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Found 12 with Last Name = 'kelleher' and Initial = 'd'
TargetGlucocorticoid receptor(Homo sapiens (Human))
Trinity College Dublin

Curated by ChEMBL
LigandPNGBDBM53721((4R)-4-[(3R,5S,7S,8R,9S,10S,13R,14S,17R)-10,13-dim...)
Affinity DataEC50:  2.99E+5nMAssay Description:Modulation of glucocorticoid receptor in human SKGT4 cells assessed as receptor translocation from cytoplasm to nucleus after 4 hrs by Hoechst staini...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Trinity College Dublin

Curated by ChEMBL
LigandPNGBDBM50334961(24-Cyclopropyl-3alpha,7beta-dihydroxy-5beta-cholan...)
Affinity DataEC50:  7.30E+3nMAssay Description:Modulation of glucocorticoid receptor in human SKGT4 cells assessed as receptor translocation from cytoplasm to nucleus after 4 hrs by Hoechst staini...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Trinity College Dublin

Curated by ChEMBL
LigandPNGBDBM50334962(24-N-Benzylpiperazine-3alpha,7beta-dihydroxy-5beta...)
Affinity DataEC50:  5.60E+3nMAssay Description:Modulation of glucocorticoid receptor in human SKGT4 cells assessed as receptor translocation from cytoplasm to nucleus after 4 hrs by Hoechst staini...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Trinity College Dublin

Curated by ChEMBL
LigandPNGBDBM50334951(24-piperazine-3alpha,7beta-dihydroxy-5beta-cholana...)
Affinity DataEC50:  5.08E+4nMAssay Description:Modulation of glucocorticoid receptor in human SKGT4 cells assessed as receptor translocation from cytoplasm to nucleus after 4 hrs by Hoechst staini...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Trinity College Dublin

Curated by ChEMBL
LigandPNGBDBM50334952(24-morpholine-3alpha,7beta-dihydroxy-5beta-cholana...)
Affinity DataEC50:  2.53E+4nMAssay Description:Modulation of glucocorticoid receptor in human SKGT4 cells assessed as receptor translocation from cytoplasm to nucleus after 4 hrs by Hoechst staini...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Trinity College Dublin

Curated by ChEMBL
LigandPNGBDBM50334959((S)-2-((3R,5S,7S,8R,9S,10S,13S,14S,17R)-3,7-dihydr...)
Affinity DataEC50:  9.97E+4nMAssay Description:Modulation of glucocorticoid receptor in human SKGT4 cells assessed as receptor translocation from cytoplasm to nucleus after 4 hrs by Hoechst staini...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Trinity College Dublin

Curated by ChEMBL
LigandPNGBDBM50334954(24-alpha-methylbenzyl-3alpha,7beta-dihydroxy-5beta...)
Affinity DataEC50:  1.24E+5nMAssay Description:Modulation of glucocorticoid receptor in human SKGT4 cells assessed as receptor translocation from cytoplasm to nucleus after 4 hrs by Hoechst staini...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Trinity College Dublin

Curated by ChEMBL
LigandPNGBDBM50334955(24-phenethyl-3alpha,7beta-dihydroxy-5beta-cholanam...)
Affinity DataEC50:  1.09E+5nMAssay Description:Modulation of glucocorticoid receptor in human SKGT4 cells assessed as receptor translocation from cytoplasm to nucleus after 4 hrs by Hoechst staini...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Trinity College Dublin

Curated by ChEMBL
LigandPNGBDBM50334956((R)-4-((3R,5S,7S,8R,9S,10S,13R,14S,17R)-3,7-dihydr...)
Affinity DataEC50:  1.01E+5nMAssay Description:Modulation of glucocorticoid receptor in human SKGT4 cells assessed as receptor translocation from cytoplasm to nucleus after 4 hrs by Hoechst staini...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Trinity College Dublin

Curated by ChEMBL
LigandPNGBDBM50334957((S)-2-((3R,5S,7S,8R,9S,10S,13R,14S,17R)-3,7-dihydr...)
Affinity DataEC50:  1.30E+5nMAssay Description:Modulation of glucocorticoid receptor in human SKGT4 cells assessed as receptor translocation from cytoplasm to nucleus after 4 hrs by Hoechst staini...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Trinity College Dublin

Curated by ChEMBL
LigandPNGBDBM50334958((R)-3-((3R,5S,7S,8R,9S,10S,13R,14S,17R)-3,7-dihydr...)
Affinity DataEC50:  1.05E+5nMAssay Description:Modulation of glucocorticoid receptor in human SKGT4 cells assessed as receptor translocation from cytoplasm to nucleus after 4 hrs by Hoechst staini...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Trinity College Dublin

Curated by ChEMBL
LigandPNGBDBM50334953(24-benzyl-3alpha,7beta-hydroxy-5beta-cholanamide |...)
Affinity DataEC50:  1.10E+5nMAssay Description:Modulation of glucocorticoid receptor in human SKGT4 cells assessed as receptor translocation from cytoplasm to nucleus after 4 hrs by Hoechst staini...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed