Affinity DataKi: 3nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Inhibition of human recombinant full length MMP13 by steady state kinetic assayMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Inhibition of muscarinic M1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Inhibition of muscarinic M2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Inhibition of 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 950nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of muscarinic M3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
Affinity DataKi: 1.80E+4nMAssay Description:Compound tested for inhibition of alpha-galactosidase from Aspergillus nigerMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+5nMAssay Description:Compound tested for inhibition of alpha-galactosidase from Aspergillus nigerMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+5nMAssay Description:Compound tested for inhibition of alpha-galactosidase from Aspergillus nigerMore data for this Ligand-Target Pair
Affinity DataIC50: 0.670nMAssay Description:Inhibition of human recombinant MMP13 catalytic domainMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Inhibition of MMP17 catalytic domainMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibition of MMP14 catalytic domainMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Inhibition of MMP12 catalytic domainMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibition of human recombinant MMP13 catalytic domainMore data for this Ligand-Target Pair
TargetComplement factor B(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human serine protease factor B by TR-FRET based competition binding assayMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Antagonist activity at rabbit Cav1.2 expressed in HEK293 cells assessed as inhibition of voltage pulse-induced calcium current by FLIPR calcium 4 ass...More data for this Ligand-Target Pair