Compile Data Set for Download or QSAR
maximum 50k data
Found 182 with Last Name = 'lopes' and Initial = 'jp'
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608244(CHEMBL5271306)
Affinity DataKi:  50nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataKi:  500nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataKi:  500nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataKi:  540nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM11682(2,3-dihydroxybutanedioic acid; 3-[(1S)-1-(dimethyl...)
Affinity DataKi:  700nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608255(CHEMBL5272999)
Affinity DataKi:  1.73E+3nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608233(CHEMBL5268833)
Affinity DataKi:  1.76E+3nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constant by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608259(CHEMBL5267382)
Affinity DataKi:  3.10E+3nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608257(CHEMBL5266593)
Affinity DataKi:  3.53E+3nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608248(CHEMBL5273862)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608245(CHEMBL5273571)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608248(CHEMBL5273862)
Affinity DataKi:  4.20E+3nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608245(CHEMBL5273571)
Affinity DataKi:  4.30E+3nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608259(CHEMBL5267382)
Affinity DataKi:  5.40E+3nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608254(CHEMBL5274058)
Affinity DataKi:  6.61E+3nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608246(CHEMBL5285312)
Affinity DataKi:  7.10E+3nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataKi:  9.37E+3nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataKi:  9.40E+3nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608252(CHEMBL5271574)
Affinity DataKi:  9.50E+3nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608258(CHEMBL5287680)
Affinity DataKi:  9.69E+3nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608238(CHEMBL5279849)
Affinity DataKi:  1.48E+4nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))TBA
LigandPNGBDBM50608225(CHEMBL5282473)
Affinity DataKi:  1.60E+4nMAssay Description:Binding affinity to horse serum BuChE using ATCh-iodide as substrate by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608240(CHEMBL5273719)
Affinity DataKi:  1.87E+4nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608247(CHEMBL5279226)
Affinity DataKi:  2.29E+4nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608237(CHEMBL5271146)
Affinity DataKi:  2.37E+4nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))TBA
LigandPNGBDBM50608227(CHEMBL5287005)
Affinity DataKi:  2.60E+4nMAssay Description:Binding affinity to horse serum BuChE using ATCh-iodide as substrate by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608243(CHEMBL5281655)
Affinity DataKi:  2.69E+4nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608241(CHEMBL5266369)
Affinity DataKi:  3.10E+4nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608242(CHEMBL5279509)
Affinity DataKi:  3.79E+4nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608239(CHEMBL5284808)
Affinity DataKi:  5.05E+4nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))TBA
LigandPNGBDBM50608228(CHEMBL5287059)
Affinity DataKi:  5.20E+4nMAssay Description:Binding affinity to horse serum BuChE using ATCh-iodide as substrate by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608240(CHEMBL5273719)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608246(CHEMBL5285312)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608247(CHEMBL5279226)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608260(CHEMBL5266941)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608256(CHEMBL5280828)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608241(CHEMBL5266369)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608253(CHEMBL5284047)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608242(CHEMBL5279509)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608251(CHEMBL5287695)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608250(CHEMBL5289835)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50608249(CHEMBL5269964)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to electrical eel AChE assessed as inhibition constant incubated for 20 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608243(CHEMBL5281655)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608237(CHEMBL5271146)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608238(CHEMBL5279849)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50608239(CHEMBL5284808)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to BuChE (unknown origin) assessed as inhibition constant incubated for 30 mins by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))TBA
LigandPNGBDBM50608226(CHEMBL5269935)
Affinity DataKi:  7.82E+5nMAssay Description:Binding affinity to horse serum BuChE using ATCh-iodide as substrate by ellman's methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Mus musculus (mouse))TBA
LigandPNGBDBM8963(CHEMBL32823 | Homodimeric Tacrine Analog 3b | N-[7...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of mouse brain AChEMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Mus musculus (mouse))TBA
LigandPNGBDBM8963(CHEMBL32823 | Homodimeric Tacrine Analog 3b | N-[7...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of AChE in Swiss Webster mouse cerebral homogenate using acetylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))TBA
LigandPNGBDBM50608266(CHEMBL5288285)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of mouse brain AChEMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
Displayed 1 to 50 (of 182 total ) | Next | Last >>
Jump to: