
Affinity DataIC50:  48nMAssay Description:Inhibitory activity against bovine pancreas alpha-chymotrypsin in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50093789(CHEMBL541829 | Succinic acid mono-(2-dimethylamino...)
Affinity DataIC50:  51nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227788(CHEMBL1743936)
Affinity DataIC50:  54nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227837(CHEMBL52131)
Affinity DataIC50:  55nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50058999(3-(3,4-Dimethyl-benzenesulfonyl)-1-(3,4-dimethyl-p...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity against human heart chymase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227787(CHEMBL1743933)
Affinity DataIC50:  62nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50059002(3-(4-Chloro-benzenesulfonyl)-1-(3-chloro-phenyl)-i...)
Affinity DataIC50:  66nMAssay Description:Inhibitory activity against human heart chymase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50058975(3-(2,5-Dioxo-3-phenyl-imidazolidine-1-sulfonyl)-be...)
Affinity DataIC50:  68nMAssay Description:Inhibitory activity against human heart chymase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50058994(3-(2,5-Dioxo-3-phenyl-imidazolidine-1-sulfonyl)-be...)
Affinity DataIC50:  82nMAssay Description:Inhibitory activity against human heart chymase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50210113(6-(5-chloro-2-ethoxybenzyl)-4-(4-chlorophenylsulfo...)
Affinity DataIC50:  83nMAssay Description:Inhibition of human recombinant chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227978(CHEMBL53316)
Affinity DataIC50:  96nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50210097(6-(2-chlorobenzyl)-4-(4-chlorophenylsulfonyl)-1,4-...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human recombinant chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM50059014(3-(3,4-Dimethoxy-benzenesulfonyl)-1-phenyl-imidazo...)
Affinity DataIC50:  110nMAssay Description:Inhibitory activity against human heart chymase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50228190(CHEMBL54263)
Affinity DataIC50:  115nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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