TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of Maryland
Curated by ChEMBL
University Of Maryland
Curated by ChEMBL
Affinity DataIC50: 3.70nMAssay Description:Blockade of Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human full length (His)6-tagged Pim-3 expressed in insect Sf21 cells using RSRHSSYPAGT as substrate measured for 30 mins by [gamma-33P]...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of human full length (His)6-tagged Pim-1 expressed in insect Sf21 cells using RSRHSSYPAGT as substrate measured for 30 mins by [gamma-33P]...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of human full length GST-tagged Pim-2 expressed in Escherichia coli using RSRHSSYPAGT as substrate measured for 30 mins by [gamma-33P]ATP-...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Inhibition of human recombinant CDK5/p25 using Histone H1 and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of human recombinant CDK5/p25 using Histone H1 and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 810nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 850nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 850nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 870nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using Histone H1 and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using Histone H1 and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair