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Found 1310 with Last Name = 'ono' and Initial = 'y'
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50165949(C-Phenyl-N-{3-[2-((S)-5-phenyl-4-phenyl-oxazol-2-y...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of [3H]-PGE-2 binding to human prostanoid EP4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010652(CHEMBL3264742)
Affinity DataKi:  0.313nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010658(CHEMBL3264747)
Affinity DataKi:  0.534nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50165945(CHEMBL371394 | N-Benzyloxy-3-[(S)-2-(4,5-diphenyl-...)
Affinity DataKi:  0.680nMAssay Description:Inhibition of [3H]-PGE-2 binding to human prostanoid EP4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50165949(C-Phenyl-N-{3-[2-((S)-5-phenyl-4-phenyl-oxazol-2-y...)
Affinity DataKi:  0.740nMAssay Description:Inhibition of rat prostanoid EP4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50165948(6-{(S)-2-[(Benzofuran-2-carbonyl)-amino]-5-benzylo...)
Affinity DataKi:  0.910nMAssay Description:Inhibition of [3H]-PGE-2 binding to human prostanoid EP4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50039029((+)-4-((alpha R)-((2S,5R)-4-allyl-2,5-dimethylpipe...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010659(CHEMBL3264748)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010656(CHEMBL3264745)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010658(CHEMBL3264747)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010659(CHEMBL3264748)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010659(CHEMBL3264748)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010653(CHEMBL3264743)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010657(CHEMBL3264746)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010652(CHEMBL3264742)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi Pharmaceutical Research Center

Curated by ChEMBL
LigandPNGBDBM50570460(CHEMBL4854629)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]-JNJ962 from BACE1 (unknown origin) expressed in HEK293 cell membrane assessed as inhibition constant by scintillation counting a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010658(CHEMBL3264747)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50165948(6-{(S)-2-[(Benzofuran-2-carbonyl)-amino]-5-benzylo...)
Affinity DataKi:  5.10nMAssay Description:Inhibition of rat prostanoid EP4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010652(CHEMBL3264742)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50165946(3-[(S)-2-(4,5-Diphenyl-oxazol-2-yl)-cyclohex-2-eny...)
Affinity DataKi:  5.5nMAssay Description:Inhibition of [3H]-PGE-2 binding to human prostanoid EP4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010654(CHEMBL3264744)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50165951(6-{(S)-2-[(Benzofuran-2-carbonyl)-amino]-6-benzylo...)
Affinity DataKi:  8.40nMAssay Description:Inhibition of [3H]-PGE-2 binding to human prostanoid EP4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613290(CHEMBL5271484)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-Angiotensin II from Angiotensin II type-1 receptor in VSMC cells (unknown origin) assessed as inhibition constant by competiti...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613288(CHEMBL5272962)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-Angiotensin II from Angiotensin II type-1 receptor in VSMC cells (unknown origin) assessed as inhibition constant by competiti...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-Angiotensin II from Angiotensin II type-1 receptor in VSMC cells (unknown origin) assessed as inhibition constant by competiti...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute Of Organic Synthesis

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]DTG from sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272503((2R,3S)-3-Methyl-2-phenylmethanesulfonylamino-pent...)
Affinity DataKi:  15nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613289(CHEMBL5271135)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]-Angiotensin II from Angiotensin II type-1 receptor in VSMC cells (unknown origin) assessed as inhibition constant by competiti...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272558(4-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  17nMAssay Description:Inhibition of human factor 11aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272539(3-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  18nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272576(3-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  20nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613294(CHEMBL5271903)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]-Angiotensin II from Angiotensin II type-1 receptor in VSMC cells (unknown origin) assessed as inhibition constant by competiti...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613286(CHEMBL5273768)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]-Angiotensin II from Angiotensin II type-1 receptor in VSMC cells (unknown origin) assessed as inhibition constant by competiti...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010653(CHEMBL3264743)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613291(CHEMBL5282200)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]-Angiotensin II from Angiotensin II type-1 receptor in VSMC cells (unknown origin) assessed as inhibition constant by competiti...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272480((S)-2-((2R,3S)-3-Methyl-2-phenylmethanesulfonylami...)
Affinity DataKi:  25nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613293(CHEMBL5277518)
Affinity DataKi:  25nMAssay Description:Displacement of [125I]-Angiotensin II from Angiotensin II type-1 receptor in VSMC cells (unknown origin) assessed as inhibition constant by competiti...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613296(CHEMBL5289070)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]-Angiotensin II from Angiotensin II type-1 receptor in VSMC cells (unknown origin) assessed as inhibition constant by competiti...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613287(CHEMBL5275739)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]-Angiotensin II from Angiotensin II type-1 receptor in VSMC cells (unknown origin) assessed as inhibition constant by competiti...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613292(CHEMBL5287876)
Affinity DataKi:  29nMAssay Description:Displacement of [125I]-Angiotensin II from Angiotensin II type-1 receptor in VSMC cells (unknown origin) assessed as inhibition constant by competiti...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272560(3-({(1S,2R)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  30nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613295(CHEMBL5276125)
Affinity DataKi:  31nMAssay Description:Displacement of [125I]-Angiotensin II from Angiotensin II type-1 receptor in VSMC cells (unknown origin) assessed as inhibition constant by competiti...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613297(CHEMBL5283862)
Affinity DataKi:  31nMAssay Description:Displacement of [125I]-Angiotensin II from Angiotensin II type-1 receptor in VSMC cells (unknown origin) assessed as inhibition constant by competiti...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272539(3-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  33nMAssay Description:Inhibition of human factor 11aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272558(4-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  35nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272502((2R,3S)-3-Methyl-2-(propane-1-sulfonylamino)-penta...)
Affinity DataKi:  35nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272537((2R,3R)-N-[(S)-1-(4-Carbamimidoyl-benzylcarbamoyl)...)
Affinity DataKi:  42nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50165943((S)-2-{(S)-5-Benzyloxycarbonylamino-2-[(1H-indole-...)
Affinity DataKi:  43nMAssay Description:Inhibition of [3H]-PGE-2 binding to human prostanoid EP4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272538(2-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  43nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010657(CHEMBL3264746)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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