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Found 44 with Last Name = 'nilius' and Initial = 'am'
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50409919(CHEMBL12282)
Affinity DataKi:  0.331nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50224090(CHEMBL410940)
Affinity DataKi:  0.851nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50224093(CHEMBL408925)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50224095(CHEMBL264043)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50423641(A-198401 | CHEMBL303274)
Affinity DataKi:  1.90nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50001560(CHEMBL273275)
Affinity DataKi:  3.90nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50224097(CHEMBL418067)
Affinity DataKi:  7.20nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50224091(CHEMBL442482)
Affinity DataKi:  7.60nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50224076(CHEMBL288534)
Affinity DataKi:  13nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50001566(CHEMBL275467)
Affinity DataKi:  19nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50224094(CHEMBL418256)
Affinity DataKi:  19nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50001573(CHEMBL273387)
Affinity DataKi:  22nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50224092(CHEMBL216252)
Affinity DataKi:  28nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50224044(CHEMBL288396)
Affinity DataKi:  79nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50224096(CHEMBL40743)
Affinity DataKi:  191nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50224098(CHEMBL384920)
Affinity DataKi:  204nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50068561((16E,24E,26E,28E)-1,18-Dihydroxy-12-[2-(4-hydroxy-...)
Affinity DataIC50:  1.60nMAssay Description:The compound was tested for binding afifnity to FK506 binding protein 12 with an ascomycin conjugate of alkaline phosphatase in a competition binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50089437(CHEMBL437064 | Rapamycin analogue)
Affinity DataIC50:  2.10nMAssay Description:The compound was tested for binding afifnity to FK506 binding protein 12 using Rapamycin as control, with an ascomycin conjugate of alkaline phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50089447(CHEMBL281297 | Rapamycin analogue)
Affinity DataIC50:  14nMAssay Description:The compound was tested for binding afifnity to FK506 binding protein 12 using Rapamycin as control, with an ascomycin conjugate of alkaline phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50089432(1,18-dihydroxy-19,30-dimethoxy-12-{2-[3-methoxy-4-...)
Affinity DataIC50: >1.00E+3nMAssay Description:The compound was tested for binding afifnity to FK506 binding protein 12 using Rapamycin as control, with an ascomycin conjugate of alkaline phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50089429(4-[2-(1,18-dihydroxy-19,30-dimethoxy-15,17,21,23,2...)
Affinity DataIC50: >1.00E+3nMAssay Description:The compound was tested for binding afifnity to FK506 binding protein 12 using Rapamycin as control, with an ascomycin conjugate of alkaline phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000090(CHEMBL66729)
Affinity DataIC50: <9.40E+3nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000089(CHEMBL69983)
Affinity DataIC50: <9.40E+3nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116067((Linezolid)N-[3-(3-Fluoro-4-morpholin-4-yl-phenyl)...)
Affinity DataIC50:  1.70E+4nMAssay Description:Compound was evaluated for inhibition of Mono aminoxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116058(4-((Z)-2-{4-[(S)-5-(Acetylamino-methyl)-2-oxo-oxaz...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116059(CHEMBL63456 | N-{(S)-3-[3-Fluoro-4-((E)-2-pyridin-...)
Affinity DataIC50:  5.90E+4nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116051(CHEMBL69528 | N-{(S)-3-[3-Fluoro-4-((Z)-2-fluoro-2...)
Affinity DataIC50:  9.80E+4nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116062(CHEMBL67796 | N-{(S)-3-[4-((Z)-2-Bromo-2-pyridin-3...)
Affinity DataIC50:  1.21E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116072(CHEMBL68290 | N-((S)-3-{4-[(Z)-2-Bromo-2-(3-cyano-...)
Affinity DataIC50: >1.50E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116052(CHEMBL67288 | N-((S)-3-{4-[(Z)-2-Bromo-2-(4-cyano-...)
Affinity DataIC50: >1.50E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116057(CHEMBL67481 | N-((S)-3-{4-[(Z)-2-Bromo-2-(2-cyano-...)
Affinity DataIC50: >1.50E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116070(CHEMBL69609 | N-((S)-3-{4-[(Z)-2-Bromo-2-(3-hydrox...)
Affinity DataIC50: >1.50E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116071(CHEMBL65595 | N-{(S)-3-[4-((Z)-2-Bromo-2-pyridin-4...)
Affinity DataIC50:  1.86E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116053(CHEMBL66269 | N-((S)-3-{4-[(Z)-2-(5-Cyano-thiophen...)
Affinity DataIC50:  2.85E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116068(CHEMBL303675 | N-((S)-3-{4-[(E)-2-(5-Cyano-pyridin...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116065(CHEMBL308441 | N-((S)-3-{3-Fluoro-4-[(Z)-2-fluoro-...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116064(CHEMBL66571 | N-((S)-3-{3-Fluoro-4-[(Z)-2-fluoro-2...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116055(3-((Z)-2-{4-[(S)-5-(Acetylamino-methyl)-2-oxo-oxaz...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116061(CHEMBL68078 | N-((S)-3-{4-[(Z)-2-(3-Cyano-phenyl)-...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116054(CHEMBL67688 | N-((S)-3-{4-[(Z)-2-(3-Acetyl-phenyl)...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116056(CHEMBL428699 | N-((S)-3-{4-[(Z)-2-Bromo-2-(3-formy...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116063(CHEMBL69975 | N-((S)-3-{4-[(Z)-2-Bromo-2-(5-cyano-...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116066(CHEMBL69166 | N-((S)-3-{4-[(Z)-2-(5-Cyano-pyridin-...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50116073(CHEMBL68180 | N-{(S)-3-[3-Fluoro-4-((Z)-2-fluoro-2...)
Affinity DataIC50:  4.75E+5nMAssay Description:Inhibition of Monoamine oxidase B in rat primary hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed