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Found 244 with Last Name = 'marler' and Initial = 'l'
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM19461(α-CA inhibitor, 5 | 5,7-dihydroxy-2-(4-hydrox...)
Affinity DataKi:  0.00110nM IC50:  1.00E+3nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92556(Neoflavonoid, 8)
Affinity DataKi:  0.00182nM IC50:  1.21E+4nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92555(Neoflavonoid, 7)
Affinity DataKi:  0.00216nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92557(Neoflavonoid, 9)
Affinity DataKi:  0.00256nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92559(Neoflavonoid, 11)
Affinity DataKi:  0.00425nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92560(Neoflavonoid, 19)
Affinity DataKi:  0.00597nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92558(Neoflavonoid, 10)
Affinity DataKi:  0.00838nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92561(Neoflavonoid, 20)
Affinity DataKi:  0.0118nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataKi:  0.0200nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM8611(4-{5H,6H,7H,8H-imidazo[1,5-a]pyridin-5-yl}benzonit...)
Affinity DataKi:  0.0500nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366125(CHEMBL1957214)
Affinity DataKi:  0.0600nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM10015(2-[3-(1-cyano-1-methylethyl)-5-(1H-1,2,4-triazol-1...)
Affinity DataKi:  0.130nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366128(CHEMBL1957217)
Affinity DataKi:  0.650nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366129(CHEMBL1957218)
Affinity DataKi:  3.20nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366127(CHEMBL1957216)
Affinity DataKi:  8.20nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366134(CHEMBL1957223)
Affinity DataKi:  35nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366120(CHEMBL1601919)
Affinity DataKi:  63nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366132(CHEMBL1957221)
Affinity DataKi:  83nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366133(CHEMBL1957222)
Affinity DataKi:  100nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366122(CHEMBL1957211)
Affinity DataKi:  234nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366130(CHEMBL1957219)
Affinity DataKi:  285nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366118(CHEMBL1957208)
Affinity DataKi:  1.16E+3nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366131(CHEMBL1957220)
Affinity DataKi:  1.48E+3nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366123(CHEMBL1957212)
Affinity DataKi:  1.72E+3nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366126(CHEMBL1957215)
Affinity DataKi:  2.55E+3nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366119(CHEMBL1957209)
Affinity DataKi:  5.32E+3nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366121(CHEMBL1957210)
Affinity DataKi:  1.26E+4nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366124(CHEMBL1957213)
Affinity DataKi:  1.50E+4nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM23926((E)-resveratrol | 5-[(E)-2-(4-hydroxyphenyl)etheny...)
Affinity DataKi:  4.17E+4nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human aromatase using dibenzylfluorescein substrate preincubated for 30 mins measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM8611(4-{5H,6H,7H,8H-imidazo[1,5-a]pyridin-5-yl}benzonit...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human aromatase using dibenzylfluorescein substrate preincubated for 30 mins measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366125(CHEMBL1957214)
Affinity DataIC50:  4nMAssay Description:Inhibition of human aromatase using dibenzylfluorescein substrate preincubated for 30 mins measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM10015(2-[3-(1-cyano-1-methylethyl)-5-(1H-1,2,4-triazol-1...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human aromatase using dibenzylfluorescein substrate preincubated for 30 mins measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366128(CHEMBL1957217)
Affinity DataIC50:  23nMAssay Description:Inhibition of human aromatase using dibenzylfluorescein substrate preincubated for 30 mins measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50322045((Z)-4-(1-(3,5-Dimethoxyphenyl)-3-(1H-imidazol-1-yl...)
Affinity DataIC50:  36nMAssay Description:Inhibition of human aromatase preincubated with NADP+ for 10 mins before substrate addition measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50322044((Z)-1-(3-(3,5-Dimethoxyphenyl)-2-(4-nitrophenyl)al...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human aromatase preincubated with NADP+ for 10 mins before substrate addition measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366129(CHEMBL1957218)
Affinity DataIC50:  78nMAssay Description:Inhibition of human aromatase using dibenzylfluorescein substrate preincubated for 30 mins measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM29227(casimiroin analogue, 1p)
Affinity DataIC50:  100nMAssay Description:Aromatase inhibition was quantified by measuring the fluorescent intensity of fluorescein, the hydrolysis product of dibenzylfluorescein (DBF), by ar...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347488(CHEMBL1802205)
Affinity DataIC50:  160nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50366127(CHEMBL1957216)
Affinity DataIC50:  164nMAssay Description:Inhibition of human aromatase using dibenzylfluorescein substrate preincubated for 30 mins measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347486(CHEMBL1802199)
Affinity DataIC50:  186nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50240895(2-(1H-Imidazol-1-yl)-1-(4-nitrophenyl)ethanone | 2...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human aromatase preincubated with NADP+ for 10 mins before substrate addition measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50361943(CHEMBL1939366)
Affinity DataIC50:  200nMAssay Description:Inhibition of human aromatase using dibenzylfluorescein as substrate preincubated for 30 mins measured after 2 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM23419((2S)-5,7-dihydroxy-2-(4-hydroxyphenyl)-3,4-dihydro...)
Affinity DataIC50:  230nMAssay Description:Inhibition of human aromatase using dibenzylfluorescein as substrate preincubated for 30 mins measured after 2 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM23419((2S)-5,7-dihydroxy-2-(4-hydroxyphenyl)-3,4-dihydro...)
Affinity DataIC50:  230nMAssay Description:Inhibition of human aromatase activity after 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM23419((2S)-5,7-dihydroxy-2-(4-hydroxyphenyl)-3,4-dihydro...)
Affinity DataIC50:  230nMAssay Description:Inhibition of aromatase after 10 mins preincubation by plate reader relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50322046(3,4,5-Trimethoxy-4'-amino-trans-stilbene | 4-[2-(3...)
Affinity DataIC50:  270nMAssay Description:Inhibition of human quinone reductase 2 expressed in Escherichia coli BL21(DE3) by UV-vis microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...)
Affinity DataIC50:  270nMAssay Description:Aromatase inhibition was quantified by measuring the fluorescent intensity of fluorescein, the hydrolysis product of dibenzylfluorescein (DBF), by ar...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347476(CHEMBL1802264)
Affinity DataIC50:  320nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347471(CHEMBL1802260)
Affinity DataIC50:  450nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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