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Found 63 with Last Name = 'moe' and Initial = 'st'
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.00720nMAssay Description:Tested for binding activity against delta1 opioid receptor using [3H]DPDPE ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity against delta-opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040487(17-(cyclopropylmethyl)4,5-alpha-epoxy-3,14-dihydro...)
Affinity DataKi:  0.0470nMAssay Description:Tested for binding activity against delta opioid receptor using [3H]naltridole ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040485(15-benzyl-4-cyclopropylmethyl-10,17-dihydroxy-(1S,...)
Affinity DataKi:  0.100nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040483(4-cyclopropylmethyl-10,17-dihydroxy-15-phenyl-(1S,...)
Affinity DataKi:  0.120nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  0.190nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  0.600nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50056628(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-phenyl-(...)
Affinity DataKi:  0.830nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040483(4-cyclopropylmethyl-10,17-dihydroxy-15-phenyl-(1S,...)
Affinity DataKi:  0.860nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040483(4-cyclopropylmethyl-10,17-dihydroxy-15-phenyl-(1S,...)
Affinity DataKi:  1.40nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50297170(7-(2'-spiroindanyl)oxymorphone | 7-(Spiroindano)Ox...)
Affinity DataKi:  1.40nMAssay Description:Antagonism against bradykinin receptor B2 in guinea pig ileal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  1.40nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040487(17-(cyclopropylmethyl)4,5-alpha-epoxy-3,14-dihydro...)
Affinity DataKi:  1.40nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  1.5nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50056628(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-phenyl-(...)
Affinity DataKi:  1.80nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50056628(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-phenyl-(...)
Affinity DataKi:  1.90nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  2.20nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  2.20nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50038641(22-cyclopropylmethyl-(2R,13S)-14-oxa-4,22-diazahep...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity against delta-opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50297170(7-(2'-spiroindanyl)oxymorphone | 7-(Spiroindano)Ox...)
Affinity DataKi:  3.30nMAssay Description:Selective binding affinity against Opioid receptor delta 2, using [3H]DSLET as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity against mu-opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  4.5nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50038641(22-cyclopropylmethyl-(2R,13S)-14-oxa-4,22-diazahep...)
Affinity DataKi:  4.90nMAssay Description:Binding affinity against mu-opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040482(17-(cyclopropylmethyl)-6,7-didehydro-4,5-alpha-epo...)
Affinity DataKi:  5.20nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040485(15-benzyl-4-cyclopropylmethyl-10,17-dihydroxy-(1S,...)
Affinity DataKi:  5.90nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  7.80nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040485(15-benzyl-4-cyclopropylmethyl-10,17-dihydroxy-(1S,...)
Affinity DataKi:  10nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50297170(7-(2'-spiroindanyl)oxymorphone | 7-(Spiroindano)Ox...)
Affinity DataKi:  11nMAssay Description:selective binding affinity against mu opioid receptor, using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040485(15-benzyl-4-cyclopropylmethyl-10,17-dihydroxy-(1S,...)
Affinity DataKi:  13nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040487(17-(cyclopropylmethyl)4,5-alpha-epoxy-3,14-dihydro...)
Affinity DataKi:  13nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  14nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  14nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040482(17-(cyclopropylmethyl)-6,7-didehydro-4,5-alpha-epo...)
Affinity DataKi:  15nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040482(17-(cyclopropylmethyl)-6,7-didehydro-4,5-alpha-epo...)
Affinity DataKi:  25nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040483(4-cyclopropylmethyl-10,17-dihydroxy-15-phenyl-(1S,...)
Affinity DataKi:  25nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50038641(22-cyclopropylmethyl-(2R,13S)-14-oxa-4,22-diazahep...)
Affinity DataKi:  33nMAssay Description:Binding affinity against kappa-opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50056628(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-phenyl-(...)
Affinity DataKi:  66nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040482(17-(cyclopropylmethyl)-6,7-didehydro-4,5-alpha-epo...)
Affinity DataKi:  121nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  332nMAssay Description:Binding affinity against kappa-opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50297170(7-(2'-spiroindanyl)oxymorphone | 7-(Spiroindano)Ox...)
Affinity DataKi:  588nMAssay Description:selective binding affinity against kappa opioid receptor, using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50038642(22-methyl-(2R,13S)-14-oxa-4,22-diazaheptacyclo[13....)
Affinity DataIC50:  920nMAssay Description:Antagonist activity against mu-opioid receptor in guinea pig ileum in the presence of morphineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50038642(22-methyl-(2R,13S)-14-oxa-4,22-diazaheptacyclo[13....)
Affinity DataIC50:  990nMAssay Description:Antagonist activity against kappa-opioid receptor in guinea pig ileum in the presence of ethylketazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50038642(22-methyl-(2R,13S)-14-oxa-4,22-diazaheptacyclo[13....)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against delta-opioid receptor in mouse vas deferens in the presence of DADLEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity against kappa-opioid receptor in guinea pig ileum in the presence of ethylketazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBotulinum neurotoxin type A2 [1-425](Clostridium botulinum)
Absolute Science

LigandPNGBDBM23274((2E)-3-(2,4-dichlorophenyl)-N-hydroxyprop-2-enamid...)
Affinity DataIC50:  2.40E+3nMpH: 7.4 T: 2°CAssay Description:Reactions between recombinant BoNTA-LC and fluorescent peptide substrate were carried out in 96-well microplates. Reaction progress was measured cont...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A2 [1-425](Clostridium botulinum)
Absolute Science

LigandPNGBDBM28913(2-mercaptoacetamide, 12l | N-[3-(4-nitrophenyl)-1H...)
Affinity DataIC50:  2.90E+3nMpH: 7.4 T: 2°CAssay Description:Reactions between recombinant BoNTA-LC and fluorescent peptide substrate were carried out in 96-well microplates. Reaction progress was measured cont...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBotulinum neurotoxin type A2 [1-425](Clostridium botulinum)
Absolute Science

LigandPNGBDBM28906(2-mercaptoacetamide, 12a | N-[3-(4-chlorophenyl)-1...)
Affinity DataIC50:  4.80E+3nMpH: 7.4 T: 2°CAssay Description:Reactions between recombinant BoNTA-LC and fluorescent peptide substrate were carried out in 96-well microplates. Reaction progress was measured cont...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A2 [1-425](Clostridium botulinum)
Absolute Science

LigandPNGBDBM28917(2-mercaptoacetamide, 12g | N-[3-(3-chlorophenyl)-1...)
Affinity DataIC50:  5.60E+3nMpH: 7.4 T: 2°CAssay Description:Reactions between recombinant BoNTA-LC and fluorescent peptide substrate were carried out in 96-well microplates. Reaction progress was measured cont...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBotulinum neurotoxin type A2 [1-425](Clostridium botulinum)
Absolute Science

LigandPNGBDBM28911(2-mercaptoacetamide, 12i | N-[3-(4-bromophenyl)-1H...)
Affinity DataIC50:  6.60E+3nMpH: 7.4 T: 2°CAssay Description:Reactions between recombinant BoNTA-LC and fluorescent peptide substrate were carried out in 96-well microplates. Reaction progress was measured cont...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBotulinum neurotoxin type A2 [1-425](Clostridium botulinum)
Absolute Science

LigandPNGBDBM28918(2-mercaptoacetamide, 12f | 2-sulfanyl-N-{3-[2-(tri...)
Affinity DataIC50:  7.20E+3nMpH: 7.4 T: 2°CAssay Description:Reactions between recombinant BoNTA-LC and fluorescent peptide substrate were carried out in 96-well microplates. Reaction progress was measured cont...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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