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Found 219 with Last Name = 'gupta' and Initial = 'mk'
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College of Pharmacy (Isfcp)

Curated by ChEMBL
LigandPNGBDBM50090023(4-(3,4-Difluoro-phenyl)-2-oxo-1,2,3,4-tetrahydro-p...)
Affinity DataKi:  0.0700nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College of Pharmacy (Isfcp)

Curated by ChEMBL
LigandPNGBDBM50090018(4-(3,4-Difluoro-phenyl)-2-oxo-1,2,3,4-tetrahydro-p...)
Affinity DataKi:  0.130nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College of Pharmacy (Isfcp)

Curated by ChEMBL
LigandPNGBDBM50090027((R)-4-(3,4-Difluoro-phenyl)-1,3,6-trimethyl-2-oxo-...)
Affinity DataKi:  0.140nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College of Pharmacy (Isfcp)

Curated by ChEMBL
LigandPNGBDBM50245653(CHEMBL4100620)
Affinity DataKi:  0.160nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College of Pharmacy (Isfcp)

Curated by ChEMBL
LigandPNGBDBM50245650(CHEMBL4062896)
Affinity DataKi:  0.170nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College of Pharmacy (Isfcp)

Curated by ChEMBL
LigandPNGBDBM50090031(4-(3,4-Difluoro-phenyl)-2-oxo-1,2,3,4-tetrahydro-p...)
Affinity DataKi:  0.170nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College of Pharmacy (Isfcp)

Curated by ChEMBL
LigandPNGBDBM50245652(CHEMBL4081581)
Affinity DataKi:  0.180nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College of Pharmacy (Isfcp)

Curated by ChEMBL
LigandPNGBDBM50090043(4-(3,4-Difluoro-phenyl)-6-methoxymethyl-2-oxo-1,2,...)
Affinity DataKi:  0.240nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College of Pharmacy (Isfcp)

Curated by ChEMBL
LigandPNGBDBM50090013(4-(3,4-Difluoro-phenyl)-6-methoxymethyl-2-oxo-1,2,...)
Affinity DataKi:  0.450nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College of Pharmacy (Isfcp)

Curated by ChEMBL
LigandPNGBDBM50090041(6-(3,4-Difluoro-phenyl)-5-{3-[4-(4-fluoro-phenyl)-...)
Affinity DataKi:  0.75nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College of Pharmacy (Isfcp)

Curated by ChEMBL
LigandPNGBDBM50090021(3-Acetyl-4-(3,4-difluoro-phenyl)-1,6-dimethyl-2-ox...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Indo-Soviet Friendship College of Pharmacy (Isfcp)

Curated by ChEMBL
LigandPNGBDBM50245651(CHEMBL4071004)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]SNAP-7941 from recombinant human MCHR1 expressed in African green monkey COS7 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235214(CHEMBL4084903)
Affinity DataIC50:  0.780nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235213(CHEMBL4102852)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235212(CHEMBL4092661)
Affinity DataIC50:  2nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50159614(2-(2-Fluoro-phenyl)-benzo[h]chromen-4-one | CHEMBL...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis)
Shri G.S. Institute Of Technology And Science

Curated by ChEMBL
LigandPNGBDBM50412347(CHEMBL499343)
Affinity DataIC50:  4nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50159673(2-(3-Fluoro-phenyl)-benzo[h]chromen-4-one | CHEMBL...)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235226(CHEMBL4083931)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50159655(2-(3-Chloro-phenyl)-benzo[h]chromen-4-one | CHEMBL...)
Affinity DataIC50:  7nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235216(CHEMBL4099439)
Affinity DataIC50:  11nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235227(CHEMBL4069506)
Affinity DataIC50:  11nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235215(CHEMBL4062213)
Affinity DataIC50:  14nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235228(CHEMBL4096846)
Affinity DataIC50:  16nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50159609(2-(4-Fluoro-phenyl)-benzo[h]chromen-4-one | CHEMBL...)
Affinity DataIC50:  20nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50159604(2-(3-Nitro-phenyl)-benzo[h]chromen-4-one | CHEMBL1...)
Affinity DataIC50:  25nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235217(CHEMBL4086963)
Affinity DataIC50:  26nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis)
Shri G.S. Institute Of Technology And Science

Curated by ChEMBL
LigandPNGBDBM23585((3-Phenoxybenzoylamino)benzoic acid deriv., 24i | ...)
Affinity DataIC50:  28.1nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235218(CHEMBL4078823)
Affinity DataIC50:  29nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235229(CHEMBL4081273)
Affinity DataIC50:  30nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235219(CHEMBL4063269)
Affinity DataIC50:  34nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50159605(2-(4-Nitro-phenyl)-benzo[h]chromen-4-one | CHEMBL1...)
Affinity DataIC50:  37nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235221(CHEMBL4070170)
Affinity DataIC50:  39nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235230(CHEMBL4097350)
Affinity DataIC50:  39nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235231(CHEMBL4067460)
Affinity DataIC50:  39nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235220(CHEMBL4093364)
Affinity DataIC50:  39nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235225(CHEMBL4073942)
Affinity DataIC50:  40nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235222(CHEMBL4080830)
Affinity DataIC50:  41nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235224(CHEMBL4088699)
Affinity DataIC50:  43nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50235223(CHEMBL4102088)
Affinity DataIC50:  43nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Sus scrofa)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50014323(2-PHENYL-4H-BENZO[H]CHROMEN-4-ONE | 2-Phenyl-benzo...)
Affinity DataIC50:  48nMAssay Description:Inhibition of porcine cholesterol esterase using para-nitrophenyl butyrate as substrate after 5 mins in presence of sodium taurocholate by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis)
Shri G.S. Institute Of Technology And Science

Curated by ChEMBL
LigandPNGBDBM23584((3-Phenoxybenzoylamino)benzoic acid deriv., 24c | ...)
Affinity DataIC50:  56.0nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis)
Shri G.S. Institute Of Technology And Science

Curated by ChEMBL
LigandPNGBDBM50412351(CHEMBL499342)
Affinity DataIC50:  62.1nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis)
Shri G.S. Institute Of Technology And Science

Curated by ChEMBL
LigandPNGBDBM23595((3-Phenoxybenzoylamino)benzoic acid deriv., 24d | ...)
Affinity DataIC50:  95.9nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis)
Shri G.S. Institute Of Technology And Science

Curated by ChEMBL
LigandPNGBDBM23594((3-Phenoxybenzoylamino)benzoic acid deriv., 24b | ...)
Affinity DataIC50:  110nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis)
Shri G.S. Institute Of Technology And Science

Curated by ChEMBL
LigandPNGBDBM23606((3-Phenoxybenzoylamino)benzoic acid deriv., 24p | ...)
Affinity DataIC50:  160nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis)
Shri G.S. Institute Of Technology And Science

Curated by ChEMBL
LigandPNGBDBM23596((3-Phenoxybenzoylamino)benzoic acid deriv., 24e | ...)
Affinity DataIC50:  160nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis)
Shri G.S. Institute Of Technology And Science

Curated by ChEMBL
LigandPNGBDBM23599((3-Phenoxybenzoylamino)benzoic acid deriv., 24h | ...)
Affinity DataIC50:  220nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis)
Shri G.S. Institute Of Technology And Science

Curated by ChEMBL
LigandPNGBDBM23602((3-Phenoxybenzoylamino)benzoic acid deriv., 24l | ...)
Affinity DataIC50:  240nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis)
Shri G.S. Institute Of Technology And Science

Curated by ChEMBL
LigandPNGBDBM23605((3-Phenoxybenzoylamino)benzoic acid deriv., 24o | ...)
Affinity DataIC50:  250nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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