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Found 1550 with Last Name = 'kawatkar' and Initial = 's'
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84465(Benzylation of mannostatin A, 1e)
Affinity DataKi:  50nM ΔG°:  -43.3kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM50078117((1R,2R,3R,4S,5R)-4-AMINO-5-(METHYLTHIO)CYCLOPENTAN...)
Affinity DataKi:  90nM ΔG°:  -41.8kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84464(Benzylation of mannostatin A, 1d)
Affinity DataKi:  100nM ΔG°:  -41.6kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84466(Benzylation of mannostatin A, 1f)
Affinity DataKi:  100nM ΔG°:  -41.6kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84462(Benzylation of mannostatin A, 1b)
Affinity DataKi:  110nM ΔG°:  -41.3kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84467(Benzylation of mannostatin A, 1g)
Affinity DataKi:  140nM ΔG°:  -40.7kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84474(Aminocyclopentitetrol, 2g)
Affinity DataKi:  160nM ΔG°:  -40.3kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84463(Benzylation of mannostatin A, 1c)
Affinity DataKi:  170nM ΔG°:  -40.2kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM50078117((1R,2R,3R,4S,5R)-4-AMINO-5-(METHYLTHIO)CYCLOPENTAN...)
Affinity DataKi:  210nM ΔG°:  -39.6kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84470(Aminocyclopentitetrol, 2c)
Affinity DataKi:  330nM ΔG°:  -38.5kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84472(Aminocyclopentitetrol, 2e)
Affinity DataKi:  330nM ΔG°:  -38.5kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84469(Aminocyclopentitetrol, 2b)
Affinity DataKi:  450nM ΔG°:  -37.7kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84473(Aminocyclopentitetrol, 2f)
Affinity DataKi:  480nM ΔG°:  -37.5kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84465(Benzylation of mannostatin A, 1e)
Affinity DataKi:  510nM ΔG°:  -37.4kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84466(Benzylation of mannostatin A, 1f)
Affinity DataKi:  520nM ΔG°:  -37.3kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84463(Benzylation of mannostatin A, 1c)
Affinity DataKi:  530nM ΔG°:  -37.3kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84471(Aminocyclopentitetrol, 2d)
Affinity DataKi:  670nM ΔG°:  -36.7kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84462(Benzylation of mannostatin A, 1b)
Affinity DataKi:  880nM ΔG°:  -36.0kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84464(Benzylation of mannostatin A, 1d)
Affinity DataKi:  910nM ΔG°:  -35.9kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84467(Benzylation of mannostatin A, 1g)
Affinity DataKi:  3.22E+3nM ΔG°:  -32.6kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84474(Aminocyclopentitetrol, 2g)
Affinity DataKi:  4.40E+3nM ΔG°:  -31.8kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84470(Aminocyclopentitetrol, 2c)
Affinity DataKi:  6.00E+3nM ΔG°:  -31.0kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84473(Aminocyclopentitetrol, 2f)
Affinity DataKi:  6.60E+3nM ΔG°:  -30.8kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84468(Mannostatin analogue, 4b | Meso-aminocyclopentitet...)
Affinity DataKi:  6.60E+3nM ΔG°:  -30.8kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84472(Aminocyclopentitetrol, 2e)
Affinity DataKi:  7.60E+3nM ΔG°:  -30.4kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84471(Aminocyclopentitetrol, 2d)
Affinity DataKi:  8.10E+3nM ΔG°:  -30.2kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84469(Aminocyclopentitetrol, 2b)
Affinity DataKi:  1.00E+4nM ΔG°:  -29.7kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
University of Georgia

LigandPNGBDBM84468(Mannostatin analogue, 4b | Meso-aminocyclopentitet...)
Affinity DataKi:  5.00E+4nM ΔG°:  -25.5kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM138200(US8871778, 141)
Affinity DataIC50:  0.0300nMAssay Description:Inhibition of recombinant full length SYK (unknown origin) by biochemical Omnia assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50548361(CHEMBL4744190)
Affinity DataIC50:  0.0300nMAssay Description:Inhibition of recombinant full length SYK (unknown origin) by biochemical Omnia assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50548350(CHEMBL4780257)
Affinity DataIC50:  0.0600nMAssay Description:Inhibition of recombinant full length SYK (unknown origin) by biochemical Omnia assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50546397(CHEMBL4776352)
Affinity DataIC50:  0.0770nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50548354(CHEMBL4753469)
Affinity DataIC50:  0.0900nMAssay Description:Inhibition of recombinant full length SYK (unknown origin) by biochemical Omnia assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50546402(CHEMBL4762995)
Affinity DataIC50:  0.0980nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50548358(CHEMBL4753141)
Affinity DataIC50:  0.110nMAssay Description:Inhibition of recombinant full length SYK (unknown origin) by biochemical Omnia assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50548362(CHEMBL4784088)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of recombinant full length SYK (unknown origin) by biochemical Omnia assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50548357(CHEMBL4752008)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of recombinant full length SYK (unknown origin) by biochemical Omnia assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50546398(CHEMBL4754597)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50546401(CHEMBL4776842)
Affinity DataIC50:  0.170nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50546400(CHEMBL4752127)
Affinity DataIC50:  0.180nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50553519(CHEMBL4758052)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50548363(CHEMBL4753164)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of recombinant full length SYK (unknown origin) by biochemical Omnia assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50553510(CHEMBL4740533)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50548356(CHEMBL4792651)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant full length SYK (unknown origin) by biochemical Omnia assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50548351(CHEMBL4786316)
Affinity DataIC50:  0.210nMAssay Description:Inhibition of recombinant full length SYK (unknown origin) by biochemical Omnia assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50546394(CHEMBL4759636)
Affinity DataIC50:  0.210nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50546407(CHEMBL4740065)
Affinity DataIC50:  0.210nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50546407(CHEMBL4740065)
Affinity DataIC50:  0.210nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50548353(CHEMBL4762290)
Affinity DataIC50:  0.220nMAssay Description:Inhibition of recombinant full length SYK (unknown origin) by biochemical Omnia assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50553508(CHEMBL4797815)
Affinity DataIC50:  0.220nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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