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Found 118 with Last Name = 'graziano' and Initial = 'mp'
TargetSuccinate receptor 1(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393161(CHEMBL2153439)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at rat GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393129(CHEMBL2153461)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393123(CHEMBL2153446)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393133(CHEMBL2153465)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393122(CHEMBL2153445)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393136(CHEMBL2153468)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393130(CHEMBL2153462)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393135(CHEMBL2153467)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393134(CHEMBL2153466)
Affinity DataIC50:  19nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393118(CHEMBL2153441)
Affinity DataIC50:  22nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393161(CHEMBL2153439)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393127(CHEMBL2153459)
Affinity DataIC50:  31nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393131(CHEMBL2153463)
Affinity DataIC50:  34nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393143(CHEMBL2153581)
Affinity DataIC50:  35nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393119(CHEMBL2153442)
Affinity DataIC50:  38nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393148(CHEMBL2153586)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393117(CHEMBL2153440)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393120(CHEMBL2153443)
Affinity DataIC50:  41nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393137(CHEMBL2153469)
Affinity DataIC50:  49nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393141(CHEMBL2153579)
Affinity DataIC50:  65nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393121(CHEMBL2153444)
Affinity DataIC50:  65nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393148(CHEMBL2153586)
Affinity DataIC50:  67nMAssay Description:Antagonist activity at rat GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393128(CHEMBL2153460)
Affinity DataIC50:  75nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393142(CHEMBL2153580)
Affinity DataIC50:  90nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393123(CHEMBL2153446)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at rat GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393149(CHEMBL2153587)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393117(CHEMBL2153440)
Affinity DataIC50:  115nMAssay Description:Antagonist activity at rat GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393143(CHEMBL2153581)
Affinity DataIC50:  135nMAssay Description:Antagonist activity at rat GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393158(CHEMBL2153596)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393156(CHEMBL2153594)
Affinity DataIC50:  170nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393157(CHEMBL2153595)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50396195(CHEMBL2172048)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat Hao2-mediated oxidation of 2-hydroxyoctanoic acid assessed as proportionate release of H2O2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50396202(CHEMBL2172039)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat Hao2-mediated oxidation of 2-hydroxyoctanoic acid assessed as proportionate release of H2O2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50396218(CHEMBL2172167)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat Hao2-mediated oxidation of 2-hydroxyoctanoic acid assessed as proportionate release of H2O2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393150(CHEMBL2153588)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393138(CHEMBL2153470)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393140(CHEMBL2153472)
Affinity DataIC50:  210nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393147(CHEMBL2153585)
Affinity DataIC50:  270nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50382412(CHEMBL2022570)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat His6-tagged Hao2 expressed in Escherichia coli BL21/DE3 using 2-hydroxyoctanoic acid as substrate measured every 10 secs by spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50382413(CHEMBL2022571)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat His6-tagged Hao2 expressed in Escherichia coli BL21/DE3 using 2-hydroxyoctanoic acid as substrate measured every 10 secs by spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50396192(CHEMBL2172051)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat Hao2-mediated oxidation of 2-hydroxyoctanoic acid assessed as proportionate release of H2O2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50382413(CHEMBL2022571)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat Hao2-mediated oxidation of 2-hydroxyoctanoic acid assessed as proportionate release of H2O2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50396198(CHEMBL2172043)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat Hao2-mediated oxidation of 2-hydroxyoctanoic acid assessed as proportionate release of H2O2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393145(CHEMBL2153583)
Affinity DataIC50:  300nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50396205(CHEMBL2172036)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat Hao2-mediated oxidation of 2-hydroxyoctanoic acid assessed as proportionate release of H2O2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50382412(CHEMBL2022570)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat Hao2-mediated oxidation of 2-hydroxyoctanoic acid assessed as proportionate release of H2O2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50396217(CHEMBL2172169)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat Hao2-mediated oxidation of 2-hydroxyoctanoic acid assessed as proportionate release of H2O2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393126(CHEMBL2153457)
Affinity DataIC50:  300nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50396203(CHEMBL2172038)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat Hao2-mediated oxidation of 2-hydroxyoctanoic acid assessed as proportionate release of H2O2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393132(CHEMBL2153464)
Affinity DataIC50:  330nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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