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Found 243 with Last Name = 'kappler' and Initial = 'f'
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367049(CHEMBL604399)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367049(CHEMBL604399)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50228186(CHEMBL3706404)
Affinity DataKi:  110nMAssay Description:Compound was tested for inhibition constant with kidney form of M-2 variants of Rat methionine adenosyltransferase when ATP was the variable substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1(Rattus norvegicus)
Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50368140(CHEMBL3706401 | CHEMBL611854)
Affinity DataKi:  110nMAssay Description:Inhibition constants with Met (L-methionine) substrate site of M-2 (kidney form) variant of rat Methionine adenosyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1(Rattus norvegicus)
Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50368140(CHEMBL3706401 | CHEMBL611854)
Affinity DataKi:  120nMAssay Description:Inhibition constants against ATP substrate site of M-T (Novikoff Ascitic Hepatoma form) variant of rat Methionine adenosyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227269(CHEMBL3706402)
Affinity DataKi:  130nMAssay Description:Inhibition constant of ATP varied compound was measured on M-2 variate Methionine adenosyltransferase in rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227269(CHEMBL3706402)
Affinity DataKi:  130nMAssay Description:Compound was tested for inhibition constant with kidney form of M-2 variants of Rat methionine adenosyltransferase when ATP was the variable substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50226974(CHEMBL603986)
Affinity DataKi:  130nMAssay Description:Inhibition constants of M-2 Forms of rat methionine adenosyltransferase using ATP as the variable substrate; Inhibition is competitive typeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1(Rattus norvegicus)
Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50227269(CHEMBL3706402)
Affinity DataKi:  130nMAssay Description:Inhibition constants against ATP substrate site of M-2 (kidney form) variant of rat Methionine adenosyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50228186(CHEMBL3706404)
Affinity DataKi:  160nMAssay Description:Compound was tested for inhibition constant with kidney form of M-T variants of Rat methionine adenosyltransferase when ATP was the variable substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1(Rattus norvegicus)
Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50227269(CHEMBL3706402)
Affinity DataKi:  210nMAssay Description:Inhibition constants against Met (L-methionine)P substrate site of M-T (Novikoff Ascitic Hepatoma form) variant of rat Methionine adenosyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227269(CHEMBL3706402)
Affinity DataKi:  210nMAssay Description:Compound was tested for inhibition constant with kidney form of M-T variants of Rat methionine adenosyltransferase when ATP was the variable substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227269(CHEMBL3706402)
Affinity DataKi:  210nMAssay Description:Inhibition constant of ATP varied compound was measured on MT variant methionine adenosyltransferase in rat ascitic hepatoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50226974(CHEMBL603986)
Affinity DataKi:  210nMAssay Description:Inhibition constants of MT Forms of rat Novikoff Ascitic Hepatomae using ATP as the variable substrate; Inhibition is competitive typeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50228185(CHEMBL3706405)
Affinity DataKi:  270nMAssay Description:Compound was tested for inhibition constant with kidney form of M-2 variants of Rat methionine adenosyltransferase when ATP was the variable substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50226770(CHEMBL609078)
Affinity DataKi:  270nMAssay Description:Inhibition constant of compound with Novikoff ascitic hepatoma (M-T) form of rat methionine adenosyltransferase when ATP was used as variable substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50226972(CHEMBL606493)
Affinity DataKi:  270nMAssay Description:Inhibition constants of MT Forms of rat Novikoff Ascitic Hepatomae using ATP as the variable substrate; Inhibition is competitive typeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50226768(CHEMBL1791426)
Affinity DataKi:  270nMAssay Description:Inhibition constant of ATP varied compound was measured on MT variant methionine adenosyltransferase in rat ascitic hepatoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50226770(CHEMBL609078)
Affinity DataKi:  360nMAssay Description:Inhibition constant of compound with kidney (M-2) form of rat methionine adenosyltransferase when ATP was used as variable substrate;Competitive type...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50226768(CHEMBL1791426)
Affinity DataKi:  360nMAssay Description:Inhibition constant of ATP varied compound was measured on M-2 variate methionine adenosyltransferase in rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50226972(CHEMBL606493)
Affinity DataKi:  360nMAssay Description:Inhibition constants of M-2 Forms of rat methionine adenosyltransferase using ATP as the variable substrate; Inhibition is competitive typeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227270(CHEMBL3706403)
Affinity DataKi:  390nMAssay Description:Inhibition constant of ATP varied compound was measured on M-2 variate methionine adenosyltransferase in rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50228185(CHEMBL3706405)
Affinity DataKi:  410nMAssay Description:Compound was tested for inhibition constant with kidney form of M-T variants of Rat methionine adenosyltransferase when ATP was the variable substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227271(CHEMBL1791425)
Affinity DataKi:  440nMAssay Description:Inhibition constant of ATP varied compound was measured on M-2 variate methionine adenosyltransferase in rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227270(CHEMBL3706403)
Affinity DataKi:  630nMAssay Description:Inhibition constant of ATP varied compound was measured on MT variant methionine adenosyltransferase in rat ascitic hepatoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227269(CHEMBL3706402)
Affinity DataKi:  650nMAssay Description:Inhibition constant of Met varied compound was measured on M-2 variant Methionine adenosyltransferase in rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227269(CHEMBL3706402)
Affinity DataKi:  650nMAssay Description:Compound was tested for inhibition constant with kidney form of M-2 variants of Rat methionine adenosyltransferase when Methionine was the variable s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50226974(CHEMBL603986)
Affinity DataKi:  650nMAssay Description:Inhibition constants of M-2 Forms of rat methionine adenosyltransferase using Methionine as the variable substrate; Inhibition is non competitive typ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1(Rattus norvegicus)
Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50227269(CHEMBL3706402)
Affinity DataKi:  650nMAssay Description:Inhibition constants with Met (L-methionine) substrate site of M-2 (kidney form) variant of rat Methionine adenosyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227269(CHEMBL3706402)
Affinity DataKi:  670nMAssay Description:Inhibition constant of Met varied compound was measured on MT variant methionine adenosyltransferase in rat ascitic hepatoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227269(CHEMBL3706402)
Affinity DataKi:  670nMAssay Description:Compound was tested for inhibition constant with kidney form of M-T variants of Rat methionine adenosyltransferase when Methionine was the variable s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50226974(CHEMBL603986)
Affinity DataKi:  670nMAssay Description:Inhibition constants of MT Forms of rat Novikoff Ascitic Hepatomae using Methionine as the variable substrate; Inhibition is non competitive typeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1(Rattus norvegicus)
Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50227269(CHEMBL3706402)
Affinity DataKi:  670nMAssay Description:Inhibition constants against Met (L-methionine)P substrate site of M-T (Novikoff Ascitic Hepatoma form) variant of rat Methionine adenosyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1(Rattus norvegicus)
Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50368140(CHEMBL3706401 | CHEMBL611854)
Affinity DataKi:  740nMAssay Description:Inhibition constants against Met (L-methionine)P substrate site of M-T (Novikoff Ascitic Hepatoma form) variant of rat Methionine adenosyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227271(CHEMBL1791425)
Affinity DataKi:  810nMAssay Description:Inhibition constant of ATP varied compound was measured on MT variant methionine adenosyltransferase in rat ascitic hepatoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50228186(CHEMBL3706404)
Affinity DataKi:  1.10E+3nMAssay Description:Compound was tested for inhibition constant with kidney form of M-T variants of Rat methionine adenosyltransferase when Methionine was the variable s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367044(CHEMBL605639)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of AMP non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227271(CHEMBL1791425)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition constant of Met varied compound was measured on MT variant methionine adenosyltransferase in rat ascitic hepatoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50228186(CHEMBL3706404)
Affinity DataKi:  2.10E+3nMAssay Description:Compound was tested for inhibition constant with kidney form of M-2 variants of Rat methionine adenosyltransferase when Methionine was the variable s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227271(CHEMBL1791425)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition constant of Met varied compound was measured on M-2 variant methionine adenosyltransferase in rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227270(CHEMBL3706403)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition constant of Met varied compound was measured on M-2 variant methionine adenosyltransferase in rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50226768(CHEMBL1791426)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition constant of Met varied compound was measured on MT variant methionine adenosyltransferase in rat ascitic hepatoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50226770(CHEMBL609078)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition constant of compound with Novikoff ascitic hepatoma (M-T) form of rat methionine adenosyltransferase when methionine was used as variable ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50226972(CHEMBL606493)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition constants of MT Forms of rat Novikoff Ascitic Hepatomae using Methionine as the variable substrate; Inhibition is non competitive typeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50132297(1-((2R,4S,5R)-5-(aminomethyl)-4-hydroxy-tetrahydro...)
Affinity DataKi:  2.40E+3nMAssay Description:Competitive inhibition against rat cytoplasmic Thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50227270(CHEMBL3706403)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition constant of Met varied compound was measured on MT variant methionine adenosyltransferase in rat ascitic hepatoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50228185(CHEMBL3706405)
Affinity DataKi:  2.70E+3nMAssay Description:Compound was tested for inhibition constant with kidney form of M-T variants of Rat methionine adenosyltransferase when Methionine was the variable s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367044(CHEMBL605639)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1(Rattus norvegicus)
Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50368140(CHEMBL3706401 | CHEMBL611854)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition constants against ATP substrate site of M-T (Novikoff Ascitic Hepatoma form) variant of rat Methionine adenosyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50226770(CHEMBL609078)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition constant of compound with kidney (M-2) form of rat methionine adenosyltransferase when methionine was used as variable substrate;Simple no...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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