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Found 41 with Last Name = 'gilardone' and Initial = 'm'
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516083(CHEMBL4470490)
Affinity DataIC50:  4nMAssay Description:Inhibition of CypD (unknown origin) PPIase activity using N-Suc-AAPF-p-nitroanilide as substrate preincubated with enzyme for 10 mins followed by chy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516083(CHEMBL4470490)
Affinity DataIC50:  60nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516100(CHEMBL4466871)
Affinity DataIC50:  190nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516080(CHEMBL4464178)
Affinity DataIC50:  600nMAssay Description:Inhibition of CypD (unknown origin) PPIase activity using N-Suc-AAPF-p-nitroanilide as substrate preincubated with enzyme for 10 mins followed by chy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516098(CHEMBL4547673)
Affinity DataIC50:  735nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516080(CHEMBL4464178)
Affinity DataIC50:  1.35E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516082(CHEMBL4464825)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of CypD (unknown origin) PPIase activity using N-Suc-AAPF-p-nitroanilide as substrate preincubated with enzyme for 10 mins followed by chy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516084(CHEMBL4520315)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516095(CHEMBL4451136)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516082(CHEMBL4464825)
Affinity DataIC50:  2.00E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516087(CHEMBL4471175)
Affinity DataIC50:  2.80E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516096(CHEMBL4540033)
Affinity DataIC50:  3.50E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516094(CHEMBL4453162)
Affinity DataIC50:  3.60E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516090(CHEMBL4563478)
Affinity DataIC50:  4.10E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516096(CHEMBL4540033)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of CypD (unknown origin) PPIase activity using N-Suc-AAPF-p-nitroanilide as substrate preincubated with enzyme for 10 mins followed by chy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDedicator of cytokinesis protein 5(Homo sapiens)
Universit£

Curated by ChEMBL
LigandPNGBDBM50554781(CHEMBL4749280)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516093(CHEMBL4445439)
Affinity DataIC50:  1.00E+4nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDedicator of cytokinesis protein 5(Mus musculus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50554780(CHEMBL4791793)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of N-terminal GFP tagged mouse DOCK5 expressed in HEK293T cells assessed as reduction in exchange activity incubated for 1 hr by Western b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDedicator of cytokinesis protein 5(Homo sapiens)
Universit£

Curated by ChEMBL
LigandPNGBDBM50554782(CHEMBL4783937)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDedicator of cytokinesis protein 5(Homo sapiens)
Universit£

Curated by ChEMBL
LigandPNGBDBM50554786(CHEMBL4745076)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDedicator of cytokinesis protein 5(Homo sapiens)
Universit£

Curated by ChEMBL
LigandPNGBDBM50554780(CHEMBL4791793)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516087(CHEMBL4471175)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of CypD (unknown origin) PPIase activity using N-Suc-AAPF-p-nitroanilide as substrate preincubated with enzyme for 10 mins followed by chy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDedicator of cytokinesis protein 5(Homo sapiens)
Universit£

Curated by ChEMBL
LigandPNGBDBM50554787(CHEMBL4752328)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516099(CHEMBL4585544)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDedicator of cytokinesis protein 5(Homo sapiens)
Universit£

Curated by ChEMBL
LigandPNGBDBM50554784(CHEMBL4759130)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDedicator of cytokinesis protein 5(Homo sapiens)
Universit£

Curated by ChEMBL
LigandPNGBDBM50554785(CHEMBL4763851)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDedicator of cytokinesis protein 5(Homo sapiens)
Universit£

Curated by ChEMBL
LigandPNGBDBM50554789(CHEMBL4758729)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDedicator of cytokinesis protein 5(Homo sapiens)
Universit£

Curated by ChEMBL
LigandPNGBDBM50554788(CHEMBL4744468)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDedicator of cytokinesis protein 5(Mus musculus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50554779(CHEMBL4794083)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of N-terminal GFP tagged mouse DOCK5 expressed in HEK293T cells assessed as reduction in exchange activity incubated for 1 hr by Western b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516081(CHEMBL4570230)
Affinity DataIC50:  4.40E+4nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDedicator of cytokinesis protein 5(Homo sapiens)
Universit£

Curated by ChEMBL
LigandPNGBDBM50554783(CHEMBL4795607)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516092(CHEMBL4456924)
Affinity DataIC50:  5.40E+4nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516097(CHEMBL4579041)
Affinity DataIC50:  8.00E+4nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516091(CHEMBL4530010)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516086(CHEMBL4450619)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516088(CHEMBL4593662)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516089(CHEMBL4526530)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516085(CHEMBL4444722)
Affinity DataIC50:  4.90E+5nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50516101(CHEMBL4436790)
Affinity DataIC50:  8.70E+5nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataKd:  30nMAssay Description:Binding affinity to CypD (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
Merck Healthcare

Curated by ChEMBL
LigandPNGBDBM50164667(CHEMBL3798755)
Affinity DataKd:  230nMAssay Description:Binding affinity to CypD (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed