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Found 240 with Last Name = 'massarelli' and Initial = 'i'
TargetVitamin D3 receptor(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50135183(CHEMBL3745798)
Affinity DataKi:  0.0200nMAssay Description:Displacement of [3H]1alpha,25-(OH)2D3 from full-length recombinant rat VDR by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50135182(CHEMBL3746107)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]1alpha,25-(OH)2D3 from full-length recombinant rat VDR by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50135184(CHEMBL3746058)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]1alpha,25-(OH)2D3 from full-length recombinant rat VDR by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50135186(CHEMBL1214620)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]1alpha,25-(OH)2D3 from full-length recombinant rat VDR by scintillation counterMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50135185(CHEMBL3746759)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]1alpha,25-(OH)2D3 from full-length recombinant rat VDR by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]1alpha,25-(OH)2D3 from full-length recombinant rat VDR by scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196014(3-(2-(trifluoromethyl)benzyl)-N-cyclopentyl-5-phen...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196002(3-(2-fluorobenzyl)-N-cyclohexyl-5-phenyl-3H-[1,2,3...)
Affinity DataKi:  1.15nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196009(3-benzyl-N-cyclohexyl-5-phenyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276769(CHEMBL514399 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276770(CHEMBL456211 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195990(3-(2-fluorobenzyl)-5-phenyl-N-propyl-3H-[1,2,3]tri...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195996(3-(3-(2-fluorobenzyl)-5-phenyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196018(3-(2-fluorobenzyl)-N-butyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195995(1-(3-(2-fluorobenzyl)-5-phenyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195992(3-benzyl-N-cyclobutyl-5-phenyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276243(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimid...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196015(3-(2-(trifluoromethyl)benzyl)-N-butyl-5-phenyl-3H-...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196003(3-(2-fluorobenzyl)-N-cyclopentyl-5-phenyl-3H-[1,2,...)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196030(3-(2-(trifluoromethyl)benzyl)-N-cyclohexyl-5-pheny...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276242(4-amino-N-(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,...)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276707(CHEMBL458346 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195999(1-(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyri...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196020(3-(2-(trifluoromethyl)benzyl)-N-cyclopropyl-5-phen...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276772(CHEMBL456011 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196011(3-(2-chlorobenzyl)-N-cyclopentyl-5-phenyl-3H-[1,2,...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276867(CHEMBL459772 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196012(3-benzyl-N-butyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196022(3-benzyl-N-cyclopentyl-5-phenyl-3H-[1,2,3]triazolo...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196010(3-(2-fluorobenzyl)-N-ethyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195997(3-(2-chlorobenzyl)-N-cyclopropyl-5-phenyl-3H-[1,2,...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195994(3-benzyl-N-cyclopropyl-5-phenyl-3H-[1,2,3]triazolo...)
Affinity DataKi:  11.3nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276866(CHEMBL517097 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276771(CHEMBL456010 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196023(3-benzyl-N-hexyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d...)
Affinity DataKi:  13.2nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196026(3-(2-(trifluoromethyl)benzyl)-N-methyl-5-phenyl-3H...)
Affinity DataKi:  14.9nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195998(3-(2-fluorobenzyl)-N-cyclopropyl-5-phenyl-3H-[1,2,...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196007(3-(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyri...)
Affinity DataKi:  21.4nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276939(CHEMBL517258 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276161(CHEMBL471022 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195993(3-(2-chlorobenzyl)-N-cyclobutyl-5-phenyl-3H-[1,2,3...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196024(3-(2-fluorobenzyl)-N-hexyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196019(3-(2-fluorobenzyl)-N-methyl-5-phenyl-3H-[1,2,3]tri...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50242664(CHEMBL455383 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196016(3-(2-chlorobenzyl)-N-hexyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276163(3-amino-N-(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196013(1-(3-(2-chlorobenzyl)-5-phenyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196029(3-(3-(2-chlorobenzyl)-5-phenyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196006(3-(2-chlorobenzyl)-N-cyclohexyl-5-phenyl-3H-[1,2,3...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276162(2-amino-N-(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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