TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.0600nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.140nMAssay Description:Displacement of [125I]Tyr3-NT from human NTS1R expressed in WiDr cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.180nMAssay Description:Displacement of [125I]Tyr3-NT from human NTS1R expressed in WiDr cellsMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.320nMAssay Description:Displacement of [125I]Tyr3-NT from human NTS1R expressed in HT29 cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Displacement of [125I-Tyr3]octreotide from sst2 receptor expressed in rat AR4-2J cellsMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.410nMAssay Description:Displacement of [125I]Tyr3-NT from human NTS1R expressed in HT29 cellsMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.460nMAssay Description:Displacement of [125I]Tyr3-NT from human NTS1R expressed in WiDr cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.470nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.510nMAssay Description:Displacement of [125I]Tyr3-NT from human NTS1R expressed in WiDr cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.620nMAssay Description:Displacement of [125I]Tyr3-NT from human NTS1R expressed in HT29 cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.650nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.660nMAssay Description:Displacement of [125I]Tyr3-NT from human NTS1R expressed in WiDr cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST2 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.720nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 0.760nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST2 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.850nMAssay Description:Displacement of [125I]Tyr3-NT from human NTS1R expressed in HT29 cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.850nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST4 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.960nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST2 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetBombesin receptor subtype-3(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of bombesin subtype 3 receptor expressed in human lung carcinoidsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST4 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST2 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]Tyr3-NT from human NTS1R expressed in HT29 cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST2 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST4 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST1 receptor expressed in CHO cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.94nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST3 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST4 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Displacement of [125I]Tyr3-NT from NTS1R in human exocrine ductal pancreatic carcinomaMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST3 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST4 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST4 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST5 receptor expressed in HEK293 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST4 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetAtrial natriuretic peptide receptor 1(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Displacement of [125I]ANP from NPR-A expressed in HeLa cells after 3 hrs by gamma countingMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Displacement of [125I-Tyr3]octreotide from sst2 receptor expressed in rat AR4-2J cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Displacement of [125I-Tyr3]octreotide from sst2 receptor expressed in rat AR4-2J cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST2 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 11.2nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST5 receptor expressed in HEK293 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST1 receptor expressed in CHO cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair