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Found 27 with Last Name = 'hu' and Initial = 'ym'
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427125(CHEMBL2323444)
Affinity DataKi:  920nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427129(CHEMBL2323441)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427131(CHEMBL2323446)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427127(CHEMBL2323442)
Affinity DataKi:  3.70E+3nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427129(CHEMBL2323441)
Affinity DataKi:  8.80E+3nMAssay Description:Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427127(CHEMBL2323442)
Affinity DataKi:  9.80E+3nMAssay Description:Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427131(CHEMBL2323446)
Affinity DataKi:  1.07E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427125(CHEMBL2323444)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427126(CHEMBL2323443)
Affinity DataKi:  6.60E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427130(CHEMBL2323447)
Affinity DataKi:  7.10E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427130(CHEMBL2323447)
Affinity DataKi:  7.70E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427128(CHEMBL2321893)
Affinity DataKi:  8.30E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427126(CHEMBL2323443)
Affinity DataKi:  8.40E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427124(CHEMBL2323445)
Affinity DataKi:  8.60E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427128(CHEMBL2321893)
Affinity DataKi:  9.50E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427124(CHEMBL2323445)
Affinity DataKi:  9.50E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM50002692((AZT) 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  12.7nMAssay Description:Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM50526706(CHEMBL4545676)
Affinity DataIC50:  270nMAssay Description:Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM192670(3-(6-methoxy-3,4-dihydroquinolin-1(2H)-yl)-1-(4-o-...)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM192678(1-(4-(3-chlorophenyl)piperazin-1-yl)-3-(6-methoxy-...)
Affinity DataIC50:  1.86E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM192669(3-(6-methoxy-3,4-dihydroquinolin-1(2H)-yl)-1-(4-ph...)
Affinity DataIC50:  2.42E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM50062551(CHEBI:76010 | Dolutegravir | GSK1349572 | S-349572)
Affinity DataEC50:  3.60nMAssay Description:Inhibition of HIV-1 NL4-3 integrase E92Q/N155H double mutantMore data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus 2)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM50062551(CHEBI:76010 | Dolutegravir | GSK1349572 | S-349572)
Affinity DataEC50:  2.30nMAssay Description:Inhibition of wild type HIV-2 ROD9 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM50526705(CHEMBL106731)
Affinity DataEC50:  1.60E+3nMAssay Description:Inhibition of wild type HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM50062551(CHEBI:76010 | Dolutegravir | GSK1349572 | S-349572)
Affinity DataEC50:  1.5nMAssay Description:Inhibition of HIV-1 NL4-3 integrase T97A/Y143C double mutantMore data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM50062551(CHEBI:76010 | Dolutegravir | GSK1349572 | S-349572)
Affinity DataEC50:  1.5nMAssay Description:Inhibition of wild type HIV-1 NL4-3 integraseMore data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM50062551(CHEBI:76010 | Dolutegravir | GSK1349572 | S-349572)
Affinity DataEC50:  6.80nMAssay Description:Inhibition of HIV-1 NL4-3 integrase G140S/Q148R double mutantMore data for this Ligand-Target Pair