Compile Data Set for Download or QSAR
maximum 50k data
Found 182 with Last Name = 'li' and Initial = 'wp'
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50291847(7-[3-(Quinolin-2-ylmethoxy)-benzyloxy]-2-(1H-tetra...)
Affinity DataKi:  0.100nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50291855(7-[3-(Quinolin-2-ylmethoxy)-phenoxymethyl]-2-(1H-t...)
Affinity DataKi:  0.120nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50009075(CHEMBL22033 | ICI 198615 | ICI-198615 | [1-(4-Benz...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50291848(7-{2-[3-(Quinolin-2-ylmethoxy)-phenyl]-ethyl}-2-(1...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50291849(CHEMBL47662 | N-[4-Oxo-2-(1H-tetrazol-5-yl)-chroma...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50291850(3-{2-Methyl-4-oxo-7-[3-(quinolin-2-ylmethoxy)-benz...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50291854(4-Oxo-6-[3-(quinolin-2-ylmethoxy)-benzyloxy]-chrom...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13304(4-hydroxy-3-[((3S)-2-oxo-3-{[(5-pyridin-3-ylthien-...)
Affinity DataKi:  2nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50291856(4-Oxo-7-[3-(quinolin-2-ylmethoxy)-benzyloxy]-chrom...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50291858(7-{2-[3-(Quinolin-2-ylmethoxy)-phenyl]-vinyl}-2-(1...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13306(4-Hydroxy-3-[3-(S)-(5-isoxazol-3-ylthiophene-2-yls...)
Affinity DataKi:  3nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13286(4-Hydroxy-3-[3-(S)-(7-methoxynaphthalen-2-ylsulfon...)
Affinity DataKi:  3nM ΔG°:  -48.2kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50006799(2-{4-[2-(1H-Tetrazol-5-ylmethyl)-benzyloxy]-phenox...)
Affinity DataKi:  3nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13283(4-amino-3-({(3S)-3-[[(7-methoxy-2-naphthyl)sulfony...)
Affinity DataKi:  4nM ΔG°:  -47.5kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13281(4-Amino-3-[3-(S)-(7-methoxynaphthalen-2-ylsulfonyl...)
Affinity DataKi:  6nM ΔG°:  -46.5kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13303(4-Amino-3-[2-oxo-3-(S)-(5-pyridin-3-ylthiophene-2-...)
Affinity DataKi:  6nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50291853(4-Oxo-7-[4-(quinolin-2-ylmethoxy)-phenoxymethyl]-c...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13279(4-{[(3S)-3-[(7-methoxynaphthalene-2-)(methyl)sulfo...)
Affinity DataKi:  6.90nM ΔG°:  -46.1kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13305(4-Amino-3-[3-(S)-(5-isoxazol-3-ylthiophene-2-ylsul...)
Affinity DataKi:  7nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13288(Sulfonamidopyrrolidinone 27 | methyl 2-(4-carbamim...)
Affinity DataKi:  8nM ΔG°:  -45.7kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Rhone-Poulenc Rorer

LigandPNGBDBM13288(Sulfonamidopyrrolidinone 27 | methyl 2-(4-carbamim...)
Affinity DataKi:  12nM ΔG°:  -44.8kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50291859(4-Oxo-8-[4-(quinolin-2-ylmethoxy)-phenoxymethyl]-c...)
Affinity DataKi:  13nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50291851(8-[4-(Quinolin-2-ylmethoxy)-phenoxymethyl]-2-(1H-t...)
Affinity DataKi:  15nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50291857(6-Chloro-4-oxo-5-[4-(quinolin-2-ylmethoxy)-benzylo...)
Affinity DataKi:  18nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13282(3-{[(3S)-3-[(7-methoxynaphthalene-2-)(methyl)sulfo...)
Affinity DataKi:  22nM ΔG°:  -43.3kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50296936(16-[(3-Fluorophenyl)methylidene]-17beta-hydroxy-4-...)
Affinity DataKi:  29nMAssay Description:Binding affinity to human ERG potassium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50291852(4-Oxo-7-[3-(quinolin-2-ylmethoxy)-phenoxymethyl]-c...)
Affinity DataKi:  30nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13298(3-[2-Oxo-3-(S)-(5-pyridin-3-ylthiophene-2-ylsulfon...)
Affinity DataKi:  41nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50296937(16-[(3,5-Difluorophenyl)methylidene]-17beta-hydrox...)
Affinity DataKi:  46nMAssay Description:Binding affinity to human ERG potassium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13280(3-{[(3S)-3-[(7-methoxynaphthalene-2-)sulfonamido]-...)
Affinity DataKi:  47nM ΔG°:  -41.4kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13301(3-[3-(S)-(5-Isoxazol-3-ylthiophene-2-ylsulfonylami...)
Affinity DataKi:  49nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13299(3-[2-Oxo-3-(S)-(5-pyridin-4-ylthiophene-2-ylsulfon...)
Affinity DataKi:  55nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13302(4-fluoro-3-[((3S)-2-oxo-3-{[(5-pyridin-3-ylthien-2...)
Affinity DataKi:  130nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13293(3-{[(3S)-2-oxo-3-{[4-(pyridin-4-yl)benzene]sulfona...)
Affinity DataKi:  130nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13297(3-{[(3S)-2-oxo-3-{[5-(pyridin-2-yl)thiophene-2-]su...)
Affinity DataKi:  140nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13300(3-{[(3S)-3-{[5-(2-methoxypyrimidin-4-yl)thiophene-...)
Affinity DataKi:  150nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13291(3-{[(3S)-2-oxo-3-{[4-(pyridin-2-yl)benzene]sulfona...)
Affinity DataKi:  150nM ΔG°:  -38.6kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13290(3-{[(3S)-2-oxo-3-[(4-phenylbenzene)sulfonamido]pyr...)
Affinity DataKi:  160nM ΔG°:  -38.4kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Rhone-Poulenc Rorer

LigandPNGBDBM13283(4-amino-3-({(3S)-3-[[(7-methoxy-2-naphthyl)sulfony...)
Affinity DataKi:  189nM ΔG°:  -38.0kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13292(3-{[(3S)-2-oxo-3-{[4-(pyridin-3-yl)benzene]sulfona...)
Affinity DataKi:  210nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50296938(16-(Phenylmethylidene)-17beta-hydroxy-4-methyl-4-a...)
Affinity DataKi:  225nMAssay Description:Binding affinity to human ERG potassium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50296935(16alpha-(3-Fluorobenzyl)-17beta-hydroxy-4-methyl-4...)
Affinity DataKi:  240nMAssay Description:Binding affinity to human ERG potassium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Rhone-Poulenc Rorer

LigandPNGBDBM13281(4-Amino-3-[3-(S)-(7-methoxynaphthalen-2-ylsulfonyl...)
Affinity DataKi:  299nM ΔG°:  -36.9kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Rhone-Poulenc Rorer

LigandPNGBDBM13286(4-Hydroxy-3-[3-(S)-(7-methoxynaphthalen-2-ylsulfon...)
Affinity DataKi:  305nM ΔG°:  -36.8kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50296941(16-(Pyridin-4-ylmethylidene)-17beta-hydroxy-4-meth...)
Affinity DataKi:  320nMAssay Description:Binding affinity to human ERG potassium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13295(4-(4-{[(3S)-1-[(3-carbamimidoylphenyl)methyl]-2-ox...)
Affinity DataKi:  330nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50006812(7-[3-(4-Acetyl-3-hydroxy-2-propyl-phenoxy)-2-hydro...)
Affinity DataKi:  510nMAssay Description:Binding affinity against LTD4 receptor in guinea pig lung membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Rhone-Poulenc Rorer

LigandPNGBDBM13282(3-{[(3S)-3-[(7-methoxynaphthalene-2-)(methyl)sulfo...)
Affinity DataKi:  704nM ΔG°:  -34.8kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Rhone-Poulenc Rorer

LigandPNGBDBM13280(3-{[(3S)-3-[(7-methoxynaphthalene-2-)sulfonamido]-...)
Affinity DataKi:  853nM ΔG°:  -34.3kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Rhone-Poulenc Rorer

LigandPNGBDBM13284(N-(4-carbamimidoyl-2-{[(3S)-3-[(7-methoxynaphthale...)
Affinity DataKi:  919nM ΔG°:  -34.1kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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