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Found 80 with Last Name = 'marton' and Initial = 'j'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551316(CHEMBL4776706)
Affinity DataKi:  0.00630nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551315(CHEMBL4762529)
Affinity DataKi:  0.0125nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551313(CHEMBL4745764)
Affinity DataKi:  0.0136nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50001714(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-(1S,2...)
Affinity DataKi:  0.0200nMAssay Description:Binding affinity to human cloned kappa opioid receptor expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551314(CHEMBL4751305)
Affinity DataKi:  0.0220nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551311(CHEMBL4746512)
Affinity DataKi:  0.0240nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551309(CHEMBL4758369)
Affinity DataKi:  0.0325nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551311(CHEMBL4746512)
Affinity DataKi:  0.0333nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551314(CHEMBL4751305)
Affinity DataKi:  0.0435nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50001714(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-(1S,2...)
Affinity DataKi:  0.0700nMAssay Description:Binding affinity to human cloned mu opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50354578(BUPRENORPHINE | US10752592, Compound buprenorphine...)
Affinity DataKi:  0.0700nMAssay Description:Binding affinity to human cloned kappa opioid receptor expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020711(CHEMBL3291216)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity to human cloned kappa opioid receptor expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50354578(BUPRENORPHINE | US10752592, Compound buprenorphine...)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity to human cloned mu opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020711(CHEMBL3291216)
Affinity DataKi:  0.100nMAssay Description:Binding affinity to human cloned mu opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020709(CHEMBL3291215)
Affinity DataKi:  0.120nMAssay Description:Binding affinity to human cloned kappa opioid receptor expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50300442((20R)-4,5-alpha-Epoxy-17-methyl-3-hydroxy-6-methox...)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]diprenorphine from human cloned kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50177895(CHEMBL200456 | fluoromethyl 1-(2-phenylethyl)-4-(N...)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]DAMGO from recombinant human mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50177898(2-Fluoro-N-[4-methoxymethyl-1-(2-thiophen-2-yl-eth...)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]DAMGO from recombinant human mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551319(CHEMBL4753839)
Affinity DataKi:  0.177nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50300442((20R)-4,5-alpha-Epoxy-17-methyl-3-hydroxy-6-methox...)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]diprenorphine from human cloned mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020708(CHEMBL3291214)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to human cloned kappa opioid receptor expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551307(CHEMBL4754079)
Affinity DataKi:  0.214nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551312(CHEMBL4761619)
Affinity DataKi:  0.218nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50001714(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-(1S,2...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity to human cloned delta opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020708(CHEMBL3291214)
Affinity DataKi:  0.240nMAssay Description:Binding affinity to human cloned mu opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020709(CHEMBL3291215)
Affinity DataKi:  0.240nMAssay Description:Binding affinity to human cloned mu opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551317(CHEMBL4764372)
Affinity DataKi:  0.252nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551312(CHEMBL4761619)
Affinity DataKi:  0.257nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551308(CHEMBL4758814)
Affinity DataKi:  0.280nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551316(CHEMBL4776706)
Affinity DataKi:  0.321nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551318(CHEMBL4787652)
Affinity DataKi:  0.326nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551310(CHEMBL4752367)
Affinity DataKi:  0.435nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020711(CHEMBL3291216)
Affinity DataKi:  0.490nMAssay Description:Binding affinity to human cloned delta opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551308(CHEMBL4758814)
Affinity DataKi:  0.531nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551317(CHEMBL4764372)
Affinity DataKi:  0.682nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50177899(CHEMBL371710 | methyl 4-[(N-1-oxopropyl)-N-phenyla...)
Affinity DataKi:  0.740nMAssay Description:Displacement of [3H]DAMGO from recombinant human mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551313(CHEMBL4745764)
Affinity DataKi:  0.796nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50354578(BUPRENORPHINE | US10752592, Compound buprenorphine...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to human cloned delta opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50177897(2-fluoroethyl 1-(2-phenylethyl)-4-(N-phenylpropana...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DAMGO from recombinant human mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551319(CHEMBL4753839)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551311(CHEMBL4746512)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551307(CHEMBL4754079)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551316(CHEMBL4776706)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020709(CHEMBL3291215)
Affinity DataKi:  2.10nMAssay Description:Binding affinity to human cloned delta opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50177894(2-Fluoro-N-(1-phenethyl-piperidin-4-yl)-N-phenyl-p...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]DAMGO from recombinant human mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551314(CHEMBL4751305)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551307(CHEMBL4754079)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551315(CHEMBL4762529)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551319(CHEMBL4753839)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50551313(CHEMBL4745764)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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