TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 111nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 123nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 183nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 198nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 245nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 265nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 332nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 361nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Affinity DataIC50: 361nMAssay Description:Antagonist activity at GAL4 DBD-fused androgen receptor LBD (unknown origin) transfected in UAS-bla GripTite 293 cells assessed as inhibition of R188...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 402nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 407nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 425nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Antagonist activity at GAL4 DBD-fused androgen receptor LBD (unknown origin) transfected in UAS-bla GripTite 293 cells assessed as inhibition of R188...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 625nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 625nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Affinity DataIC50: 710nMAssay Description:Antagonist activity at GAL4 DBD-fused androgen receptor LBD (unknown origin) transfected in UAS-bla GripTite 293 cells assessed as inhibition of R188...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 736nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 775nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 777nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 811nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.07E+3nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
School Of Pharmacy And Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.17E+3nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Antagonist activity at GAL4 DBD-fused androgen receptor LBD (unknown origin) transfected in UAS-bla GripTite 293 cells assessed as inhibition of R188...More data for this Ligand-Target Pair
Affinity DataIC50: 3.76E+3nMAssay Description:Antagonist activity against androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity against androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5.09E+3nMAssay Description:Antagonist activity against androgen receptor (unknown origin)More data for this Ligand-Target Pair