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Found 104 with Last Name = 'goeldner' and Initial = 'm'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50012477(1-Phenethyl-4-(phenyl-propionyl-amino)-piperidine-...)
Affinity DataKi:  0.0900nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.180nMAssay Description:In vitro inhibitory potency for preventing ET-1 induced constriction of rat aortic rings (ETA receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012477(1-Phenethyl-4-(phenyl-propionyl-amino)-piperidine-...)
Affinity DataKi:  0.25nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50125187(2-(2-Chloro-pyrimidin-5-yl)-7-aza-bicyclo[2.2.1]he...)
Affinity DataKi:  0.310nMAssay Description:In vitro inhibitory potency for preventing sarafotoxin S6c induced constriction of rat tracheal rings (ETB receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50013849(14-[4-azido(methyl)anilino]-4-cyclopropylmethyl-12...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013847(CHEMBL312040 | Etonitazene | {2-[2-(4-Ethoxy-benzy...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  0.550nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013857(14-[4-diazo(methyl)anilino]-4-cyclopropylmethyl-12...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013857(14-[4-diazo(methyl)anilino]-4-cyclopropylmethyl-12...)
Affinity DataKi:  0.600nMAssay Description:Opioid receptor delta 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013849(14-[4-azido(methyl)anilino]-4-cyclopropylmethyl-12...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50013847(CHEMBL312040 | Etonitazene | {2-[2-(4-Ethoxy-benzy...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013849(14-[4-azido(methyl)anilino]-4-cyclopropylmethyl-12...)
Affinity DataKi:  0.700nMAssay Description:Opioid receptor delta 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013849(14-[4-azido(methyl)anilino]-4-cyclopropylmethyl-12...)
Affinity DataKi:  0.700nMAssay Description:Opioid receptor kappa 1 apparent binding constant from guinea pig cerebellum using [3H]diprenorphine binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013857(14-[4-diazo(methyl)anilino]-4-cyclopropylmethyl-12...)
Affinity DataKi:  1nMAssay Description:Opioid receptor kappa 1 apparent binding constant from guinea pig cerebellum using [3H]diprenorphine binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50013857(14-[4-diazo(methyl)anilino]-4-cyclopropylmethyl-12...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013854(CHEMBL310829 | {2-[5-Azido-2-(4-ethoxy-benzyl)-ben...)
Affinity DataKi:  2nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013855(1-(4-Azido-phenyl)-8-[1-(4-chloro-phenyl)-ethyl]-1...)
Affinity DataKi:  3nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013848(8-[1-(4-Chloro-phenyl)-ethyl]-1-phenyl-1,3,8-triaz...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50013854(CHEMBL310829 | {2-[5-Azido-2-(4-ethoxy-benzyl)-ben...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50013855(1-(4-Azido-phenyl)-8-[1-(4-chloro-phenyl)-ethyl]-1...)
Affinity DataKi:  5nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  6.70nMAssay Description:Opioid receptor delta 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Université

Curated by ChEMBL
LigandPNGBDBM50082020(2-Chloro-N-{2-[3-(7-chloro-4-hydroxy-2-oxo-1,2-dih...)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]-5-7 dichlorokynurenic acid ([3H]- DCKA) from N-methyl-D-aspartate glutamate receptor glycine site of rat brain membrane homogen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013853(1-[2-(4-Azido-phenyl)-ethyl]-4-(phenyl-propionyl-a...)
Affinity DataKi:  8nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50013853(1-[2-(4-Azido-phenyl)-ethyl]-4-(phenyl-propionyl-a...)
Affinity DataKi:  8nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  8.70nMAssay Description:Opioid receptor kappa 1 apparent binding constant from guinea pig cerebellum using [3H]diprenorphine binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50012477(1-Phenethyl-4-(phenyl-propionyl-amino)-piperidine-...)
Affinity DataKi:  9nMAssay Description:Opioid receptor kappa 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50013848(8-[1-(4-Chloro-phenyl)-ethyl]-1-phenyl-1,3,8-triaz...)
Affinity DataKi:  10nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50007674((+)-erythro 4-[2-(4-Benzyl-piperidin-1-yl)-1-hydro...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]ifenprodil from rat brain membrane NR2B receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013852(1-(2-Diethylamino-ethyl)-2-(4-ethoxy-benzyl)-1H-be...)
Affinity DataKi:  11nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013850(4-{8-[1-(4-Chloro-phenyl)-ethyl]-4-oxo-1,3,8-triaz...)
Affinity DataKi:  11nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Université

Curated by ChEMBL
LigandPNGBDBM50082027(2-Chloro-N-{3-[3-(7-chloro-4-hydroxy-2-oxo-1,2-dih...)
Affinity DataKi:  13.8nMAssay Description:Displacement of [3H]-5-7 dichlorokynurenic acid ([3H]- DCKA) from N-methyl-D-aspartate glutamate receptor glycine site of rat brain membrane homogen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Université

Curated by ChEMBL
LigandPNGBDBM50038168(7-Chloro-4-hydroxy-3-(3-phenoxy-phenyl)-1H-quinoli...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-5-7 dichlorokynurenic acid ([3H]- DCKA) from N-methyl-D-aspartate glutamate receptor glycine site of rat brain membrane homogen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50125188(CHEMBL268176 | N-[5-(7-Aza-bicyclo[2.2.1]hept-2-yl...)
Affinity DataKi:  16nMAssay Description:In vitro inhibitory potency for preventing ET-1 induced constriction of rat aortic rings (ETA receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50013852(1-(2-Diethylamino-ethyl)-2-(4-ethoxy-benzyl)-1H-be...)
Affinity DataKi:  18nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Université

Curated by ChEMBL
LigandPNGBDBM50082022(2-[3-(7-Chloro-4-hydroxy-2-oxo-1,2-dihydro-quinoli...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]-5-7 dichlorokynurenic acid ([3H]- DCKA) from N-methyl-D-aspartate glutamate receptor glycine site of rat brain membrane homogen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Université

Curated by ChEMBL
LigandPNGBDBM50082021(4-Fluorosulfonyl-benzoic acid 7-chloro-2-oxo-3-(3-...)
Affinity DataKi:  24.2nMAssay Description:Displacement of [3H]-5-7 dichlorokynurenic acid ([3H]- DCKA) from N-methyl-D-aspartate glutamate receptor glycine site of rat brain membrane homogen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Université

Curated by ChEMBL
LigandPNGBDBM50082024(2-{2-[3-(7-Chloro-4-hydroxy-2-oxo-1,2-dihydro-quin...)
Affinity DataKi:  26.8nMAssay Description:Displacement of [3H]-5-7 dichlorokynurenic acid ([3H]- DCKA) from N-methyl-D-aspartate glutamate receptor glycine site of rat brain membrane homogen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50013856(1-[2-(4-Azido-3-iodo-phenyl)-ethyl]-4-(phenyl-prop...)
Affinity DataKi:  27nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Université

Curated by ChEMBL
LigandPNGBDBM50082016(2-Chloro-N-[3-(7-chloro-4-hydroxy-2-oxo-1,2-dihydr...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-5-7 dichlorokynurenic acid ([3H]- DCKA) from N-methyl-D-aspartate glutamate receptor glycine site of rat brain membrane homogen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013856(1-[2-(4-Azido-3-iodo-phenyl)-ethyl]-4-(phenyl-prop...)
Affinity DataKi:  45nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Université

Curated by ChEMBL
LigandPNGBDBM50082023(7-Chloro-4-hydroxy-3-(3-isothiocyanato-phenyl)-1H-...)
Affinity DataKi:  47.6nMAssay Description:Displacement of [3H]-5-7 dichlorokynurenic acid ([3H]- DCKA) from N-methyl-D-aspartate glutamate receptor glycine site of rat brain membrane homogen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50377833(CHEMBL413998)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]ifenprodil from rat brain membrane NR2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50377825(CHEMBL258032)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]ifenprodil from rat brain membrane NR2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50013850(4-{8-[1-(4-Chloro-phenyl)-ethyl]-4-oxo-1,3,8-triaz...)
Affinity DataKi:  62nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Université

Curated by ChEMBL
LigandPNGBDBM50082025(4-Hydroxy-7-isothiocyanato-3-(3-phenoxy-phenyl)-1H...)
Affinity DataKi:  64.3nMAssay Description:Displacement of [3H]-5-7 dichlorokynurenic acid ([3H]- DCKA) from N-methyl-D-aspartate glutamate receptor glycine site of rat brain membrane homogen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013848(8-[1-(4-Chloro-phenyl)-ethyl]-1-phenyl-1,3,8-triaz...)
Affinity DataKi:  75nMAssay Description:Opioid receptor delta 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50012477(1-Phenethyl-4-(phenyl-propionyl-amino)-piperidine-...)
Affinity DataKi:  92nMAssay Description:Opioid receptor kappa 1 apparent binding constant from guinea pig cerebellum using [3H]diprenorphine binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50377831(CHEMBL255697)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]ifenprodil from rat brain membrane NR2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50377831(CHEMBL255697)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]ifenprodil from rat brain membrane NR2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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