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Found 73 with Last Name = 'little' and Initial = 's'
TargetGenome polyprotein(Human rhinovirus B)
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065621(CHEMBL94688 | [(S)-1-((S)-1-{(S)-3-Carbamoyl-1-[2-...)
Affinity DataKi:  30nMAssay Description:Catalytic rate constant (Kobs/[I]) of the compound was evaluated against human rhinovirus (HRV) serotype 14 3C Protease (3CP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288762((1S,10R)-14-[2-Oxo-2-(3,4,5-trimethoxy-phenyl)-ace...)
Affinity DataKi:  280nMAssay Description:Compound was evaluated for inhibitory activity against human FKBP-12 rotamaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288763((1S,9R)-5-Benzyloxymethyl-13-[2-oxo-2-(3,4,5-trime...)
Affinity DataKi:  1.20E+3nMAssay Description:Compound was evaluated for inhibitory activity against human FKBP-12 rotamaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288765((1S,9R)-5-(tert-Butyl-dimethyl-silanyloxymethyl)-1...)
Affinity DataKi:  1.50E+3nMAssay Description:Compound was evaluated for inhibitory activity against human FKBP-12 rotamaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288764((1S,9R)-13-[2-((1S,2R,5R)-1-Hydroxy-5-isopropyl-2-...)
Affinity DataKi:  8.10E+3nMAssay Description:Compound was evaluated for inhibitory activity against human FKBP-12 rotamaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288768((1R,10S)-14-(3,3-Dimethyl-2-oxo-pentanoyl)-3,8-dio...)
Affinity DataKi:  8.30E+3nMAssay Description:Compound was evaluated for inhibitory activity against human FKBP-12 rotamaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288767((1R,9S)-13-(3,3-Dimethyl-2-oxo-pentanoyl)-3,7-diox...)
Affinity DataKi:  1.00E+4nMAssay Description:Compound was evaluated for inhibitory activity against human FKBP-12 rotamaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288766((1S,9R)-13-{2-[(1S,2R,5R)-1-Hydroxy-5-(2-methoxy-1...)
Affinity DataKi: >5.00E+4nMAssay Description:Compound was evaluated for inhibitory activity against human FKBP-12 rotamaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288769((S)-1-[2-((1S,2R,5R)-1-Hydroxy-5-isopropyl-2-methy...)
Affinity DataKi:  2.10E+5nMAssay Description:Compound was evaluated for inhibitory activity against human FKBP-12 rotamaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195627(22,26-azasterol | CHEMBL425634)
Affinity DataIC50:  28nMAssay Description:Inhibition of Leishmania major recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50084636(5-[1-[4-(4-Benzoyl-3-hydroxy-2-propyl-benzyloxy)-p...)
Affinity DataIC50:  210nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50080991(5-[1-[4-(4-Benzoyl-3-hydroxy-2-propyl-phenoxymethy...)
Affinity DataIC50:  340nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287763(5-[1-{4-[3-Hydroxy-4-(2-hydroxy-benzoyl)-2-propyl-...)
Affinity DataIC50:  620nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287749(5-[1-[4-(4-Acetyl-3-hydroxy-2-propyl-benzyloxy)-ph...)
Affinity DataIC50:  640nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287758(5-(2-Hydroxy-4-{4-[4-oxo-2-thioxo-thiazolidin-(5Z)...)
Affinity DataIC50:  690nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287743(5-[1-[4-(4-Benzoyl-phenoxymethyl)-phenyl]-meth-(Z)...)
Affinity DataIC50:  780nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287747(5-[1-[4-(4-Benzoyl-2-benzyl-3-hydroxy-phenoxymethy...)
Affinity DataIC50:  820nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50080991(5-[1-[4-(4-Benzoyl-3-hydroxy-2-propyl-phenoxymethy...)
Affinity DataIC50:  1.30E+3nMAssay Description:Compound was evaluated for the inhibition of cathepsin D at an enzyme level of 50 ng/mLMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287761(5-[1-[4-(4-Benzoyl-benzyloxy)-phenyl]-meth-(Z)-yli...)
Affinity DataIC50:  1.31E+3nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287759(5-[1-{4-[3-Hydroxy-2-propyl-4-(pyridine-3-carbonyl...)
Affinity DataIC50:  1.46E+3nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195627(22,26-azasterol | CHEMBL425634)
Affinity DataIC50:  1.76E+3nMAssay Description:Inhibition of Trypanosoma brucei brucei recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287742(5-[1-[4-(4-Acetyl-3-methoxy-2-propyl-benzyloxy)-ph...)
Affinity DataIC50:  1.86E+3nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287750(5-[1-[4-(4-Acetyl-3-hydroxy-2-propyl-phenoxymethyl...)
Affinity DataIC50:  2.56E+3nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287757(5-[1-[4-(3-Methoxy-2-propyl-phenoxymethyl)-phenyl]...)
Affinity DataIC50:  2.76E+3nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287762(5-[1-[4-(3-Hydroxy-2-propyl-phenoxymethyl)-phenyl]...)
Affinity DataIC50:  2.94E+3nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287752(Acetic acid 6-acetyl-3-{4-[4-oxo-2-thioxo-thiazoli...)
Affinity DataIC50:  2.98E+3nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287745(5-[1-[4-(3-Hydroxy-4-propionyl-2-propyl-benzyloxy)...)
Affinity DataIC50:  3.69E+3nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195636(3beta-ol-23,24-bisnor-5-en-22-(butanoic acid) amin...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Leishmania major recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287760(2-Hydroxy-4-{4-[4-oxo-2-thioxo-thiazolidin-(5Z)-yl...)
Affinity DataIC50:  5.13E+3nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287751(5-[1-[3-(4-Acetyl-3-hydroxy-2-propyl-benzyloxy)-ph...)
Affinity DataIC50:  6.64E+3nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287753(5-[1-[4-(4-Benzoyl-3-hydroxy-phenoxymethyl)-phenyl...)
Affinity DataIC50:  7.20E+3nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287748(5-[1-{4-[3-Hydroxy-2-propyl-4-(pyridine-4-carbonyl...)
Affinity DataIC50:  7.94E+3nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287746(2-Hydroxy-4-{4-[4-oxo-2-thioxo-thiazolidin-(5Z)-yl...)
Affinity DataIC50:  9.74E+3nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287755(5-[1-[4-(4-Acetyl-3-hydroxy-benzyloxy)-phenyl]-met...)
Affinity DataIC50:  1.41E+4nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287754(5-[1-[4-(4-Acetyl-2-ethyl-3-hydroxy-benzyloxy)-phe...)
Affinity DataIC50:  1.76E+4nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287744(Acetic acid 6-acetyl-3-{4-[4-oxo-2-thioxo-thiazoli...)
Affinity DataIC50:  3.30E+4nMAssay Description:Compound was evaluated for the inhibition of cathepsin D at concentration of 4.15 microg/mLMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287756(5-[1-[4-(4-Acetyl-3-methoxy-2-propyl-phenoxymethyl...)
Affinity DataIC50:  4.84E+4nMAssay Description:In vitro inhibition of cathepsin D.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195640(3beta-ol-23,24-bisnor-5-en-22-(pentanoic acid) ami...)
Affinity DataIC50:  4.89E+4nMAssay Description:Inhibition of Leishmania major recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195646(3beta-ol-23,24-bisnor-5-en-22-(pentanoic acid) ami...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Leishmania major recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195642(3beta-acetoxy-23,24-bisnor-chol-5-en-22-(methyl bu...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma brucei brucei recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195649(3beta-ol-23,24-bisnor-5-en-22-(hexanoic acid) amin...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Leishmania major recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195651(3beta-acetoxy-23,24-bisnor-chol-5-en-22-(hexanoic ...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Leishmania major recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195653(3beta-ol-23,24-bisnor-5-en-22-(ethanoic acid) amid...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Leishmania major recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195652(3beta-ol-23,24-bisnor-5-en-22-(5-(2-Z-amino)pentan...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Leishmania major recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195654(3beta-acetoxy-23,24-bisnor-5-en-22-(4-(2-Boc-amino...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Leishmania major recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195621(3beta-acetoxy-23,24-bisnor-chol-5-en-22-(methyl he...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Leishmania major recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195645(3beta-ol-23,24-bisnor-5-en-22-(octanoic acid) amid...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Leishmania major recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195644(3beta-ol-23,24-bisnor-5-en-22-(6-(2-amino) hexanoa...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Leishmania major recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195647(3beat-ol-23,24-bisnor-5-en-22-(6-(2-Z-amino) hexan...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Leishmania major recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCycloartenol-C-24-methyltransferase(Arabidopsis thaliana)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50195650(3beta-acetoxy-23,24-bisnor-5-en-22-(3-(2-Boc-amino...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Leishmania major recombinant 24-SMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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