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Found 68 with Last Name = 'lovdahl' and Initial = 'm'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50078087((S)-6-[2-(4-Amino-phenyl)-ethyl]-3-(2-tert-butyl-4...)
Affinity DataIC50:  0.110nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50409219(CHEMBL2092879)
Affinity DataIC50:  0.130nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101460(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  0.170nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101485(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  0.190nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101491(CHEMBL77497 | x3-(2-tert-Butyl-4-hydroxymethyl-5-m...)
Affinity DataIC50:  0.240nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101482(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  0.280nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101480(CHEMBL78261 | x3-(2-tert-Butyl-4-hydroxymethyl-5-m...)
Affinity DataIC50:  0.340nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101474(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  0.350nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101467(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  0.410nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM2536(6-Alkyl-6-phenethyldihydropyrone 13y | 6-[2-(4-ami...)
Affinity DataIC50:  0.430nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101466(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  0.450nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101478(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  0.570nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101470(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  0.580nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101472(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  0.720nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101487(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  0.780nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101469(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  0.800nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220643(6-((cyclopropylmethyl)(propyl)amino)-4-(trifluorom...)
Affinity DataIC50:  0.800nMAssay Description:Displacement of [3H]dihydrotestosterone from human androgen receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101488(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  0.940nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101456(6-[2-(2-Amino-thiazol-4-yl)-ethyl]-3-(2-tert-butyl...)
Affinity DataIC50:  0.950nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101475(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  0.980nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101462(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  1.20nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101476(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  1.30nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101465(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  1.30nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101490(6-(2-Benzothiazol-2-yl-ethyl)-3-(2-tert-butyl-4-hy...)
Affinity DataIC50:  1.40nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101458(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  1.5nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101464(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  1.60nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220635(6-(butyl(methyl)amino)-4-(trifluoromethyl)nicotino...)
Affinity DataIC50:  3.80nMAssay Description:Displacement of [3H]dihydrotestosterone from human androgen receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101463(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  5nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101479(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  5.80nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220642(6-(sec-butyl(methyl)amino)-4-(trifluoromethyl)nico...)
Affinity DataIC50:  7nMAssay Description:Displacement of [3H]dihydrotestosterone from human androgen receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50369832(CHEMBL1907857)
Affinity DataIC50:  11.5nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101471(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  13nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101457(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  14nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101459(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  14nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25428(4-[3-(4-hydroxybutyl)-4,4-dimethyl-2,5-dioxoimidaz...)
Affinity DataIC50:  15.9nMAssay Description:Displacement of [3H]dihydrotestosterone from human androgen receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25428(4-[3-(4-hydroxybutyl)-4,4-dimethyl-2,5-dioxoimidaz...)
Affinity DataIC50:  16nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101481(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  17nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101473(CHEMBL431976 | N-(4-{2-[5-(2-tert-Butyl-4-hydroxym...)
Affinity DataIC50:  18nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101468(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  19nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25432(6-{methyl[(1R)-1-phenylethyl]amino}-4-(trifluorome...)
Affinity DataIC50:  20nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25432(6-{methyl[(1R)-1-phenylethyl]amino}-4-(trifluorome...)
Affinity DataIC50:  20nMAssay Description:Displacement of [3H]dihydrotestosterone from human androgen receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25434(4-(2-hydroxycyclohexyl)-2-(trifluoromethyl)benzoni...)
Affinity DataIC50:  26nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25428(4-[3-(4-hydroxybutyl)-4,4-dimethyl-2,5-dioxoimidaz...)
Affinity DataIC50:  31.1nMAssay Description:Antagonist activity at human androgen receptor expressed in MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM2512(3-[(2-tert-butyl-5-methylphenyl)sulfanyl]-4-hydrox...)
Affinity DataIC50:  35nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25436(4-[(1R,2R)-2-hydroxycyclohexyl]-2-(trifluoromethyl...)
Affinity DataIC50:  37nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25431(4-(2-hydroxyphenyl)-2-methoxybenzonitrile | diaryl...)
Affinity DataIC50:  37nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25430(4-(2-hydroxyphenyl)-2-(trifluoromethyl)benzonitril...)
Affinity DataIC50:  39.9nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25432(6-{methyl[(1R)-1-phenylethyl]amino}-4-(trifluorome...)
Affinity DataIC50:  45nMAssay Description:Antagonist activity at human androgen receptor expressed in MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25437((trifluoromethyl)benzonitrile, 14 | 4-{[(1R,2S)-2-...)
Affinity DataIC50:  60nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50101461(3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsul...)
Affinity DataIC50:  70nMAssay Description:HIV-1 protease inhibition.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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