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Found 1510 with Last Name = 'peng' and Initial = 'h'
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Barrow Neurological Institute

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0120nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312599(CHEMBL1093735 | N-Cyclohexyl-4-[(2,4-dichloropheny...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312599(CHEMBL1093735 | N-Cyclohexyl-4-[(2,4-dichloropheny...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cells pretreated for 10 mins measured after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312597(CHEMBL1093377 | N-Cyclohexyl-4-[(2,4-dichloropheny...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50355892(CHEMBL1910035)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cells pretreated for 10 mins measured after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156616((7RS,9aRS)-5-[7-(3-fluoro-phenoxymethyl)-octahydro...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50242582(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-c...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Barrow Neurological Institute

Curated by PDSP Ki Database
LigandPNGBDBM86311(CAS_485-35-8 | Cytisine | Cytisine-(-) | NSC_22407...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156605((7RS,9aRS)-2-furan-2-yl-5-(7-imidazol-1-ylmethyloc...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156595((7RS,9aRS)-2-furan-2-yl-N5-(2-pyrimidin-2-yloctahy...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156606((7RS,9aRS)-2-furan-2-yl-5-[7-(pyridin-3-yloxymethy...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156646(2-(furan-2-yl)-5-((7S,9aS)-7-((quinolin-6-yloxy)me...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  0.740nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156638((7RS,9aRS)-5-[7-(2-fluoro-phenoxymethyl)-octahydro...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312602(CHEMBL1091814 | N-cyclohexyl-4-[(2,4-dichloropheny...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50355891(CHEMBL1910034)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cells pretreated for 10 mins measured after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312603(CHEMBL1084429 | N-cyclohexyl-4-{(2,4-dichloropheny...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312596(4-[(2,4-Dichlorophenyl)(phenyl)methyl]-N-piperidin...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312582(CHEMBL1088728 | N-Cyclohexyl-4-[(2,4-dichloropheny...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312586(4-[(4-bromo-2-fluorophenyl)(phenyl)methyl]-N-cyclo...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Barrow Neurological Institute

Curated by PDSP Ki Database
LigandPNGBDBM50047021(2-(6-(2-hydroxy-2-phenylethyl)-1-methylpiperidin-2...)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Barrow Neurological Institute

Curated by PDSP Ki Database
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156650(5-((7R,9aS)-7-((bis(pyridin-3-ylmethyl)amino)methy...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156635(5-((7S,9aS)-7-(aminomethyl)-hexahydro-1H-pyrido[1,...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156660(5-((7R,9aS)-7-((2,4-difluorobenzylamino)methyl)-he...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312585(CHEMBL1087250 | N-cyclohexyl-4-[(2,6-dichloropheny...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312598(4-[(3-chlorophenyl)(2,4-dichlorophenyl)methyl]-N-c...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312604(CHEMBL1084695 | N-cyclohexyl-4-[(2,4-dichloropheny...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312601(CHEMBL1091813 | N-cyclohexyl-4-[(2,4-dichloropheny...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156644((7RS,9aRS)-5-{7-[(bispyridin-4-ylmethylamino)-meth...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312600(4-[(2,4-Dichlorophenyl)(p-tolyl)methyl]-N-piperidi...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156662((6RS,9aRS)-[2-(7-amino-2-furan-2-yl[1,2,4]triazolo...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312588(4-[(2-fluoro-4-chlorophenyl)(phenyl)methyl]-N-cycl...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156604(CHEMBL173672 | N*5*-[(R)-1-(2,6-Difluoro-benzyl)-p...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156624(5-((7S,9aS)-7-((bis(pyridin-3-ylmethyl)amino)methy...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156652((7RS,9aRS)-2-furan-2-yl-5-(7-[1,2,4]triazol-1-ylme...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156640((7RS,9aRS)-5-[7-(3-fluoro-phenoxymethyl)-octahydro...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50370922(CHEMBL1237041)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312591(1-(Cyclohexylcarbonyl)-4-[(2,4-dichlorophenyl)(phe...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312592(1-(1-adamantylcarbonyl)-4-[(2,4-dichlorophenyl)(ph...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312584(CHEMBL1087874 | N-cyclohexyl-4-((2,5-dichloropheny...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156633((7RS,9aRS)-2-furan-2-yl-5-[7-(isoquinolin-5-yloxym...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156643(2-(furan-2-yl)-5-((7R,9aS)-7-((quinolin-2-yloxy)me...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50312587(4-[(2-chloro-4-fluorophenyl)(phenyl)methyl]-N-cycl...)
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156618((7RS,9aRS)-2-furan-2-yl-5-[7-(pyrimidin-2-ylaminom...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156667(5-((7R,9aS)-7-((bis(pyridin-2-ylmethyl)amino)methy...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156621((+/-)-2-furan-2-yl-5-(octahydropyrido[1,2-a]pyrazi...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Barrow Neurological Institute

Curated by PDSP Ki Database
LigandPNGBDBM85207(CAS_123990 | NSC_123990 | Suberyldicholine)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50156599((6RS,9aRS)-2-furan-2-yl-5-(6-phenoxymethyl-octahyd...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50151188(5-(4-((5-chloro-1-methyl-3-(trifluoromethyl)-1H-py...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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