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Found 341 with Last Name = 'mayer' and Initial = 'c'
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425360(CHEMBL2316207)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425359(CHEMBL2316490)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425384(CHEMBL2316466)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425358(CHEMBL2316491)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425352(CHEMBL2316486)
Affinity DataIC50:  1nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) in presence of 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425353(CHEMBL2316206)
Affinity DataIC50:  1nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425354(CHEMBL2316497)
Affinity DataIC50:  1nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425357(CHEMBL2316485)
Affinity DataIC50:  1nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425356(CHEMBL2316489)
Affinity DataIC50:  1nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425352(CHEMBL2316486)
Affinity DataIC50:  1nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425355(CHEMBL2316494)
Affinity DataIC50:  1nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425344(CHEMBL2316205)
Affinity DataIC50:  2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425345(CHEMBL2316201)
Affinity DataIC50:  2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425346(CHEMBL2316479)
Affinity DataIC50:  2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425347(CHEMBL2316474)
Affinity DataIC50:  2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425348(CHEMBL2316472)
Affinity DataIC50:  2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425349(CHEMBL2316492)
Affinity DataIC50:  2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425350(CHEMBL2316488)
Affinity DataIC50:  2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425351(CHEMBL2316483)
Affinity DataIC50:  2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286792((R)-2-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4...)
Affinity DataIC50:  2.5nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425352(CHEMBL2316486)
Affinity DataIC50:  3nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) in presence of 300 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398191(CHEMBL2182085)
Affinity DataIC50:  3nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425338(CHEMBL2316202)
Affinity DataIC50:  3nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425343(CHEMBL2316470)
Affinity DataIC50:  3nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425340(CHEMBL2316477)
Affinity DataIC50:  3nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425341(CHEMBL2316476)
Affinity DataIC50:  3nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425342(CHEMBL2316473)
Affinity DataIC50:  3nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425339(CHEMBL2316481)
Affinity DataIC50:  3nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425369(CHEMBL2316208)
Affinity DataIC50:  4nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398165(CHEMBL2182072)
Affinity DataIC50:  4nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Technische UniversitÄT Dortmund

LigandPNGBDBM92356(Chir98014, 20)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of UmGSK3 by kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative glycogen synthase kinase 3 alpha(Ustilago maydis (Smut fungus))
Technische UniversitÄT Dortmund

LigandPNGBDBM92356(Chir98014, 20)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of UmGSK3 by kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425382(CHEMBL2316197)
Affinity DataIC50:  5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425379(CHEMBL2316478)
Affinity DataIC50:  5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398153(CHEMBL2177215)
Affinity DataIC50:  5nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50392175(CHEMBL2152944)
Affinity DataIC50:  5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425375(CHEMBL2316475)
Affinity DataIC50:  5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286804((R)-2-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4...)
Affinity DataIC50:  5.30nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425372(CHEMBL2316196)
Affinity DataIC50:  6nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425377(CHEMBL2316493)
Affinity DataIC50:  7nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425367(CHEMBL2316199)
Affinity DataIC50:  7nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425370(CHEMBL2316203)
Affinity DataIC50:  8nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286800((R)-2-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4...)
Affinity DataIC50:  8nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286795((R)-2-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4...)
Affinity DataIC50:  8nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPutative glycogen synthase kinase 3 alpha(Ustilago maydis (Smut fungus))
Technische UniversitÄT Dortmund

LigandPNGBDBM25036(CHEMBL393525 | N'-[(1E)-{6-bromoimidazo[1,2-a]pyri...)
Affinity DataIC50:  8nMAssay Description:Inhibition of UmGSK3 by kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425383(CHEMBL2316480)
Affinity DataIC50:  9nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM28104(3-cyanoquinoline, 29 | 4-({3-chloro-4-[(1-ethyl-4,...)
Affinity DataIC50:  9nMpH: 7.5 T: 2°CAssay Description:Assays were performed in microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified kinase in the presence of test com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398166(CHEMBL2182071)
Affinity DataIC50:  9nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425378(CHEMBL2316194)
Affinity DataIC50:  10nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50425381(CHEMBL2316469)
Affinity DataIC50:  10nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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