Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.149nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.159nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.188nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.221nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.259nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:In vitro radioligand binding assay on Dopamine receptor D2 of rat striatum using [3H]- spiperoneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.288nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.312nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepineMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.350nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.435nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:In vitro radioligand binding assay on Dopamine receptor D2 of rat striatum using [3H]- spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:In vitro radioligand binding assay on Dopamine receptor D2 of rat striatum using [3H]- spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity of the compound was evaluated against Dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand; ND = Not determinedMore data for this Ligand-Target Pair
Affinity DataKi: 0.724nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.724nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.780nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.820nMAssay Description:Binding affinity for rat salivary gland muscarinic acetylcholine receptor M3 using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepineMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepineMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepineMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:In vitro radioligand binding assay on Dopamine receptor D2 of rat striatum using [3H]- spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepineMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:In vitro radioligand binding assay on Dopamine receptor D2 of rat striatum using [3H]- spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:In vitro radioligand binding assay on Dopamine receptor D2 of rat striatum using [3H]- spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepineMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity for rat salivary gland muscarinic acetylcholine receptor M3 using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 2.31nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 2.34nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 2.67nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 2.99nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 3.02nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 3.07nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:In vitro radioligand binding assay on Dopamine receptor D2 of rat striatum using [3H]- spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity for rat salivary gland muscarinic acetylcholine receptor M3 using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Binding affinity for rat salivary gland muscarinic acetylcholine receptor M3 using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Binding affinity for rat salivary gland muscarinic acetylcholine receptor M3 using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepineMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepineMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 4.04nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair