Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 9.80E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 1.10E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 1.50E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 1.60E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 1.80E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 1.90E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 2.10E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 3.80E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-inhibitor complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 5.80E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate-inhibitor complex state after 30 mins by fluorescence assa...More data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 7.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-inhibitor complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 9.90E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-inhibitor complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 1.25E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate-inhibitor complex state after 30 mins by fluorescence assa...More data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 2.60E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-inhibitor complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 4.34E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate-inhibitor complex state after 30 mins by fluorescence assa...More data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 5.18E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate-inhibitor complex state after 30 mins by fluorescence assa...More data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 5.63E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate-inhibitor complex state after 30 mins by fluorescence assa...More data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 5.72E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate-inhibitor complex state after 30 mins by fluorescence assa...More data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 7.23E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate-inhibitor complex state after 30 mins by fluorescence assa...More data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 8.32E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-inhibitor complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 8.32E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-inhibitor complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate-inhibitor complex state after 30 mins by fluorescence assa...More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of recombinant human NaV1.7 alpha subunit expressed in HEK293 cells at -65 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibition of recombinant human NaV1.7 alpha subunit expressed in HEK293 cells at -65 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibition of recombinant human NaV1.7 alpha subunit expressed in HEK293 cells at -65 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Inhibition of recombinant human NaV1.7 alpha subunit expressed in HEK293 cells at -65 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Inhibition of recombinant human NaV1.7 alpha subunit expressed in HEK293 cells at -65 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
Affinity DataIC50: 73nMAssay Description:Inhibition of recombinant human NaV1.7 alpha subunit expressed in HEK293 cells at -65 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of recombinant rat NaV1.7 alpha subunit expressed in HEK293 cells at -65 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of recombinant rat NaV1.7 alpha subunit expressed in HEK293 cells at -65 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant human NaV1.7 alpha subunit expressed in HEK293 cells at -90 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant human NaV1.7 alpha subunit expressed in HEK293 cells at -90 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Inhibition of recombinant human NaV1.7 alpha subunit expressed in HEK293 cells at -65 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:Inhibition of recombinant human NaV1.7 alpha subunit expressed in HEK293 cells at -65 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Inhibition of recombinant human NaV1.7 alpha subunit expressed in HEK293 cells at -65 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Inhibition of recombinant human NaV1.7 alpha subunit expressed in HEK293 cells at -65 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Inhibition of recombinant human NaV1.7 alpha subunit expressed in HEK293 cells at -65 mV holding potential by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair