Compile Data Set for Download or QSAR
maximum 50k data
Found 49 with Last Name = 'mingeot-leclercq' and Initial = 'mp'
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50470665(CHEMBL3143220)
Affinity DataIC50:  4.94E+4nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activityMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011913(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-3,...)
Affinity DataIC50:  6.00E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011901(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-6-...)
Affinity DataIC50:  6.50E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50470662(CHEMBL357385)
Affinity DataIC50:  7.55E+4nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activity.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011899(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-6-...)
Affinity DataIC50:  7.70E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011914(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-6-...)
Affinity DataIC50:  7.80E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011926(4-amino-2-[2,4-diamino-5-(3-amino-6-aminomethyl-4,...)
Affinity DataIC50:  7.90E+4nMAssay Description:in vitro inhibitory activity against Lysosomal phospholipase A1 consisting of negatively charged liposomes and lysosomal extracts. p<0.05More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50031282(CHEBI:17630 | Kanamycin)
Affinity DataIC50:  8.04E+4nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011904(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-3,...)
Affinity DataIC50:  8.10E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011897(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-3,...)
Affinity DataIC50:  8.30E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011902(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-6-...)
Affinity DataIC50:  8.30E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011898(2-{4-Amino-6-[4,6-diamino-3-(3-amino-6-aminomethyl...)
Affinity DataIC50:  8.70E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011905(CHEMBL285200 | N-{4-Amino-6-[4,6-diamino-3-(3-amin...)
Affinity DataIC50:  8.80E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011894(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-6-...)
Affinity DataIC50:  8.90E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50470660(CHEMBL142949)
Affinity DataIC50:  9.14E+4nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activity.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50470660(CHEMBL142949)
Affinity DataIC50:  9.14E+4nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activity.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011925(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-3,...)
Affinity DataIC50:  9.30E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011912(4-amino-2-[4,6-diamino-3-(3-amino-6-aminomethyl-4,...)
Affinity DataIC50:  9.30E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50366389(GENTAMICIN)
Affinity DataIC50:  9.42E+4nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011929(4-amino-2-azidomethyl-6-[2,4-diamino-5-(3-amino-6-...)
Affinity DataIC50:  9.50E+4nMAssay Description:in vitro inhibitory activity against Lysosomal phospholipase A1 consisting of negatively charged liposomes and lysosomal extracts. p<0.05More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011920(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-3,...)
Affinity DataIC50:  9.60E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011893(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-6-...)
Affinity DataIC50:  9.60E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011896(CHEMBL286153 | N-{4-Amino-6-[4,6-diamino-3-(3-amin...)
Affinity DataIC50:  9.70E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011900(CHEMBL34605 | N-{4-Amino-6-[4,6-diamino-3-(3-amino...)
Affinity DataIC50:  9.90E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011924(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-6-...)
Affinity DataIC50:  9.90E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50470663(CHEMBL3143222)
Affinity DataIC50:  1.01E+5nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activityMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011922(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-3,...)
Affinity DataIC50:  1.02E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011907(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-6-...)
Affinity DataIC50:  1.04E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011927(4-amino-2-chloromethyl-6-[2,4-diamino-5-(3-amino-6...)
Affinity DataIC50:  1.05E+5nMAssay Description:in vitro inhibitory activity against Lysosomal phospholipase A1 consisting of negatively charged liposomes and lysosomal extracts.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011919(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-3,...)
Affinity DataIC50:  1.06E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011921(CHEMBL34670 | N-{4-Amino-6-[4,6-diamino-3-(3-amino...)
Affinity DataIC50:  1.09E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50368267(KANAMYCIN B | Kanamycin | Kantrex | Klebcil)
Affinity DataIC50:  1.10E+5nMAssay Description:In vitro inhibitory activity against Lysosomal phospholipase A1 consisting of negatively charged liposomes and lysosomal extracts.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011906(CHEMBL287699 | Hexanoic acid {4-amino-6-[4,6-diami...)
Affinity DataIC50:  1.10E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50031282(CHEBI:17630 | Kanamycin)
Affinity DataIC50:  1.10E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011918(CHEMBL415861 | N-{4-Amino-6-[4,6-diamino-3-(3-amin...)
Affinity DataIC50:  1.15E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011895(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-3,...)
Affinity DataIC50:  1.15E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50470664(Netilmicin)
Affinity DataIC50:  1.15E+5nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011915(CHEMBL287846 | N-{4-Amino-6-[4,6-diamino-3-(3-amin...)
Affinity DataIC50:  1.16E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011917(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-3,...)
Affinity DataIC50:  1.18E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50470666(CHEMBL143885)
Affinity DataIC50:  1.18E+5nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011928(CHEMBL289737 | N-{4-Amino-6-[2,4-diamino-5-(3-amin...)
Affinity DataIC50:  1.19E+5nMAssay Description:in vitro inhibitory activity against Lysosomal phospholipase A1 consisting of negatively charged liposomes and lysosomal extracts.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011910(CHEMBL36133 | N-{4-Amino-6-[4,6-diamino-3-(3-amino...)
Affinity DataIC50:  1.20E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011923(CHEMBL34486 | N-{4-Amino-6-[4,6-diamino-3-(3-amino...)
Affinity DataIC50:  1.21E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011911(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-6-...)
Affinity DataIC50:  1.23E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011909(CHEMBL416222 | N-{4-Amino-6-[4,6-diamino-3-(3-amin...)
Affinity DataIC50:  1.25E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011892(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-3,...)
Affinity DataIC50:  1.29E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011908(5-amino-2-aminomethyl-6-[4,6-diamino-3-(4-amino-6-...)
Affinity DataIC50:  1.29E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50470661(CHEMBL356044)
Affinity DataIC50:  1.32E+5nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50011916(CHEMBL285021 | N-{4-Amino-6-[4,6-diamino-3-(3-amin...)
Affinity DataIC50:  1.34E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed