TargetSolute carrier organic anion transporter family member 1B3(Homo sapiens (Human))
German Cancer Research Center
Curated by PDSP Ki Database
German Cancer Research Center
Curated by PDSP Ki Database
TargetSolute carrier organic anion transporter family member 1B3(Homo sapiens (Human))
German Cancer Research Center
Curated by PDSP Ki Database
German Cancer Research Center
Curated by PDSP Ki Database
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
German Cancer Research Center
Curated by PDSP Ki Database
German Cancer Research Center
Curated by PDSP Ki Database
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of BMG uptake in membrane vesicles from Mrp2-expressing HEK cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
German Cancer Research Center
Curated by PDSP Ki Database
German Cancer Research Center
Curated by PDSP Ki Database
Affinity DataKi: 2.10E+4nMAssay Description:TP_TRANSPORTER: inhibition of BMG uptake in membrane vesicles from MRP2-expressing HEK cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.05 uM) in bile canalicular membranes from Wistar ratMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.05 uM) in bile canalicular membranes from Wistar ratMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
German Cancer Research Center
Curated by PDSP Ki Database
German Cancer Research Center
Curated by PDSP Ki Database
Affinity DataIC50: 280nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.05 uM) in HepG2 cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
German Cancer Research Center
Curated by PDSP Ki Database
German Cancer Research Center
Curated by PDSP Ki Database
Affinity DataIC50: 400nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.05 uM) in HepG2 cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.05 uM) in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.05 uM) in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
German Cancer Research Center
Curated by PDSP Ki Database
German Cancer Research Center
Curated by PDSP Ki Database
Affinity DataIC50: 3.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake (PAH: 0.1uM) in membrane vesicles from MRP2-expressing HEK cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
German Cancer Research Center
Curated by PDSP Ki Database
German Cancer Research Center
Curated by PDSP Ki Database
Affinity DataIC50: 4.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake (PAH: 0.1uM) in membrane vesicles from MRP2-expressing HEK cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
German Cancer Research Center
Curated by PDSP Ki Database
German Cancer Research Center
Curated by PDSP Ki Database
Affinity DataIC50: 5.80E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake (PAH: 0.1uM) in membrane vesicles from MRP2-expressing HEK cellsMore data for this Ligand-Target Pair