Affinity DataKi: >0.0700nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 0.467nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 0.476nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition of human somatostatin receptor type 4More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of human somatostatin receptor type 2 (n=6)More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Binding affinity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 32.8nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Tested for binding affinity at human Somatostatin receptor type 4 using ([3-125I-Tyr11)]-SRIF-14 as the radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Inhibition of human somatostatin receptor type 4More data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:Inhibition of human somatostatin receptor type 4 (n=5)More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of human somatostatin receptor type 4More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Tested for binding affinity at human Somatostatin receptor type 4 using ([3-125I-Tyr11)]-SRIF-14 as the radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 109nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 124nMAssay Description:Inhibition of human somatostatin receptor type 4More data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Binding affinity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 152nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 218nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 486nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Inhibition of human somatostatin receptor type 4More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 759nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 1.07E+3nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
Affinity DataKi: 2.60E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair