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Found 214 with Last Name = 'prachayasittikul' and Initial = 'v'
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279582(CHEMBL488769 | N-[(1S,2S,4R,5R)-5-Guanidino-4-(4-g...)
Affinity DataKi:  6nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279584(CHEMBL485694 | N-[(1S,2S,4R,5R)-5-Guanidino-2,4-bi...)
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279581(CHEMBL522615 | N-[(1S,2S,4R,5R)-2-(2-Amino-4-guani...)
Affinity DataKi:  22nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279605(CHEMBL487946 | N-[(1S,2S,4R,5R)-5-Guanidino-2,4-bi...)
Affinity DataKi:  42nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279606(1-[(1R,2R,4S,5S)-2,4-bis(4-carbamimidamidophenoxy)...)
Affinity DataKi:  46nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279583(CHEMBL505581 | N-[(1S,2S,4R,5R)-5-Guanidino-2,4-bi...)
Affinity DataKi:  69nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279559(CHEMBL490273 | N-{4-[(1S,2S,4R,5R)-2,4-Diguanidino...)
Affinity DataKi:  89nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50241035(1-[(1R,2R,4S,5S)-5-carbamimidamido-2,4-bis(2,4-dic...)
Affinity DataKi:  169nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279560(CHEMBL448513 | N-{4-[(1S,2S,4R,5R)-2,4-Diguanidino...)
Affinity DataKi:  404nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279607(1-[(1R,2R,4S,5S)-5-[(4-carbamimidamidonaphthalen-1...)
Affinity DataKi:  423nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279608((1S,2S,4R,5R)-2,4-dicarbamimidamido-5-{[(4-carbami...)
Affinity DataKi:  812nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279609((1S,2S,4R,5R)-2,4-dicarbamimidamido-5-{[(3-carbami...)
Affinity DataKi:  1.77E+3nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279612(CHEMBL519572 | N-[(1S,2S,4R,5R)-5-Guanidino-2,4-bi...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279634(1,1'-((1R,3S,4S,6R)-4,6-bis(2-amino-1H-benzo[d]imi...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279636((1R,3S,4S,6R)-4,6-diguanidinocyclohexane-1,3-diyl ...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279635(1,1'-((1R,3S,4S,6R)-4,6-bis(pyridin-2-yloxy)cycloh...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279610(CHEMBL487131 | N-[(1S,2S,4R,5R)-5-Guanidino-2,4-bi...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50279611(CHEMBL487333 | N-[(1S,2S,4R,5R)-5-Guanidino-2,4-bi...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of human recombinant furin-dependent anthrax protective antigen processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of CYP19 (unknown origin) using O-benzyl fluorescein benzyl ester substrate preincubated for 10 mins by fluorimetric analysis relative to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of CYP19 (unknown origin) using O-benzyl fluorescein benzyl ester substrate preincubated for 10 mins by fluorimetric analysis relative to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515597(CHEMBL4460718)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515597(CHEMBL4460718)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515582(CHEMBL4590541)
Affinity DataIC50:  60nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515582(CHEMBL4590541)
Affinity DataIC50:  60nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515580(CHEMBL4449929)
Affinity DataIC50:  130nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515580(CHEMBL4449929)
Affinity DataIC50:  130nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515583(CHEMBL4444996)
Affinity DataIC50:  160nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515583(CHEMBL4444996)
Affinity DataIC50:  160nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50094259(CHEMBL3589965)
Affinity DataIC50:  200nMAssay Description:Inhibition of CYP19 (unknown origin) using O-benzyl fluorescein benzyl ester substrate preincubated for 10 mins by fluorimetric analysis relative to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50094259(CHEMBL3589965)
Affinity DataIC50:  200nMAssay Description:Inhibition of CYP19 (unknown origin) using O-benzyl fluorescein benzyl ester substrate preincubated for 10 mins by fluorimetric analysis relative to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515581(CHEMBL4462178)
Affinity DataIC50:  210nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515581(CHEMBL4462178)
Affinity DataIC50:  210nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515578(CHEMBL4567479)
Affinity DataIC50:  280nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515578(CHEMBL4567479)
Affinity DataIC50:  280nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515589(CHEMBL4570681)
Affinity DataIC50:  370nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515589(CHEMBL4570681)
Affinity DataIC50:  370nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515579(CHEMBL4556427)
Affinity DataIC50:  430nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515579(CHEMBL4556427)
Affinity DataIC50:  430nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515595(CHEMBL4543747)
Affinity DataIC50:  530nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515595(CHEMBL4543747)
Affinity DataIC50:  530nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515586(CHEMBL4527809)
Affinity DataIC50:  660nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515586(CHEMBL4527809)
Affinity DataIC50:  660nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284238(CHEMBL4173941)
Affinity DataIC50:  700nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284238(CHEMBL4173941)
Affinity DataIC50:  700nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515587(CHEMBL4446561)
Affinity DataIC50:  780nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50515587(CHEMBL4446561)
Affinity DataIC50:  780nMAssay Description:Inhibition of recombinant human aromatase expressed in baculovirus infected insect cells using O-benzyl fluorescein benzyl ester as substrate in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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