Compile Data Set for Download or QSAR
maximum 50k data
Found 118 with Last Name = 'hill' and Initial = 'rg'
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000091((6S,11R)-3-Cyclopropylmethyl-6-ethyl-8-hydroxy-11-...)
Affinity DataKi:  0.570nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000091((6S,11R)-3-Cyclopropylmethyl-6-ethyl-8-hydroxy-11-...)
Affinity DataKi:  1.70nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity towards mu opioid receptor was determinedMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018786(CHEMBL538309 | N-(2-Azocan-1-yl-cyclohexyl)-N-meth...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50008854(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity towards opioid receptor kappa was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018768(CHEMBL556957 | N-(2-Azepan-1-yl-cyclohexyl)-2-(4-c...)
Affinity DataKi:  4nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018762(2-Benzofuran-4-yl-N-methyl-N-(2-pyrrolidin-1-yl-cy...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018767(CHEMBL535581 | N-(2-Azocan-1-yl-cyclohexyl)-N-meth...)
Affinity DataKi:  5.60nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018771(CHEMBL535801 | N-(2-Azepan-1-yl-cyclohexyl)-N-meth...)
Affinity DataKi:  6.40nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50017495(2-Benzo[b]thiophen-4-yl-N-[2-(3-hydroxymethyl-pyrr...)
Affinity DataKi:  7nMAssay Description:Binding affinity towards opioid receptor kappa was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM21130(N-methyl-2-phenyl-N-[(5R,7S,8S)-7-(pyrrolidin-1-yl...)
Affinity DataKi:  7.30nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50008854(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  9.60nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 15 min of incubation at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50008854(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  9.60nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  10nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018781(CHEMBL557426 | N-Methyl-N-(2-pyrrolidin-1-yl-cyclo...)
Affinity DataKi:  12nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018762(2-Benzofuran-4-yl-N-methyl-N-(2-pyrrolidin-1-yl-cy...)
Affinity DataKi:  12nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 60 min of incubation at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018762(2-Benzofuran-4-yl-N-methyl-N-(2-pyrrolidin-1-yl-cy...)
Affinity DataKi:  12nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 0 min of incubation at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50017500(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  12nMAssay Description:Binding affinity towards Opioid receptor kappa 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50017488(2-Benzofuran-4-yl-N-(4,5-dimethoxy-2-pyrrolidin-1-...)
Affinity DataKi:  16nMAssay Description:Binding affinity towards Opioid receptor kappa 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50017498(2-Benzofuran-4-yl-N-[2-(3-hydroxymethyl-pyrrolidin...)
Affinity DataKi:  17nMAssay Description:Binding affinity towards Opioid receptor kappa 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50017494(2-Benzo[b]thiophen-7-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  17nMAssay Description:Binding affinity towards opioid receptor kappa was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM83436(2-(3,4-dichlorophenyl)-N-methyl-N-[(5R,7S,8S)-7-(1...)
Affinity DataKi:  17nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50013147(2-Benzo[b]thiophen-4-yl-N-(4,5-dimethoxy-2-pyrroli...)
Affinity DataKi:  18nMAssay Description:Binding affinity towards opioid receptor kappa was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018778(2-Benzo[b]thiophen-4-yl-N-methyl-N-[2-(methyl-phen...)
Affinity DataKi:  26nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018784(CHEMBL559217 | N-(2-Azepan-1-yl-cyclohexyl)-2-benz...)
Affinity DataKi:  29nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018778(2-Benzo[b]thiophen-4-yl-N-methyl-N-[2-(methyl-phen...)
Affinity DataKi:  30nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018764(2-(3,4-Dichloro-phenoxy)-N-methyl-N-(2-pyrrolidin-...)
Affinity DataKi:  35nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018788(CHEMBL537169 | N-(2-Azepan-1-yl-cyclohexyl)-2-benz...)
Affinity DataKi:  40nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018783(CHEMBL539582 | N-[2-(Allyl-methyl-amino)-cyclohexy...)
Affinity DataKi:  52nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM21130(N-methyl-2-phenyl-N-[(5R,7S,8S)-7-(pyrrolidin-1-yl...)
Affinity DataKi:  52nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50017504(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  53nMAssay Description:Binding affinity towards Opioid receptor kappa 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50017499(2-Benzo[b]thiophen-3-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  69nMAssay Description:Binding affinity towards Opioid receptor kappa 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018776(CHEMBL537615 | N-(2-Azepan-1-yl-cyclohexyl)-2-(3,5...)
Affinity DataKi:  72nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018763(2-(1H-Indol-3-yl)-N-methyl-N-(2-pyrrolidin-1-yl-cy...)
Affinity DataKi:  74nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018779(2-Benzo[b]thiophen-4-yl-N-methyl-N-{2-[methyl-(2-t...)
Affinity DataKi:  81nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018779(2-Benzo[b]thiophen-4-yl-N-methyl-N-{2-[methyl-(2-t...)
Affinity DataKi:  82nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  86nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  86nMAssay Description:Binding affinity towards Opioid receptor kappa 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50017489(2-Benzo[b]thiophen-5-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  94nMAssay Description:Binding affinity towards opioid receptor kappa was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50452622(CHEMBL2093981)
Affinity DataKi: >100nMAssay Description:Binding affinity towards opioid receptor mu was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018781(CHEMBL557426 | N-Methyl-N-(2-pyrrolidin-1-yl-cyclo...)
Affinity DataKi:  140nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50017501(2-Benzo[b]thiophen-6-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  146nMAssay Description:Binding affinity towards opioid receptor kappa was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018772(CHEMBL535130 | N-Methyl-2-(4-nitro-3-trifluorometh...)
Affinity DataKi:  150nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50017497(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  154nMAssay Description:Binding affinity towards opioid receptor kappa was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50017510(CHEMBL540277 | Succinic acid bis-(1-{2-[(2-benzofu...)
Affinity DataKi:  180nMAssay Description:Binding affinity towards opioid receptor kappa was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50017507(CHEMBL553665 | Pentanedioic acid bis-(1-{2-[(2-ben...)
Affinity DataKi:  180nMAssay Description:Binding affinity towards opioid receptor kappa was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018766(2-Benzo[b]thiophen-4-yl-N-[2-(cyclopropylmethyl-me...)
Affinity DataKi:  190nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018766(2-Benzo[b]thiophen-4-yl-N-[2-(cyclopropylmethyl-me...)
Affinity DataKi:  200nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018783(CHEMBL539582 | N-[2-(Allyl-methyl-amino)-cyclohexy...)
Affinity DataKi:  210nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 118 total ) | Next | Last >>
Jump to: