Affinity DataKi: 2.80nMAssay Description:In vivo antagonistic activity against cloned human oxytocin receptor overexpressed in a stable HEK293 cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:In vivo antagonistic activity against cloned human oxytocin receptor overexpressed in a stable HEK293 cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:In vivo antagonistic activity against cloned human oxytocin receptor over-expressed in a stable HEK293 cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity to human vasopressin V2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:In vivo antagonistic activity against cloned human oxytocin receptor overexpressed in a stable HEK293 cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity to human vasopressin V2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to oxytocin receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to oxytocin receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to oxytocin receptor (unknown origin)More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 5.60nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 6.40nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 6.90nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.70nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.70nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.20nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.60nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.90nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 9.10nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 9.5nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 10.7nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 10.8nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 10.8nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 350nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
Affinity DataEC50: 380nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
Affinity DataEC50: 47nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair