Compile Data Set for Download or QSAR
maximum 50k data
Found 235 with Last Name = 'ninomiya' and Initial = 'k'
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227831(CHEMBL52242)
Affinity DataKi:  1.20nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227791(CHEMBL53815)
Affinity DataKi:  4.60nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227978(CHEMBL53316)
Affinity DataKi:  6.30nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50228190(CHEMBL54263)
Affinity DataKi:  9.80nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227787(CHEMBL1743933)
Affinity DataKi:  13nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227837(CHEMBL52131)
Affinity DataKi:  14nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50093789(CHEMBL541829 | Succinic acid mono-(2-dimethylamino...)
Affinity DataKi:  18nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227788(CHEMBL1743936)
Affinity DataKi:  23nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227974(CHEMBL298554)
Affinity DataKi:  26nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227976(CHEMBL299389)
Affinity DataKi:  38nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227653(CHEMBL299207)
Affinity DataKi:  41nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227977(CHEMBL300631)
Affinity DataKi:  68nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227790(CHEMBL53344)
Affinity DataKi:  71nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227789(CHEMBL412653)
Affinity DataKi:  75nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataKi:  190nMAssay Description:Inhibition of recombinant human maltase-glucoamylase using p-nitrophenyl-alpha-D-glucopyranoside as substrate incubated for 35 mins by microtiter pla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227832(CHEMBL54101)
Affinity DataKi:  198nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50228189(CHEMBL52710)
Affinity DataKi:  416nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50228052(CHEMBL52982)
Affinity DataKi:  517nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50549692(CHEMBL4749306)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of recombinant human maltase-glucoamylase using p-nitrophenyl-alpha-D-glucopyranoside as substrate incubated for 35 mins by microtiter pla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50549691(CHEMBL4754034)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of recombinant human maltase-glucoamylase using p-nitrophenyl-alpha-D-glucopyranoside as substrate incubated for 35 mins by microtiter pla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50549693(CHEMBL4750690)
Affinity DataKi:  5.10E+4nMAssay Description:Inhibition of recombinant human maltase-glucoamylase using p-nitrophenyl-alpha-D-glucopyranoside as substrate incubated for 35 mins by microtiter pla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227831(CHEMBL52242)
Affinity DataIC50:  13nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227791(CHEMBL53815)
Affinity DataIC50:  34nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180584(CHEMBL3814496)
Affinity DataIC50:  42nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50093789(CHEMBL541829 | Succinic acid mono-(2-dimethylamino...)
Affinity DataIC50:  51nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227788(CHEMBL1743936)
Affinity DataIC50:  54nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227837(CHEMBL52131)
Affinity DataIC50:  55nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227787(CHEMBL1743933)
Affinity DataIC50:  62nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50049730(2-(5-(2-methyl-3-phenylallylidene)-4-oxo-2-thioxot...)
Affinity DataIC50:  72nMAssay Description:Inhibition of rat lens aldose reductase using DL-glyceraldehyde as substrate after 30 mins by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180583(CHEMBL3815109)
Affinity DataIC50:  90nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180582(CHEMBL3814988)
Affinity DataIC50:  90nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227978(CHEMBL53316)
Affinity DataIC50:  96nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50228190(CHEMBL54263)
Affinity DataIC50:  115nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180520(CHEMBL3814838)
Affinity DataIC50:  120nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50342937((1S,2R,3S,4S)-1-((2S,3S)-3-ethoxy-2,4-dihydroxybut...)
Affinity DataIC50:  120nMAssay Description:Inhibition of rat small intestinal sucrase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227653(CHEMBL299207)
Affinity DataIC50:  133nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50342939((1S,2R,3S,4S)-1-((2S,3S)-3-(benzyloxy)-2,4-dihydro...)
Affinity DataIC50:  140nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180584(CHEMBL3814496)
Affinity DataIC50:  150nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227789(CHEMBL412653)
Affinity DataIC50:  152nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227790(CHEMBL53344)
Affinity DataIC50:  157nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat small intestinal sucrase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180584(CHEMBL3814496)
Affinity DataIC50:  210nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180580(CHEMBL3814911)
Affinity DataIC50:  240nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180580(CHEMBL3814911)
Affinity DataIC50:  250nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50342937((1S,2R,3S,4S)-1-((2S,3S)-3-ethoxy-2,4-dihydroxybut...)
Affinity DataIC50:  270nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180520(CHEMBL3814838)
Affinity DataIC50:  270nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180583(CHEMBL3815109)
Affinity DataIC50:  280nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50327501(CHEMBL1258528 | ponkoranol)
Affinity DataIC50:  290nMAssay Description:Inhibition of rat intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180586(CHEMBL1182462)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 235 total ) | Next | Last >>
Jump to: