Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Antagonist activity at human mGLUR1More data for this Ligand-Target Pair
Affinity DataKi: 6.76nMAssay Description:Binding affinity to human mGluR5More data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 8.78nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Antagonist activity at mGLUR5 in rat E17 cells assessed as calcium accumulation by fluorimetryMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Antagonist activity at mGLUR5 in rat E17 cells assessed as calcium accumulation by fluorimetryMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Antagonist activity at mGLUR5 in rat E17 cells assessed as calcium accumulation by fluorimetryMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Antagonist activity at human mGLUR1More data for this Ligand-Target Pair
Affinity DataKi: 36.3nMAssay Description:Binding affinity to human mGluR5More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 49.0nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 57.5nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 72.4nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 77.6nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 83.2nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 87.1nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 89.1nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 102nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 104nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 105nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 117nMAssay Description:Antagonist activity at mGLUR5 in rat E17 cells assessed as calcium accumulation by fluorimetryMore data for this Ligand-Target Pair
Affinity DataKi: 123nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 138nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 145nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Displacement of [3H]-M-MPEP from rat mGLUR5More data for this Ligand-Target Pair
Affinity DataKi: 182nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 186nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 195nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 195nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 204nMAssay Description:Binding affinity to human mGluR5More data for this Ligand-Target Pair
Affinity DataKi: 229nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 438nMAssay Description:Antagonist activity at mGLUR5 in rat E17 cells assessed as calcium accumulation by fluorimetryMore data for this Ligand-Target Pair
Affinity DataKi: 457nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 741nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Antagonist activity at mGLUR5 in rat E17 cells assessed as calcium accumulation by fluorimetryMore data for this Ligand-Target Pair