TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 9.70nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 83nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 88nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 94nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 127nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 157nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 201nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 252nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 277nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 397nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Competitive inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) assessed as formation of G6P by continuou...More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMAssay Description:Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair