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Found 242 with Last Name = 'mannoury la cour' and Initial = 'c'
TargetSubstance-P receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50220136(3-[2-{1-[3,5-di(trifluoromethyl)phenyl]ethoxy}-3-(...)
Affinity DataKi:  0.0794nMAssay Description:Binding affinity to NK1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetNeuromedin-K receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50291261((S)-(+)-N-((3-[1-Benzoyl-3-(3,4-dichlorophenyl)pip...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to NK3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM85672(S33084)
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50445820(CHEMBL3104783)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptor expressed in recombinant CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.410nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetNeuromedin-K receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50445819(CHEMBL3104785)
Affinity DataKi:  0.501nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptor expressed in recombinant CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50206981(CHEMBL3948819)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50207038(CHEMBL3961596)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50207046(CHEMBL3929918)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50051293((S)-(-)-N-(R-ethylbenzyl)-3-hydroxy-2-phenylquinol...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I][MePhe7]neurokinin B from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020120(CHEMBL3288169)
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]-Bolton Hunter-substance P from human NK1 receptor expressed in human U373MG cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020118(CHEMBL3288167)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptor expressed in recombinant CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  2.88nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50050467(1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)piperi...)
Affinity DataKi:  2.95nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50207039(CHEMBL3890882)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020127(CHEMBL3288170)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]-Bolton Hunter-substance P from human NK1 receptor expressed in human U373MG cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50413618(CHEMBL484598)
Affinity DataKi:  4.17nMAssay Description:Displacement of [3H]spiperone form human cloned dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50413630(CHEMBL485128)
Affinity DataKi:  7.59nMAssay Description:Displacement of [3H]spiperone form human cloned dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50207042(CHEMBL3895173)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020120(CHEMBL3288169)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptor expressed in recombinant CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM86473(S32504 (+))
Affinity DataKi:  8.91nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM86475(S32504)
Affinity DataKi:  8.91nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50207043(CHEMBL3959964)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50445808(CHEMBL3104784)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50207045(CHEMBL3944687)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50445808(CHEMBL3104784)
Affinity DataKi:  13nMAssay Description:Binding affinity to NK1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM86473(S32504 (+))
Affinity DataKi:  14.8nMAssay Description:Displacement of [3H]spiperone form human cloned dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020112(CHEMBL3288165)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]-Bolton Hunter-substance P from human NK1 receptor expressed in human U373MG cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020119(CHEMBL3288168)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]-Bolton Hunter-substance P from human NK1 receptor expressed in human U373MG cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50445809(CHEMBL3104786)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50413621(CHEMBL482556)
Affinity DataKi:  19.1nMAssay Description:Displacement of [3H]spiperone form human cloned dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM86473(S32504 (+))
Affinity DataKi:  19.5nMAssay Description:Displacement of [3H]spiperone form human cloned dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM86474((+-)-trans-3,4,4a,5,6,10b-hexahydro-9-carbamoyl- 4...)
Affinity DataKi:  19.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020094(CHEMBL3288161)
Affinity DataKi:  20nMAssay Description:Displacement of [125I]-Bolton Hunter-substance P from human NK1 receptor expressed in human U373MG cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020117(CHEMBL3288166)
Affinity DataKi:  20nMAssay Description:Displacement of [125I]-Bolton Hunter-substance P from human NK1 receptor expressed in human U373MG cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020112(CHEMBL3288165)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptor expressed in recombinant CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020127(CHEMBL3288170)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptor expressed in recombinant CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50206983(CHEMBL3908917)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM85672(S33084)
Affinity DataKi:  29.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020114(CHEMBL3286415)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptor expressed in recombinant CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020118(CHEMBL3288167)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]-Bolton Hunter-substance P from human NK1 receptor expressed in human U373MG cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50020680(4-[2-(dipropylamino)ethyl]-1,3-dihydro-2H-indol-2-...)
Affinity DataKi:  36.3nMAssay Description:Displacement of [3H]spiperone form human cloned dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50020680(4-[2-(dipropylamino)ethyl]-1,3-dihydro-2H-indol-2-...)
Affinity DataKi:  37.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50413624(CHEMBL484732)
Affinity DataKi:  38.0nMAssay Description:Displacement of [3H]spiperone form human cloned dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50413626(CHEMBL485352)
Affinity DataKi:  39.8nMAssay Description:Displacement of [3H]spiperone form human cloned dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020114(CHEMBL3286415)
Affinity DataKi:  40nMAssay Description:Displacement of [125I]-Bolton Hunter-substance P from human NK1 receptor expressed in human U373MG cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020096(CHEMBL3288163)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptor expressed in recombinant CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50207044(CHEMBL3916787)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50207037(CHEMBL3889852)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020094(CHEMBL3288161)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptor expressed in recombinant CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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