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Found 305 with Last Name = 'muraoka' and Initial = 'o'
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50612995(CHEMBL5276586)
Affinity DataKi:  0.160nMAssay Description:Binding affinity to sucrase in rat small intestinal brush border membrane vesicles assessed as inhibition constant using sucrose as substrate incubat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50612998(CHEMBL5269400)
Affinity DataKi:  0.190nMAssay Description:Binding affinity to sucrase in rat small intestinal brush border membrane vesicles assessed as inhibition constant using sucrose as substrate incubat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50613001(CHEMBL5268739)
Affinity DataKi:  0.210nMAssay Description:Binding affinity to sucrase in rat small intestinal brush border membrane vesicles assessed as inhibition constant using sucrose as substrate incubat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50613004(CHEMBL5282029)
Affinity DataKi:  0.240nMAssay Description:Binding affinity to sucrase in rat small intestinal brush border membrane vesicles assessed as inhibition constant using sucrose as substrate incubat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50612994(CHEMBL5283777)
Affinity DataKi:  0.310nMAssay Description:Binding affinity to sucrase in rat small intestinal brush border membrane vesicles assessed as inhibition constant using sucrose as substrate incubat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50612995(CHEMBL5276586)
Affinity DataKi:  0.510nMAssay Description:Binding affinity to maltase in rat small intestinal brush border membrane vesicles assessed as inhibition constant using maltose as substrate incubat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50612998(CHEMBL5269400)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to maltase in rat small intestinal brush border membrane vesicles assessed as inhibition constant using maltose as substrate incubat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50613001(CHEMBL5268739)
Affinity DataKi:  0.690nMAssay Description:Binding affinity to maltase in rat small intestinal brush border membrane vesicles assessed as inhibition constant using maltose as substrate incubat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50613004(CHEMBL5282029)
Affinity DataKi:  0.770nMAssay Description:Binding affinity to maltase in rat small intestinal brush border membrane vesicles assessed as inhibition constant using maltose as substrate incubat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50612994(CHEMBL5283777)
Affinity DataKi:  0.840nMAssay Description:Binding affinity to maltase in rat small intestinal brush border membrane vesicles assessed as inhibition constant using maltose as substrate incubat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147013(CHEMBL3764559)
Affinity DataKi:  185nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147016(CHEMBL3763300)
Affinity DataKi:  210nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147107(CHEMBL3763319)
Affinity DataKi:  216nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147158(CHEMBL3764745)
Affinity DataKi:  353nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147159(CHEMBL3764813)
Affinity DataKi:  785nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180584(CHEMBL3814496)
Affinity DataIC50:  42nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50049730(2-(5-(2-methyl-3-phenylallylidene)-4-oxo-2-thioxot...)
Affinity DataIC50:  72nMAssay Description:Inhibition of rat lens aldose reductase using DL-glyceraldehyde as substrate after 30 mins by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180582(CHEMBL3814988)
Affinity DataIC50:  90nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180583(CHEMBL3815109)
Affinity DataIC50:  90nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50612995(CHEMBL5276586)
Affinity DataIC50:  100nMAssay Description:Inhibition of sucrase in rat small intestinal brush border membrane vesicles using sucrose as substrate incubated for 30 mins by glucose-oxidase meth...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50342937((1S,2R,3S,4S)-1-((2S,3S)-3-ethoxy-2,4-dihydroxybut...)
Affinity DataIC50:  120nMAssay Description:Inhibition of rat small intestinal sucrase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180520(CHEMBL3814838)
Affinity DataIC50:  120nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50342939((1S,2R,3S,4S)-1-((2S,3S)-3-(benzyloxy)-2,4-dihydro...)
Affinity DataIC50:  140nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180584(CHEMBL3814496)
Affinity DataIC50:  150nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)
Affinity DataIC50:  200nMAssay Description:Inhibition of sucrase in rat small intestinal brush border membrane vesicles using sucrose as substrate incubated for 30 mins by glucose-oxidase meth...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50612995(CHEMBL5276586)
Affinity DataIC50:  200nMAssay Description:Inhibition of maltase in rat small intestinal brush border membrane vesicles using maltose as substrate incubated for 30 mins by glucose-oxidase meth...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat small intestinal sucrase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147107(CHEMBL3763319)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147014(CHEMBL3764223)
Affinity DataIC50:  210nMAssay Description:Inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180584(CHEMBL3814496)
Affinity DataIC50:  210nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50612998(CHEMBL5269400)
Affinity DataIC50:  220nMAssay Description:Inhibition of sucrase in rat small intestinal brush border membrane vesicles using sucrose as substrate incubated for 30 mins by glucose-oxidase meth...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50612998(CHEMBL5269400)
Affinity DataIC50:  230nMAssay Description:Inhibition of maltase in rat small intestinal brush border membrane vesicles using maltose as substrate incubated for 30 mins by glucose-oxidase meth...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180580(CHEMBL3814911)
Affinity DataIC50:  240nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180580(CHEMBL3814911)
Affinity DataIC50:  250nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50342937((1S,2R,3S,4S)-1-((2S,3S)-3-ethoxy-2,4-dihydroxybut...)
Affinity DataIC50:  270nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147012(CHEMBL3763591)
Affinity DataIC50:  270nMAssay Description:Inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180520(CHEMBL3814838)
Affinity DataIC50:  270nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180583(CHEMBL3815109)
Affinity DataIC50:  280nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50338672(CHEMBL1209027 | Salaprinol)
Affinity DataIC50:  290nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50327501(CHEMBL1258528 | ponkoranol)
Affinity DataIC50:  290nMAssay Description:Inhibition of rat intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180586(CHEMBL1182462)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147008(CHEMBL3765363)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50612999(CHEMBL5277322)
Affinity DataIC50:  300nMAssay Description:Inhibition of sucrase in rat small intestinal brush border membrane vesicles using sucrose as substrate incubated for 30 mins by glucose-oxidase meth...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50338669(CHEMBL1684162 | Neosalacinol)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50338676(1,4-Dideoxy-1,4-{(R)-[(2S,3R,4R,5S)-2,3,4,5,6-pent...)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50338669(CHEMBL1684162 | Neosalacinol)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147013(CHEMBL3764559)
Affinity DataIC50:  320nMAssay Description:Inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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