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Found 39 with Last Name = 'giannini' and Initial = 'a'
TargetIntegrase(Human immunodeficiency virus 1)
Irbm

Curated by ChEMBL
LigandPNGBDBM25351(N-[2-(4-{[(4-fluorophenyl)methyl]carbamoyl}-5-hydr...)
Affinity DataIC50:  27nMAssay Description:Inhibition of wild type recombinant HIV1 His6-tagged integrase expressed in Escherichia coli BL21 using 18 nucleotide 3'-biotin labeled DNA acceptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552035(CHEMBL4792698)
Affinity DataIC50:  100nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552040(CHEMBL4764675)
Affinity DataIC50:  120nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552034(CHEMBL4743218)
Affinity DataIC50:  140nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552041(CHEMBL4744776)
Affinity DataIC50:  150nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50537058(CHEMBL4531719)
Affinity DataIC50:  300nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552022(CHEMBL4785115)
Affinity DataIC50:  400nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552031(CHEMBL4741968)
Affinity DataIC50:  490nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552032(CHEMBL4742331)
Affinity DataIC50:  820nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552024(CHEMBL4741684)
Affinity DataIC50:  890nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552033(CHEMBL4787707)
Affinity DataIC50:  940nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552037(CHEMBL4784714)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552023(CHEMBL4799050)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552038(CHEMBL4790390)
Affinity DataIC50:  1.51E+3nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552039(CHEMBL4795681)
Affinity DataIC50:  2.02E+3nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552036(CHEMBL4761720)
Affinity DataIC50:  2.49E+3nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552027(CHEMBL4742051)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552021(CHEMBL4764209)
Affinity DataIC50:  5.09E+3nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552025(CHEMBL4786545)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552026(CHEMBL4783844)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540670(CHEMBL4633550)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human microsomal CYP2D6 expressed in baculovirus infected insect cells using luciferin-ME as substrate preincubated with enzyme/substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540669(CHEMBL4637524)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human microsomal CYP2D6 expressed in baculovirus infected insect cells using luciferin-ME as substrate preincubated with enzyme/substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540668(CHEMBL4637717)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human microsomal CYP2D6 expressed in baculovirus infected insect cells using luciferin-ME as substrate preincubated with enzyme/substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540671(CHEMBL4635907)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human microsomal CYP1A2 expressed in baculovirus infected insect cells using luciferin-1A2 as substrate preincubated with enzyme-substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540670(CHEMBL4633550)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human microsomal CYP1A2 expressed in baculovirus infected insect cells using luciferin-1A2 as substrate preincubated with enzyme-substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540669(CHEMBL4637524)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human microsomal CYP1A2 expressed in baculovirus infected insect cells using luciferin-1A2 as substrate preincubated with enzyme-substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540668(CHEMBL4637717)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human microsomal CYP1A2 expressed in baculovirus infected insect cells using luciferin-1A2 as substrate preincubated with enzyme-substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540671(CHEMBL4635907)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of Tracer Red from human ERG measured after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540670(CHEMBL4633550)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of Tracer Red from human ERG measured after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540671(CHEMBL4635907)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human microsomal CYP2D6 expressed in baculovirus infected insect cells using luciferin-ME as substrate preincubated with enzyme/substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540668(CHEMBL4637717)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human microsomal CYP3A4 expressed in baculovirus infected insect cells using luciferin-IPA as substrate preincubated with enzyme/substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540671(CHEMBL4635907)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human microsomal CYP3A4 expressed in baculovirus infected insect cells using luciferin-IPA as substrate preincubated with enzyme/substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540670(CHEMBL4633550)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human microsomal CYP3A4 expressed in baculovirus infected insect cells using luciferin-IPA as substrate preincubated with enzyme/substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540669(CHEMBL4637524)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human microsomal CYP3A4 expressed in baculovirus infected insect cells using luciferin-IPA as substrate preincubated with enzyme/substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540668(CHEMBL4637717)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of Tracer Red from human ERG measured after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Irbm

Curated by ChEMBL
LigandPNGBDBM50540669(CHEMBL4637524)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of Tracer Red from human ERG measured after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552028(CHEMBL4764635)
Affinity DataIC50:  4.01E+4nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552029(CHEMBL4758562)
Affinity DataIC50:  5.38E+4nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50552030(CHEMBL4743223)
Affinity DataIC50:  5.97E+4nMAssay Description:Inhibition of human DDX3X using dsRNA as substrate measured every 30 sec for 40 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed