TargetNeuromedin-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by PDSP Ki Database
Schering-Plough Research Institute
Curated by PDSP Ki Database
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by PDSP Ki Database
Schering-Plough Research Institute
Curated by PDSP Ki Database
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by PDSP Ki Database
Schering-Plough Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 0.800nMAssay Description:Binding afinity against Histamine H3 receptorMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by PDSP Ki Database
Schering-Plough Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 1.5nMAssay Description:Binding affinity of compound towards Histamine H3 receptor was determined in guinea pig brain tissue using [3H]- N alpha-methylhistamine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding afinity against Histamine H3 receptorMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by PDSP Ki Database
Schering-Plough Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Inhibition of [3H]-N-alpha-methylhistamine binding to guinea pig brain Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Inhibition of [3H]-N-alpha-methylhistamine binding to guinea pig brain Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding afinity against Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding afinity against Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of [3H]-N-alpha-methylhistamine binding to guinea pig brain Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of [3H]-N-alpha-methylhistamine binding to guinea pig brain Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of [3H]-N-alpha-methylhistamine binding to guinea pig brain Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of [3H]-N-alpha-methylhistamine binding to guinea pig brain Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding afinity against Histamine H3 receptorMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by PDSP Ki Database
Schering-Plough Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 21nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Binding afinity against Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Inhibition of [3H]-N-alpha-methylhistamine binding to guinea pig brain Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Inhibition of [3H]-N-alpha-methylhistamine binding to guinea pig brain Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Inhibition of [3H]-N-alpha-methylhistamine binding to guinea pig brain Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibition of [3H]-N-alpha-methylhistamine binding to guinea pig brain Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by PDSP Ki Database
Schering-Plough Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 290nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by PDSP Ki Database
Schering-Plough Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 320nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 720nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 740nMAssay Description:Binding afinity against Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by PDSP Ki Database
Schering-Plough Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 1.50E+3nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of [3H]-N-alpha-methylhistamine binding to guinea pig brain Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of [3H]-N-alpha-methylhistamine binding to guinea pig brain Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:Binding afinity against Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:Binding afinity against Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair