Compile Data Set for Download or QSAR
maximum 50k data
Found 69 with Last Name = 'gynther' and Initial = 'm'
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50107595((S)-1-(2-Amino-2-carboxyethyl)-6,7-dihydro-1H-cycl...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK1 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50107595((S)-1-(2-Amino-2-carboxyethyl)-6,7-dihydro-1H-cycl...)
Affinity DataKi:  223nMAssay Description:Displacement of [3H]AMPA from recombinant homomeric rat GluA2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263221(CHEMBL4077177)
Affinity DataKi:  331nMAssay Description:Displacement of [3H]AMPA from recombinant homomeric rat GluA2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263220(CHEMBL4075364)
Affinity DataKi:  356nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK1 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  390nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2A expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263221(CHEMBL4077177)
Affinity DataKi:  586nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK1 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263224(CHEMBL4066795)
Affinity DataKi:  869nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK1 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263220(CHEMBL4075364)
Affinity DataKi:  1.99E+3nMAssay Description:Displacement of [3H]AMPA from recombinant homomeric rat GluA2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263220(CHEMBL4075364)
Affinity DataKi:  2.15E+3nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK3 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263224(CHEMBL4066795)
Affinity DataKi:  2.37E+3nMAssay Description:Displacement of [3H]AMPA from recombinant homomeric rat GluA2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  2.80E+3nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2B expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  4.70E+3nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2A expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50107595((S)-1-(2-Amino-2-carboxyethyl)-6,7-dihydro-1H-cycl...)
Affinity DataKi:  5.09E+3nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK3 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  5.90E+3nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2C expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  1.00E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2B expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246919(CHEMBL4099104)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246919(CHEMBL4099104)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263224(CHEMBL4066795)
Affinity DataKi:  1.81E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK3 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2D(RAT)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  2.10E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2D expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  2.40E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2C expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263223(CHEMBL4083716)
Affinity DataKi:  3.60E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK1 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2D(RAT)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  4.10E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2D expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246917(CHEMBL4068651)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263223(CHEMBL4083716)
Affinity DataKi:  1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK3 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246918(CHEMBL4091369)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263223(CHEMBL4083716)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]AMPA from recombinant homomeric rat GluA2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246911(CHEMBL4076785)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246914(CHEMBL4088958)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246914(CHEMBL4088958)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246911(CHEMBL4076785)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246916(CHEMBL4102488)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246918(CHEMBL4091369)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246915(CHEMBL4060745)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246917(CHEMBL4068651)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246916(CHEMBL4102488)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246919(CHEMBL4099104)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246914(CHEMBL4088958)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246916(CHEMBL4102488)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246911(CHEMBL4076785)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246918(CHEMBL4091369)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246917(CHEMBL4068651)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263221(CHEMBL4077177)
Affinity DataKi:  1.11E+5nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK3 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  1.31E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  1.54E+5nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50263224(CHEMBL4066795)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246913(CHEMBL4083586)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50246915(CHEMBL4060745)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246913(CHEMBL4083586)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246915(CHEMBL4060745)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 69 total ) | Next | Last >>
Jump to: