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Found 357 with Last Name = 'kiss' and Initial = 'r'
TargetHistamine H4 receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM22911(2-(3H-imidazol-4-yl)ethylsulfanylmethanimidamide |...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SK-NM-C cellsMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM22541(Clobenpropit | N''-[(4-chlorophenyl)methyl]{[3-(1H...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SK-NM-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM22913(CHEMBL1237146 | CHEMBL498770 | Iodophenpropit | {[...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SK-NM-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM7966(2-(1H-imidazol-4-yl)ethan-1-amine | CHEMBL544208 |...)
Affinity DataKi:  13.4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SK-NM-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistamine H4 receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM22566(5-chloro-2-[(4-methylpiperazin-1-yl)carbonyl]-1H-i...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SK-NM-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268759(CHEMBL496032 | N-butyl-2-chloro-N-(2-(4-(4-chlorop...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268683(CHEMBL496812 | N-butyl-2-chloro-N-(2-(4-(4-methoxy...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268633(CHEMBL498425 | N-butyl-N-(2-(4-(4-methoxyphenyl)py...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50261080(N-(amino(4,6-dimethylpyrimidin-2-ylamino)methylene...)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SK-NM-C cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM22883(CHEMBL12344 | Dimaprit | [3-(carbamimidoylsulfanyl...)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SK-NM-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408099(CHEMBL57087)
Affinity DataKi:  120nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268634(CHEMBL498627 | N-butyl-N-(2-(4-(4-methoxyphenyl)py...)
Affinity DataKi:  124nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268514(CHEMBL522247 | N-butyl-2-chloro-N-(2-(4-(4-methoxy...)
Affinity DataKi:  137nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408102(CHEMBL55646)
Affinity DataKi:  150nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268758(CHEMBL495836 | N-butyl-2-chloro-N-(2-(4-(4-fluorop...)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM22904((2R)-1-(1H-imidazol-5-yl)propan-2-amine | (R)-alph...)
Affinity DataKi:  184nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SK-NM-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408104(CHEMBL292238)
Affinity DataKi:  200nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268632(CHEMBL498424 | N-butyl-N-(2-(4-(4-methoxyphenyl)py...)
Affinity DataKi:  214nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50261081([amino({2-[(1Z)-4-{[4-(ethoxycarbonyl)phenyl]amino...)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SK-NM-C cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268454(2-chloro-N-isopropyl-N-(2-(4-(4-methoxyphenyl)pyrr...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408110(CHEMBL293284)
Affinity DataKi:  220nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268569(CHEMBL496596 | N-butyl-N-(2-(4-(4-methoxyphenyl)py...)
Affinity DataKi:  236nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268721(CHEMBL496221 | N-butyl-2-chloro-N-(2-oxo-2-(4-phen...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  328nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SK-NM-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268568(CHEMBL521738 | N-butyl-2-fluoro-N-(2-(4-(4-methoxy...)
Affinity DataKi:  349nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408096(CHEMBL301025)
Affinity DataKi:  350nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408101(CHEMBL293519)
Affinity DataKi:  370nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408094(CHEMBL59256)
Affinity DataKi:  390nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268682(CHEMBL496207 | N-butyl-2-methoxy-N-(2-(4-(4-methox...)
Affinity DataKi:  461nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268567(CHEMBL497006 | N-butyl-N-(2-(4-(4-methoxyphenyl)py...)
Affinity DataKi:  503nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268681(CHEMBL521717 | N-butyl-N-(2-(4-(4-methoxyphenyl)py...)
Affinity DataKi:  539nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408105(CHEMBL294146)
Affinity DataKi:  550nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408100(CHEMBL57674)
Affinity DataKi:  570nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268570(CHEMBL496597 | N-butyl-N-(2-(4-(4-methoxyphenyl)py...)
Affinity DataKi:  602nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408103(CHEMBL293294)
Affinity DataKi:  790nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268513(CHEMBL526749 | N-butyl-3,5-dichloro-N-(2-(4-(4-met...)
Affinity DataKi:  831nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50261079((4Z,6E)-2,10-diamino-5,7-dimethyl-1,3,4,8,9,11-hex...)
Affinity DataKi:  897nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SK-NM-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50261037([amino({[6-({[amino(iminiumyl)methyl]amino}methyl)...)
Affinity DataKi:  1.24E+3nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SK-NM-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50261036((E)-{amino[(Z)-2-(1-{12-[(1Z)-1-(2-methylcarbamimi...)
Affinity DataKi:  1.48E+3nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SK-NM-C cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408107(CHEMBL56789)
Affinity DataKi:  6.50E+3nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408097(CHEMBL56270)
Affinity DataKi:  7.20E+3nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408109(CHEMBL54055)
Affinity DataKi:  8.40E+3nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408106(CHEMBL56927)
Affinity DataKi:  1.40E+4nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408098(CHEMBL298828)
Affinity DataKi:  2.40E+4nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408095(CHEMBL292166)
Affinity DataKi:  6.70E+4nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408108(CHEMBL299276)
Affinity DataKi:  8.30E+4nMAssay Description:Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Texas State University-San Marcos

Curated by ChEMBL
LigandPNGBDBM50434372(CHEMBL2386889)
Affinity DataIC50:  3nMAssay Description:Competitive inhibition of recombinant His-tagged CHK1 (unknown origin) expressed in baculovirus expression system using CDC25C and ATP as substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50216416(1-(4-bromo-benzyl)-5-[2-(pyridin-3-yl-oxymethyl)-p...)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of human recombinant caspase 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50216421(1-(4-hydroxy-benzyl)-5-[2-(pyridin-3-yl-oxymethyl)...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of human recombinant caspase 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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