TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) in presence of 100 uM ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) in presence of 300 uM ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Inhibition of UmGSK3 by kinase inhibitors.More data for this Ligand-Target Pair
TargetPutative glycogen synthase kinase 3 alpha(Ustilago maydis (Smut fungus))
Technische UniversitÄT Dortmund
Technische UniversitÄT Dortmund
Affinity DataIC50: 4.70nMAssay Description:Inhibition of UmGSK3 by kinase inhibitors.More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
TargetPutative glycogen synthase kinase 3 alpha(Ustilago maydis (Smut fungus))
Technische UniversitÄT Dortmund
Technische UniversitÄT Dortmund
Affinity DataIC50: 8nMAssay Description:Inhibition of UmGSK3 by kinase inhibitors.More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMpH: 7.5 T: 2°CAssay Description:Assays were performed in microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified kinase in the presence of test com...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of T£Bingen
Curated by ChEMBL
University Of T£Bingen
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) by ELISAMore data for this Ligand-Target Pair