Affinity DataIC50: 367nMAssay Description:Inhibition of human HDAC4 catalytic domain (residues Thr648-Thr1057) expressed in Escherichia coli BL21using fluorogenic substrate by fluorescence as...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of HDAC8 assessed as substrate deacetylation using N-acetyl-L-Arg-LHis-L-Lys(epsilon-acetyl)-L-Lys(epsilon-acetyl)-coumarin as substrate p...More data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
Drexel University
Curated by ChEMBL
Drexel University
Curated by ChEMBL
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of Mycoplana ramosa acetylpolyamine amidohydrolase assessed as substrate deacetylation using L-Lys(epsilon-acetyl)-coumarin as substrate p...More data for this Ligand-Target Pair
Affinity DataKd: 6.00E+4nMAssay Description:Displacement of [14C-guanidino]-L-arginine from human recombinant full length arginase 1 expressed in Escherichia coli BL21(DE3) by fixed point assayMore data for this Ligand-Target Pair