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Found 107 with Last Name = 'mansuri' and Initial = 'mm'
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367489(CHEMBL1269499)
Affinity DataKi:  90nMAssay Description:Compound was evaluated for Kinetic constant for viral thymidine kinase of Herpes simplex virus (HSV) -1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367488(FIALURIDINE)
Affinity DataKi:  140nMAssay Description:Compound was evaluated for Kinetic constant for viral thymidine kinase of Herpes simplex virus (HSV) -2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367487(CHEMBL475717)
Affinity DataKi:  180nMAssay Description:Compound was evaluated for Kinetic constant for viral thymidine kinase of Herpes simplex virus (HSV) -1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367489(CHEMBL1269499)
Affinity DataKi:  440nMAssay Description:Compound was evaluated for Kinetic constant for viral thymidine kinase of Herpes simplex virus (HSV) -2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367488(FIALURIDINE)
Affinity DataKi:  950nMAssay Description:Compound was evaluated for Kinetic constant for viral thymidine kinase of Herpes simplex virus (HSV) -2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367487(CHEMBL475717)
Affinity DataKi:  1.40E+3nMAssay Description:Compound was evaluated for Kinetic constant for viral thymidine kinase of Herpes simplex virus (HSV) -1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282061(1-((2R,4S,5R)-5-Ethynyl-4-hydroxy-tetrahydro-furan...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity of the compound against HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282067(1-((2R,4S,5S)-4-Hydroxy-5-methoxy-tetrahydro-furan...)
Affinity DataKi:  2.90E+3nMAssay Description:Binding affinity of the compound against HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282063(1-[(2R,4S,5S)-4-Hydroxy-5-(3-phenyl-propoxy)-tetra...)
Affinity DataKi:  4.30E+3nMAssay Description:Binding affinity of the compound against HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282072(1-((2R,4S,5S)-4-Hydroxy-5-phenethyloxy-tetrahydro-...)
Affinity DataKi:  2.60E+4nMAssay Description:Binding affinity of the compound against HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021776(2-Amino-9-(2-hydroxy-ethoxymethyl)-5,9-dihydro-pur...)
Affinity DataKi:  4.50E+4nMAssay Description:Compound was evaluated for Kinetic constant for viral thymidine kinase of Herpes simplex virus (HSV) -1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021776(2-Amino-9-(2-hydroxy-ethoxymethyl)-5,9-dihydro-pur...)
Affinity DataKi:  1.80E+5nMAssay Description:Compound was evaluated for Kinetic constant for viral thymidine kinase of Herpes simplex virus (HSV) -2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Cyclin-dependent kinase 1-cyclin B1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM50088615(2-(4-Chloro-phenyl)-5,7-dihydroxy-8-(1-methyl-1,2,...)
Affinity DataIC50:  550nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM50088606(2-(2-Bromo-phenyl)-5,7-dihydroxy-8-(1-methyl-1,2,3...)
Affinity DataIC50:  650nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM50451015(CHEMBL9052)
Affinity DataIC50:  800nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM50088612(2-(2-Chloro-phenyl)-5,7-dihydroxy-8-(1-methyl-1,2,...)
Affinity DataIC50:  800nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50088606(2-(2-Bromo-phenyl)-5,7-dihydroxy-8-(1-methyl-1,2,3...)
Affinity DataIC50:  980nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM50451018(CHEMBL8675)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50088612(2-(2-Chloro-phenyl)-5,7-dihydroxy-8-(1-methyl-1,2,...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50088610(2-(3-Chloro-phenyl)-5,7-dihydroxy-8-(1-methyl-1,2,...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM50088608(2-(2,4-Dichloro-phenyl)-5,7-dihydroxy-8-(1-methyl-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50088615(2-(4-Chloro-phenyl)-5,7-dihydroxy-8-(1-methyl-1,2,...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibitory activity against Cyclin-dependent kinase 1-cyclin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50088608(2-(2,4-Dichloro-phenyl)-5,7-dihydroxy-8-(1-methyl-...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM50088619(2-(2-Fluoro-phenyl)-5,7-dihydroxy-8-(1-methyl-1,2,...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291391(3-[(E)-1-((E)-2-Carboxy-1-methyl-vinyl)-4-(5,5,8,8...)
Affinity DataIC50:  2.00E+3nMAssay Description:Compound was measured for the inhibition of human platelet PLA2 (HP-PLA2)More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50088619(2-(2-Fluoro-phenyl)-5,7-dihydroxy-8-(1-methyl-1,2,...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM50088610(2-(3-Chloro-phenyl)-5,7-dihydroxy-8-(1-methyl-1,2,...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM50451019(CHEMBL269124)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282061(1-((2R,4S,5R)-5-Ethynyl-4-hydroxy-tetrahydro-furan...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCytosolic phospholipase A2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291389(3-{(E)-3-Carbamoyl-2-methyl-1-[1-(5,5,8,8-tetramet...)
Affinity DataIC50:  4.00E+3nMAssay Description:Compound was measured for the inhibition of human platelet PLA2 (HP-PLA2)More data for this Ligand-Target Pair
In DepthDetails Article
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282067(1-((2R,4S,5S)-4-Hydroxy-5-methoxy-tetrahydro-furan...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCytosolic phospholipase A2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291390(3-{(E)-3-Carboxy-1-[1-(4-decyloxy-phenyl)-meth-(E)...)
Affinity DataIC50:  7.00E+3nMAssay Description:Compound was measured for the inhibition of human platelet PLA2 (HP-PLA2)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM50451014(CHEMBL8815)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibitory activity against Cyclin-dependent kinase 1-cyclin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM50088607(4-[2-(2-Chloro-phenyl)-5,7-dihydroxy-4-oxo-4H-chro...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291388(3-[(E)-4-(4-Adamantan-1-yl-3-hydroxy-phenyl)-1-((E...)
Affinity DataIC50:  8.00E+3nMAssay Description:Compound was measured for the inhibition of human platelet PLA2 (HP-PLA2)More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50088607(4-[2-(2-Chloro-phenyl)-5,7-dihydroxy-4-oxo-4H-chro...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282063(1-[(2R,4S,5S)-4-Hydroxy-5-(3-phenyl-propoxy)-tetra...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50088614(2-(2-Chloro-phenyl)-5,7-dihydroxy-8-((S)-2-hydroxy...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory activity against Cyclin-dependent kinase 1-cyclin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291387(3-{(E)-3-Carboxy-1-[1-(6-decyloxy-naphthalen-2-yl)...)
Affinity DataIC50:  1.40E+4nMAssay Description:Compound was measured for the inhibition of human platelet PLA2 (HP-PLA2)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCytosolic phospholipase A2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291392(3-{(E)-3-Carboxy-2-methyl-1-[1-(5,5,8,8-tetramethy...)
Affinity DataIC50:  1.70E+4nMAssay Description:Compound was measured for the inhibition of human platelet PLA2 (HP-PLA2)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCytosolic phospholipase A2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291386(3-{(E)-3-Carboxy-2-methyl-1-[1-[6-(3-phenyl-propox...)
Affinity DataIC50:  1.70E+4nMAssay Description:Compound was measured for the inhibition of human platelet PLA2 (HP-PLA2)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM50088609(2-(2-Chloro-phenyl)-5,7-dihydroxy-8-pyridin-4-yl-c...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50088609(2-(2-Chloro-phenyl)-5,7-dihydroxy-8-pyridin-4-yl-c...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM50451020(CHEMBL8620)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282072(1-((2R,4S,5S)-4-Hydroxy-5-phenethyloxy-tetrahydro-...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Mitotix

Curated by ChEMBL
LigandPNGBDBM50088614(2-(2-Chloro-phenyl)-5,7-dihydroxy-8-((S)-2-hydroxy...)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibitory activity against cyclin-dependent kinase 4-cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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