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Found 127 with Last Name = 'maroun' and Initial = 'c'
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM93149(2-oxoimidazolidine-1-carboxamide, 16)
Affinity DataIC50:  2nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM93147(2-oxoimidazolidine-1-carboxamide, 14)
Affinity DataIC50:  3nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM93145(2-oxoimidazolidine-1-carboxamide, 5)
Affinity DataIC50:  4nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM93150(2-oxoimidazolidine-1-carboxamide, 17)
Affinity DataIC50:  4nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM93148(2-oxoimidazolidine-1-carboxamide, 15)
Affinity DataIC50:  5nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50255852(4-(((R)-3-(4-hydroxybenzyl)-2,3-dihydro-2-oxoquino...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant histone deacetylase 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50306503(4,4,4-trifluoro-3-(3-fluoro-4-(2-(1-methyl-1H-imid...)
Affinity DataIC50:  10nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50299777(CHEMBL573761 | N-(4-(6,7-dimethoxyquinolin-4-yloxy...)
Affinity DataIC50:  10nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50247984(CHEMBL453613 | N-(4-(2-(1-ethyl-1H-imidazol-4-yl)t...)
Affinity DataIC50:  10nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50255096(4-(((R)-3-benzyl-2,3-dihydro-2-oxoquinoxalin-4(1H)...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant histone deacetylase 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM19130((2E,4E,6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant histone deacetylase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50255853(4-(((R)-2,3-dihydro-2-oxo-3-phenethylquinoxalin-4(...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant histone deacetylase 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50247962(CHEMBL462232 | N-(3-fluoro-4-(2-(1-methyl-1H-imida...)
Affinity DataIC50:  10nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM19130((2E,4E,6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant histone deacetylase 6More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM93146(2-oxoimidazolidine-1-carboxamide, 13)
Affinity DataIC50:  20nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50247984(CHEMBL453613 | N-(4-(2-(1-ethyl-1H-imidazol-4-yl)t...)
Affinity DataIC50:  20nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50247962(CHEMBL462232 | N-(3-fluoro-4-(2-(1-methyl-1H-imida...)
Affinity DataIC50:  20nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50317335(CHEMBL1095356 | N-(4-(2-(4-(dimethylcarbamoyl)phen...)
Affinity DataIC50:  30nMAssay Description:Inhibition of TPR-tagged RON catalytic domain expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM93143(Oxo-3-phenylimidazolidine-1-carboxamide, 4)
Affinity DataIC50:  30nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50317333((S)-N-(3-fluoro-4-(2-(4-((N-(1-methoxypropan-2-yl)...)
Affinity DataIC50:  30nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50317336(CHEMBL1095357 | N-(4-(2-(4-((2-(dimethylamino)ethy...)
Affinity DataIC50:  30nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50299777(CHEMBL573761 | N-(4-(6,7-dimethoxyquinolin-4-yloxy...)
Affinity DataIC50:  30nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50317338(6-(7-(2-fluoro-4-(1-phenyl-5-(trifluoromethyl)-1H-...)
Affinity DataIC50:  30nMAssay Description:Inhibition of TPR-tagged RON catalytic domain expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50317339(6-(7-(2-fluoro-4-(1-phenyl-5-(trifluoromethyl)-1H-...)
Affinity DataIC50:  40nMAssay Description:Inhibition of TPR-tagged RON catalytic domain expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50255914(4-(((R)-2,3-dihydro-2-oxo-3-((thiophen-2-yl)methyl...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human recombinant histone deacetylase 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50255809(4-(((R)-3-(3,4-difluorobenzyl)-2,3-dihydro-2-oxoqu...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human recombinant histone deacetylase 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50255854((R)-tert-butyl 4-(1-(4-(hydroxycarbamoyl)benzyl)-3...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human recombinant histone deacetylase 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50317337((S)-N-(4-(2-(4-(3-(dimethylamino)pyrrolidine-1-car...)
Affinity DataIC50:  40nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50317338(6-(7-(2-fluoro-4-(1-phenyl-5-(trifluoromethyl)-1H-...)
Affinity DataIC50:  40nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM93142(Oxo-3-phenylimidazolidine-1-carboxamide, 3)
Affinity DataIC50:  50nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50317323(CHEMBL1094718 | N-(3-fluoro-4-(2-(1-methyl-1H-imid...)
Affinity DataIC50:  50nMAssay Description:Inhibition of TPR-tagged RON catalytic domain expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50317340(CHEMBL1095361 | N-(4-(2-(1-acetyl-1,2,3,6-tetrahyd...)
Affinity DataIC50:  50nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50317335(CHEMBL1095356 | N-(4-(2-(4-(dimethylcarbamoyl)phen...)
Affinity DataIC50:  50nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50255910(4-(((R)-3-(4-tert-butoxybenzyl)-2,3-dihydro-2-oxoq...)
Affinity DataIC50:  50nMAssay Description:Inhibition of human recombinant histone deacetylase 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50317334(CHEMBL1095036 | N-(3-fluoro-4-(2-(4-((2-(methylsul...)
Affinity DataIC50:  60nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50317339(6-(7-(2-fluoro-4-(1-phenyl-5-(trifluoromethyl)-1H-...)
Affinity DataIC50:  60nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50317332(CHEMBL1095034 | N-(3-fluoro-4-(2-(1-methyl-1H-imid...)
Affinity DataIC50:  60nMAssay Description:Inhibition of TPR-tagged RON catalytic domain expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50317333((S)-N-(3-fluoro-4-(2-(4-((N-(1-methoxypropan-2-yl)...)
Affinity DataIC50:  60nMAssay Description:Inhibition of TPR-tagged RON catalytic domain expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50317330(CHEMBL1098157 | N-(3-fluoro-4-(2-(1-methyl-1H-imid...)
Affinity DataIC50:  60nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50317326(CHEMBL1086932 | N-(3-fluoro-4-(2-(1-methyl-1H-imid...)
Affinity DataIC50:  70nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50317327(CHEMBL1086675 | N-(3-fluoro-4-(2-(1-methyl-1H-imid...)
Affinity DataIC50:  70nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50247962(CHEMBL462232 | N-(3-fluoro-4-(2-(1-methyl-1H-imida...)
Affinity DataIC50:  70nMAssay Description:Inhibition of c-Met phosphorylation in human MKN45 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50317331(1-tert-butyl-N-(3-fluoro-4-(2-(1-methyl-1H-imidazo...)
Affinity DataIC50:  70nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50317328(CHEMBL1086676 | N-(3-fluoro-4-(2-(1-methyl-1H-imid...)
Affinity DataIC50:  80nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50247962(CHEMBL462232 | N-(3-fluoro-4-(2-(1-methyl-1H-imida...)
Affinity DataIC50:  80nMAssay Description:Inhibition of c-Met-mediated scattering in HGF-stimulated human DU145 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM50247962(CHEMBL462232 | N-(3-fluoro-4-(2-(1-methyl-1H-imida...)
Affinity DataIC50:  80nMAssay Description:Inhibition of c-Met-mediated cell migration of human A549 cells by would healingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50317324(CHEMBL1087984 | N-(4-(6,7-dimethoxyquinolin-4-ylox...)
Affinity DataIC50:  80nMAssay Description:Inhibition of TPR-tagged RON catalytic domain expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50317334(CHEMBL1095036 | N-(3-fluoro-4-(2-(4-((2-(methylsul...)
Affinity DataIC50:  80nMAssay Description:Inhibition of TPR-tagged RON catalytic domain expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50317336(CHEMBL1095357 | N-(4-(2-(4-((2-(dimethylamino)ethy...)
Affinity DataIC50:  90nMAssay Description:Inhibition of TPR-tagged RON catalytic domain expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50317340(CHEMBL1095361 | N-(4-(2-(1-acetyl-1,2,3,6-tetrahyd...)
Affinity DataIC50:  90nMAssay Description:Inhibition of TPR-tagged RON catalytic domain expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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