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Found 124 with Last Name = 'krobert' and Initial = 'ka'
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483188(CHEMBL1632166)
Affinity DataKi:  0.00145nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483175(CHEMBL1632165)
Affinity DataKi:  0.0427nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50327858((1-Butylpiperidin-4-yl)methyl 8-amino-7-iodo-2,3-d...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM85026(N-(1-Butylpiperidine-4-ylmethyl)-1,2-(trimethylene...)
Affinity DataKi:  0.0525nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483174(CHEMBL1632163)
Affinity DataKi:  0.0537nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483187(CHEMBL1632169)
Affinity DataKi:  0.0646nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.0741nMAssay Description:Antagonistic activity at human 5HT4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50327858((1-Butylpiperidin-4-yl)methyl 8-amino-7-iodo-2,3-d...)
Affinity DataKi:  0.0790nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.0790nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483173(CHEMBL1632157)
Affinity DataKi:  0.102nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483172(CHEMBL1632158)
Affinity DataKi:  0.107nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483186(CHEMBL1632167)
Affinity DataKi:  0.141nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483171(CHEMBL1632159)
Affinity DataKi:  0.195nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483191(CHEMBL1632162)
Affinity DataKi:  0.234nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483169(CHEMBL1632160)
Affinity DataKi:  0.339nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483170(CHEMBL1632168)
Affinity DataKi:  0.339nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483182(CHEMBL1632161)
Affinity DataKi:  0.759nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483178(CHEMBL1632154)
Affinity DataKi:  0.813nMAssay Description:Antagonistic activity at human 5HT4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483184(CHEMBL1632171)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM85778(CAS_135938-17-9 | SB203186)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483181(CHEMBL1632164)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483176(CHEMBL1632174)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483183(CHEMBL1632172)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM85778(CAS_135938-17-9 | SB203186)
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483180(CHEMBL1632173)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483177(CHEMBL1632175)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483190(CHEMBL1632170)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483189(CHEMBL1632176)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50005836(4-Amino-5-chloro-N-{1-[3-(4-fluoro-phenoxy)-propyl...)
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50005836(4-Amino-5-chloro-N-{1-[3-(4-fluoro-phenoxy)-propyl...)
Affinity DataKi:  50.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50007871(CHEMBL8197 | ICS 205-930 | TROPISETRON)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483185(CHEMBL1632155)
Affinity DataKi:  107nMAssay Description:Antagonistic activity at human 5HT4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50007871(CHEMBL8197 | ICS 205-930 | TROPISETRON)
Affinity DataKi:  158nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataKi:  159nMMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM82422(CAS_109872-41-5 | NSC_3035240 | RENZAPRIDE)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM82087(2-(5-methoxy-1H-indol-3-yl)ethanamine | 5-MT | 5-M...)
Affinity DataKi:  251nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM82422(CAS_109872-41-5 | NSC_3035240 | RENZAPRIDE)
Affinity DataKi:  251nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483172(CHEMBL1632158)
Affinity DataKi:  316nMAssay Description:Binding affinity to 5HT2B receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM82087(2-(5-methoxy-1H-indol-3-yl)ethanamine | 5-MT | 5-M...)
Affinity DataKi:  316nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483172(CHEMBL1632158)
Affinity DataKi:  398nMAssay Description:Binding affinity to opioid receptor Sigma1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483172(CHEMBL1632158)
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity to alpha2B adrenergic receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483172(CHEMBL1632158)
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity to Histamine receptor H1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483172(CHEMBL1632158)
Affinity DataKi:  2.51E+3nMAssay Description:Binding affinity to muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483172(CHEMBL1632158)
Affinity DataKi:  2.51E+3nMAssay Description:Binding affinity to 5HT3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483172(CHEMBL1632158)
Affinity DataKi:  3.16E+3nMAssay Description:Binding affinity to Histamine receptor H2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483172(CHEMBL1632158)
Affinity DataKi:  3.16E+3nMAssay Description:Binding affinity to 5HT1D receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483179(CHEMBL1632156)
Affinity DataKi:  3.63E+3nMAssay Description:Antagonistic activity at human 5HT4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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