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Found 14 with Last Name = 'hummel-eisenbeiss' and Initial = 'j'
TargetSolute carrier organic anion transporter family member 1B3(Homo sapiens (Human))
German Cancer Research Center

Curated by PDSP Ki Database
LigandPNGBDBM86671(CAS_60719 | MK 571 | NSC_60719)
Affinity DataKi:  600nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1B3(Homo sapiens (Human))
German Cancer Research Center

Curated by PDSP Ki Database
LigandPNGBDBM86672(CAS_2909 | Cyclosporin A | NSC_2909)
Affinity DataKi:  1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
German Cancer Research Center

Curated by PDSP Ki Database
LigandPNGBDBM86671(CAS_60719 | MK 571 | NSC_60719)
Affinity DataKi:  8.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
Deutsches Krebsforschungszentrum

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataKi:  1.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of BMG uptake in membrane vesicles from Mrp2-expressing HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
German Cancer Research Center

Curated by PDSP Ki Database
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataKi:  2.10E+4nMAssay Description:TP_TRANSPORTER: inhibition of BMG uptake in membrane vesicles from MRP2-expressing HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
Deutsches Krebsforschungszentrum

Curated by ChEMBL
LigandPNGBDBM50420230(CHEMBL2074750)
Affinity DataIC50:  100nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.05 uM) in bile canalicular membranes from Wistar ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
Deutsches Krebsforschungszentrum

Curated by ChEMBL
LigandPNGBDBM50420229(CHEMBL2074720)
Affinity DataIC50:  120nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.05 uM) in bile canalicular membranes from Wistar ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
German Cancer Research Center

Curated by PDSP Ki Database
LigandPNGBDBM50420229(CHEMBL2074720)
Affinity DataIC50:  280nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.05 uM) in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
German Cancer Research Center

Curated by PDSP Ki Database
LigandPNGBDBM50420230(CHEMBL2074750)
Affinity DataIC50:  400nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.05 uM) in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Deutsches Krebsforschungszentrum

Curated by ChEMBL
LigandPNGBDBM50420229(CHEMBL2074720)
Affinity DataIC50:  420nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.05 uM) in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Deutsches Krebsforschungszentrum

Curated by ChEMBL
LigandPNGBDBM50420230(CHEMBL2074750)
Affinity DataIC50:  750nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.05 uM) in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
German Cancer Research Center

Curated by PDSP Ki Database
LigandPNGBDBM50485596(LEUKOTRIEN C4 | Leukotriene C4)
Affinity DataIC50:  3.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake (PAH: 0.1uM) in membrane vesicles from MRP2-expressing HEK cellsMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
German Cancer Research Center

Curated by PDSP Ki Database
LigandPNGBDBM50001285((E)-3-((3-(2-(7-chloroquinolin-2-yl)vinyl)phenyl)(...)
Affinity DataIC50:  4.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake (PAH: 0.1uM) in membrane vesicles from MRP2-expressing HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
German Cancer Research Center

Curated by PDSP Ki Database
LigandPNGBDBM50485598(3R14S-OCHRATOXIN A | CHEBI:7719)
Affinity DataIC50:  5.80E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake (PAH: 0.1uM) in membrane vesicles from MRP2-expressing HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed