Affinity DataKi: 2.70E+4nMAssay Description:Competitive inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 5.06E+4nMAssay Description:Competitive inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of chymotrypsin-like activity of Proteasome subunit beta 5 (unknown origin) assessed as inhibition of beta-amyloid production by cell-base...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibitory concentration against calf tubulin polymerizationMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of recombinant human HGK using Ulight-FLGFTYVAP as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibitory concentration against calf tubulin polymerizationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibitory concentration against calf tubulin polymerizationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: 3.35E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of recombinant human HGK using Ulight-FLGFTYVAP as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase activities were assayed according to the methodology developed by the Cell Cycle Group of the Station Biologique (CNRS).More data for this Ligand-Target Pair
Affinity DataIC50: 5.57E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.20E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.09E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.39E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.59E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human HGK using Ulight-FLGFTYVAP as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human HGK using Ulight-FLGFTYVAP as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human HGK using Ulight-FLGFTYVAP as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human HGK using Ulight-FLGFTYVAP as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+5nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair