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Found 16 with Last Name = 'hirohama' and Initial = 'm'
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50439441(CHEMBL2420738)
Affinity DataIC50:  1.11E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin) assessed as SUMO E1-SUMO thioester bond formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50439440(CHEMBL2420739)
Affinity DataIC50:  1.17E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin) assessed as SUMO E1-SUMO thioester bond formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50278299(1-(6-(7-chloroquinazolin-4-yloxy)pyridin-3-yl)-3-(...)
Affinity DataIC50:  1.34E+4nMAssay Description:Inhibition of recombinant GST-fused SUMO E1 (unknown origin) using RanGAP1 as substrate after 2 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1/2(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50278299(1-(6-(7-chloroquinazolin-4-yloxy)pyridin-3-yl)-3-(...)
Affinity DataIC50:  1.34E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin)-mediated RanGAP1 sumoylation by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50143899(CHEMBL3759613)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibition of recombinant GST-fused SUMO E1 (unknown origin) using RanGAP1 as substrate after 2 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50439442(CHEMBL2420737)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin) assessed as SUMO E1-SUMO thioester bond formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50143901(CHEMBL3758249)
Affinity DataIC50:  3.04E+4nMAssay Description:Inhibition of recombinant GST-fused SUMO E1 (unknown origin) using RanGAP1 as substrate after 2 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50143897(CHEMBL3758566)
Affinity DataIC50:  3.32E+4nMAssay Description:Inhibition of recombinant GST-fused SUMO E1 (unknown origin) using RanGAP1 as substrate after 2 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50439436(CHEMBL2420740)
Affinity DataIC50:  3.54E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin)-mediated RanGAP1 sumoylation by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50439439(CHEMBL1900956)
Affinity DataIC50:  3.56E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin)-mediated RanGAP1 sumoylation by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50439437(CHEMBL1572155)
Affinity DataIC50:  3.57E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin)-mediated RanGAP1 sumoylation by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50439438(CHEMBL1448459)
Affinity DataIC50:  5.73E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin)-mediated RanGAP1 sumoylation by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50143900(CHEMBL3758383)
Affinity DataIC50:  7.30E+4nMAssay Description:Inhibition of recombinant GST-fused SUMO E1 (unknown origin) using RanGAP1 as substrate after 2 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM96736(1-[6-(7-chloranylquinazolin-4-yl)oxypyridin-3-yl]-...)
Affinity DataIC50:  7.30E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin)-mediated RanGAP1 sumoylation by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50143896(CHEMBL3758250)
Affinity DataIC50:  9.26E+4nMAssay Description:Inhibition of recombinant GST-fused SUMO E1 (unknown origin) using RanGAP1 as substrate after 2 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50143898(CHEMBL3759177)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant GST-fused SUMO E1 (unknown origin) using RanGAP1 as substrate after 2 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed