TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidad De Santiago
Curated by ChEMBL
Universidad De Santiago
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:In vitro ability to displace [3H]ketanserin binding from 5-hydroxytryptamine 2A receptor in rat striatal membrane.More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.210nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.290nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.320nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]OSIP339391 from human recombinant adenosine A2B receptor expressed in HEK293 cell membranes after 60 mins by liquid scintillation...More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.501nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.501nMAssay Description:Displacement of [3H]ketanserin human cloned serotonin 5HT2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.501nMAssay Description:Binding affinity towards serotonin 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.537nMAssay Description:In vitro ability to displace [3H]spiperone binding from dopamine receptor D2 in rat striatal membrane.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.562nMAssay Description:Antagonist activity at human cloned 5HT2A receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.603nMAssay Description:Binding affinity towards dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.603nMAssay Description:Displacement of [3H]spiperone human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.603nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.603nMAssay Description:Displacement of [3H]spiperone from human D2 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.603nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.724nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.930nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidad De Santiago
Curated by ChEMBL
Universidad De Santiago
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:In vitro ability to displace [3H]ketanserin binding from 5-hydroxytryptamine 2A receptor in rat striatal membrane.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.55nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidad De Santiago
Curated by ChEMBL
Universidad De Santiago
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:In vitro ability to displace [3H]ketanserin binding from 5-hydroxytryptamine 2A receptor in rat striatal membrane.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidad De Santiago
Curated by ChEMBL
Universidad De Santiago
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Compound was measured for the inhibition of [3H]ketanserin binding to rat frontal cortex membrane (5-HT2A receptor)More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidad De Santiago
Curated by ChEMBL
Universidad De Santiago
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:In vitro ability to displace [3H]ketanserin binding from 5-hydroxytryptamine 2A receptor in rat striatal membrane.More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]ZM241385/[125I]IABOPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]4-(2-[7-amino-2-(2-furyl)[1,2,4]triazolo[2,3-a][1,3,5]triazin-5-ylamino]ethyl)phenol from human adenosine A2A receptor expressed ...More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]ketanserin human cloned serotonin 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidad De Santiago
Curated by ChEMBL
Universidad De Santiago
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:In vitro ability to displace [3H]ketanserin binding from 5-hydroxytryptamine 2A receptor in rat striatal membrane.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 2.51nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidad De Santiago
Curated by ChEMBL
Universidad De Santiago
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Compound was tested in vitro for its binding affinity towards 5-hydroxytryptamine 2A receptor from rat frontal cortex using [3H]-ketanserin as radiol...More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Santiago De Compostela
Curated by ChEMBL
University Of Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:In vitro ability to displace [3H]spiperone binding from dopamine receptor D2 in rat striatal membrane.More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Compound was measured for the inhibition of [3H]spiperone binding to striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair