Compile Data Set for Download or QSAR
maximum 50k data
Found 37 with Last Name = 'li' and Initial = 'yn'
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577060(SIGA-246 | ST 246 | ST-246 | Tecovirimat | Tpoxx)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM8610(1-[4-(4-{[(2R,4S)-2-(2,4-dichlorophenyl)-2-(1H-imi...)
Affinity DataIC50:  65nMAssay Description:Inhibition of recombinant human CYP3A4 in presence of NADPH generating system by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577042(CHEMBL4864184)
Affinity DataIC50:  133nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577048(CHEMBL4867155)
Affinity DataIC50:  216nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577045(CHEMBL4871145)
Affinity DataIC50:  270nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577057(CHEMBL4878636)
Affinity DataIC50:  515nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577049(CHEMBL4850454)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataIC50:  1.65E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization incubated for 60 mins by fluorescence-based assayMore data for this Ligand-Target Pair
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577058(CHEMBL4872088)
Affinity DataIC50:  1.66E+3nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology

Curated by ChEMBL
LigandPNGBDBM50421320(CHEMBL2088175)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of MerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology

Curated by ChEMBL
LigandPNGBDBM50421321(CHEMBL2088176)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of MerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  2.48E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization incubated for 60 mins by fluorescence-based assayMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50101086(CHEMBL20684 | E-7010 | N-(2-(4-hydroxyphenylamino)...)
Affinity DataIC50:  2.79E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization incubated for 60 mins by fluorescence-based assayMore data for this Ligand-Target Pair
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577054(CHEMBL4857491)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology

Curated by ChEMBL
LigandPNGBDBM50421322(CHEMBL2088178)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of MerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577047(CHEMBL4865942)
Affinity DataIC50:  3.06E+3nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577055(CHEMBL4852852)
Affinity DataIC50:  3.52E+3nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577043(CHEMBL4879134)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50533422(CHEMBL4465886)
Affinity DataIC50:  4.62E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization incubated for 60 mins by fluorescence-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577044(CHEMBL4877767)
Affinity DataIC50:  4.85E+3nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50533423(CHEMBL4448192)
Affinity DataIC50:  5.33E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization incubated for 60 mins by fluorescence-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM81939(CAS_52-53-9 | NSC_62969 | VERAPAMIL)
Affinity DataIC50:  8.19E+3nMAssay Description:Inhibition of recombinant human CYP3A4 in presence of NADPH generating system by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577046(CHEMBL4860346)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577059(CHEMBL4856490)
Affinity DataIC50:  8.98E+3nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology

Curated by ChEMBL
LigandPNGBDBM50421320(CHEMBL2088175)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AxlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology

Curated by ChEMBL
LigandPNGBDBM50421322(CHEMBL2088178)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AxlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577056(CHEMBL4853135)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577051(CHEMBL4865823)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50288831(CHEMBL4161738)
Affinity DataIC50:  1.72E+4nMAssay Description:Inhibition of recombinant human CYP3A4 in presence of NADPH generating system by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology

Curated by ChEMBL
LigandPNGBDBM50421321(CHEMBL2088176)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Tyro3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology

Curated by ChEMBL
LigandPNGBDBM50421322(CHEMBL2088178)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Tyro3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology

Curated by ChEMBL
LigandPNGBDBM50421321(CHEMBL2088176)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of AxlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology

Curated by ChEMBL
LigandPNGBDBM50421320(CHEMBL2088175)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Tyro3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577050(CHEMBL4873414)
Affinity DataIC50:  3.09E+4nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577052(CHEMBL4866978)
Affinity DataIC50:  3.63E+4nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable maltase-glucoamylase 2(Homo sapiens)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50236527((-)-catechin | (2S,3R)-2-(3,4-dihydroxyphenyl)-3,4...)
Affinity DataIC50:  5.38E+4nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl beta-D-glucopyranoside as substrate measured after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope phospholipase F13(Vaccinia virus (strain Western Reserve) (VACV) (Va...)
Samara State Technical University

Curated by ChEMBL
LigandPNGBDBM50577053(CHEMBL4876679)
Affinity DataIC50:  1.98E+5nMAssay Description:Inhibition of p37 in Vaccinia virus Copenhagen infected in African green monkey Vero cells assessed as reduction in viral reproduction incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed